(Q42578482)

3 November 2017

Evaluating modulators of "Regulator of G-protein Signaling" (RGS) proteins (English)

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3 November 2017

4

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3 November 2017

Dustin E Bosch

1

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3 November 2017

Thomas Zielinski

series ordinal

2

1 reference

3 November 2017

Robert G Lowery

series ordinal

3

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3 November 2017

1 March 2012

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Current protocols in pharmacology

3 November 2017

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3 November 2017

Chapter 2

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3 November 2017

Unit2.8

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Regulators of G-protein signaling and their Gα substrates: promises and challenges in their use as drug discovery targets

3 November 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

Two Galpha(i1) rate-modifying mutations act in concert to allow receptor-independent, steady-state measurements of RGS protein activity

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

Heterotrimeric G protein activation by G-protein-coupled receptors

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

The RGS protein inhibitor CCG-4986 is a covalent modifier of the RGS4 Galpha-interaction face

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

Assays of RGS protein modulation by phosphatidylinositides and calmodulin

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

Allosteric regulation of GAP activity by phospholipids in regulators of G-protein signaling

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

Fluorescence-based assays for RGS box function

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

RGS12 and RGS14 GoLoco motifs are G alpha(i) interaction sites with guanine nucleotide dissociation inhibitor Activity

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

The regulators of G protein signaling (RGS) domains of RGS4, RGS10, and GAIP retain GTPase activating protein activity in vitro

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

GAIP and RGS4 are GTPase-activating proteins for the Gi subfamily of G protein alpha subunits

28 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3306263

10.1002/0471141755.PH0208S56

28 May 2018

Identifiers

DOI

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3 November 2017

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3 November 2017

PubMed publication ID

22382998

1 reference