(Q42664010)

4 November 2017

GABA(A) receptor beta 2 Tyr97 and Leu99 line the GABA-binding site. Insights into mechanisms of agonist and antagonist actions (English)

1 reference

4 November 2017

Andrew J Boileau

1

1 reference

4 November 2017

J Glen Newell

series ordinal

2

1 reference

4 November 2017

Cynthia Czajkowski

series ordinal

3

1 reference

4 November 2017

language of work or name

English

0 references

publication date

15 November 2001

1 reference

Journal of Biological Chemistry

4 November 2017

1 reference

4 November 2017

277

1 reference

4 November 2017

4

1 reference

4 November 2017

2931-2937

1 reference

Sequence and functional expression of the GABA A receptor shows a ligand-gated receptor super-family.

4 November 2017

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Ligand-gated ion channels in the brain: the amino acid receptor superfamily

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Chloride Channel Expression with the Tandem Construct of α6-β2 GABAA Receptor Subunit Requires a Monomeric Subunit of α6 or γ2

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Stoichiometry of a ligand-gated ion channel determined by fluorescence energy transfer

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Functional domains of GABAA receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Arginine residue 120 of the human GABAA receptor alpha 1, subunit is essential for GABA binding and chloride ion current gating

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

GABAA receptor needs two homologous domains of the beta-subunit for activation by GABA but not by pentobarbital.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

The major site of photoaffinity labeling of the gamma-aminobutyric acid type A receptor by [3H]flunitrazepam is histidine 102 of the alpha subunit.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Amino acids of the Torpedo marmorata acetylcholine receptor alpha subunit labeled by a photoaffinity ligand for the acetylcholine binding site

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Mapping the agonist binding site of the nicotinic acetylcholine receptor. Orientation requirements for activation by covalent agonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Preservation and staining of myelinated nerve fibers.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

NMDAR channel segments forming the extracellular vestibule inferred from the accessibility of substituted cysteines.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Identification of acetylcholine receptor channel-lining residues in the M1 segment of the alpha-subunit.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

The fourth transmembrane segment of the dopamine D2 receptor: accessibility in the binding-site crevice and position in the transmembrane bundle

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Architecture of Ca(2+) channel pore-lining segments revealed by covalent modification of substituted cysteines.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Cysteine mutagenesis reveals novel structure-function features within the predicted third extracellular loop of the type IIa Na(+)/P(i) cotransporter

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Identification of acetylcholine receptor channel-lining residues in the entire M2 segment of the alpha subunit.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Identification of channel-lining residues in the M2 membrane-spanning segment of the GABA(A) receptor alpha1 subunit

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Negatively charged amino acid residues in the nicotinic receptor delta subunit that contribute to the binding of acetylcholine

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Crystal structure of an ACh-binding protein reveals the ligand-binding domain of nicotinic receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

A general method of in vitro preparation and specific mutagenesis of DNA fragments: study of protein and DNA interactions

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Subunit stoichiometry of a mammalian K+ channel determined by construction of multimeric cDNAs.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Potassium currents expressed from Drosophila and mouse eag cDNAs in Xenopus oocytes.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Protein engineering and the study of structure--function relationships in receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Binding, gating, affinity and efficacy: the interpretation of structure-activity relationships for agonists and of the effects of mutating receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

An arylaminopyridazine derivative of gamma-aminobutyric acid (GABA) is a selective and competitive antagonist at the GABAA receptor site

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

The differential antagonism by bicuculline and SR95531 of pentobarbitone-induced currents in cultured hippocampal neurons.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Mechanisms for activation and antagonism of an AMPA-sensitive glutamate receptor: crystal structures of the GluR2 ligand binding core

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Two novel residues in M2 of the gamma-aminobutyric acid type A receptor affecting gating by GABA and picrotoxin affinity.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Nature of the 5' residue in the M2 domain affects function of the human alpha 1 beta 1 GABAA receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

Analysis of the ligand binding site of the 5-HT3 receptor using site directed mutagenesis: importance of glutamate 106.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M109334200

21 January 2018

Identifiers

DOI

10.1074/JBC.M109334200

1 reference

4 November 2017

1 reference