(Q42727402)

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Synthesis, structure-affinity relationships, and modeling of AMDA analogs at 5-HT2A and H1 receptors: structural factors contributing to selectivity.

scientific article published on 13 August 2009

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scholarly article

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19700330%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

Synthesis, structure-affinity relationships, and modeling of AMDA analogs at 5-HT2A and H1 receptors: structural factors contributing to selectivity (English)

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19700330%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

Glen E. Kellogg

4

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6 February 2020

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Jitesh R Shah

1

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6 February 2020

Philip D Mosier

2

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6 February 2020

Bryan L Roth

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6 February 2020

Richard B Westkaemper

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6 February 2020

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13 August 2009

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6 February 2020

Bioorganic & Medicinal Chemistry

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6 February 2020

17

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6 February 2020

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6 February 2020

6496-6504

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27 May 2018

Potential modes of interaction of 9-aminomethyl-9,10-dihydroanthracene (AMDA) derivatives with the 5-HT2A receptor: a ligand structure-affinity relationship, receptor mutagenesis and receptor modeling investigation

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Exploring the relationship between binding modes of 9-(aminomethyl)-9,10-dihydroanthracene and cyproheptadine analogues at the 5-HT2A serotonin receptor

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Mutational analysis of the antagonist-binding site of the histamine H(1) receptor

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9-(Aminomethyl)-9,10-dihydroanthracene is a novel and unlikely 5-HT2A receptor antagonist

1 reference

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Identifiers

10.1016/J.BMC.2009.08.016

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Europe PubMed Central

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6 February 2020

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Europe PubMed Central

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6 February 2020

PubMed publication ID

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19700330%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

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