(Q42910400)

English

Binding kinetics of darunavir to human immunodeficiency virus type 1 protease explain the potent antiviral activity and high genetic barrier

scientific article published on 10 October 2007

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Binding kinetics of darunavir to human immunodeficiency virus type 1 protease explain the potent antiviral activity and high genetic barrier (English)

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

1 reference

based on heuristic

inferred from title

author name string

Inge Dierynck

1

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Mieke De Wit

2

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Emmanuel Gustin

3

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Inge Keuleers

4

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Johan Vandersmissen

5

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Sabine Hallenberger

6

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Kurt Hertogs

7

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

language of work or name

0 references

publication date

10 October 2007

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

number of pages

7

1 reference

based on heuristic

inferred from page(s)

Journal of Virology

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

81

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

24

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

13845-13851

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Ultra-high resolution crystal structure of HIV-1 protease mutant reveals two binding sites for clinical inhibitor TMC114

1 reference

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Drug-target residence time and its implications for lead optimization

1 reference

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Kinetic determinations of molecular interactions using Biacore--minimum data requirements for efficient experimental design

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2168871

27 May 2018

TMC114, a novel human immunodeficiency virus type 1 protease inhibitor active against protease inhibitor-resistant viruses, including a broad range of clinical isolates

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2168871

27 May 2018

Discovery and selection of TMC114, a next generation HIV-1 protease inhibitor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2168871

27 May 2018

Structural and thermodynamic basis for the binding of TMC114, a next-generation human immunodeficiency virus type 1 protease inhibitor

1 reference

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The prevalence of antiretroviral drug resistance in the United States

1 reference

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27 May 2018

Kinetic and thermodynamic characterization of HIV-1 protease inhibitors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2168871

27 May 2018

Novel bis-tetrahydrofuranylurethane-containing nonpeptidic protease inhibitor (PI) UIC-94017 (TMC114) with potent activity against multi-PI-resistant human immunodeficiency virus in vitro.

1 reference

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27 May 2018

Lack of synergy for inhibitors targeting a multi-drug-resistant HIV-1 protease

1 reference

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27 May 2018

Determination of interaction kinetic constants for HIV-1 protease inhibitors using optical biosensor technology

1 reference

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27 May 2018

BIACORE data processing: an evaluation of the global fitting procedure

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2168871

27 May 2018

Affinity analysis of non-steady-state data obtained under mass transport limited conditions using BIAcore technology

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2168871

27 May 2018

Potent HIV protease inhibitors incorporating high-affinity P2-ligands and (R)-(hydroxyethylamino)sulfonamide isostere

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2168871

27 May 2018

A rapid method for simultaneous detection of phenotypic resistance to inhibitors of protease and reverse transcriptase in recombinant human immunodeficiency virus type 1 isolates from patients treated with antiretroviral drugs

1 reference

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27 May 2018

Declining morbidity and mortality among patients with advanced human immunodeficiency virus infection. HIV Outpatient Study Investigators

1 reference

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27 May 2018

Interpreting complex binding kinetics from optical biosensors: a comparison of analysis by linearization, the integrated rate equation, and numerical integration.

1 reference

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27 May 2018

Real-time biospecific interaction analysis using surface plasmon resonance and a sensor chip technology

1 reference

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27 May 2018

Update of the drug resistance mutations in HIV-1: Fall 2005.

1 reference

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16 August 2018

Multidrug Resistance to HIV-1 Protease Inhibition Requires Cooperative Coupling between Distal Mutations

1 reference

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16 August 2018

Utilization of molybdenum- and palladium-catayzed dynamic kinetic asymmetric transformations for the preparation of tertiary and quaternary stereogenic centers: a concise synthesis of tipranavir

1 reference

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16 August 2018

Phenotypic and genotypic analysis of clinical HIV-1 isolates reveals extensive protease inhibitor cross-resistance: a survey of over 6000 samples.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2168871

16 August 2018

Kinetic analysis of macromolecular interactions using surface plasmon resonance biosensors

1 reference

https://pubmed.ncbi.nlm.nih.gov/17928344

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Why you should be using more SPR biosensor technology

1 reference

https://pubmed.ncbi.nlm.nih.gov/17928344

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Efficacy and safety of TMC114/ritonavir in treatment-experienced HIV patients: 24-week results of POWER 1

1 reference

https://pubmed.ncbi.nlm.nih.gov/17928344

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1128/JVI.01184-07

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

ResearchGate publication ID

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