(Q42948655)

English

Synthesis of omeprazole analogues and evaluation of these as potential inhibitors of the multidrug efflux pump NorA of Staphylococcus aureus

scientific article published on 13 November 2006

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Synthesis of omeprazole analogues and evaluation of these as potential inhibitors of the multidrug efflux pump NorA of Staphylococcus aureus (English)

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Staphylococcus aureus

1 reference

based on heuristic

inferred from title

1 reference

based on heuristic

inferred from title

3

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

author name string

Céline Vidaillac

1

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Jean Guillon

2

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Isabelle Forfar-Bares

4

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Boubakar B Ba

5

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Jean Grellet

6

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Stéphane Moreau

7

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Daniel-Henri Caignard

8

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Christian Jarry

9

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Claudine Quentin

10

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

language of work or name

0 references

publication date

13 November 2006

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Antimicrobial Agents and Chemotherapy

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

51

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

3

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

831-838

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

Activity of gatifloxacin in an in vitro pharmacokinetic-pharmacodynamic model against Staphylococcus aureus strains either susceptible to ciprofloxacin or exhibiting various levels and mechanisms of ciprofloxacin resistance

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Bacterial efflux systems and efflux pumps inhibitors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Bacterial efflux pump inhibition.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Inhibition of antibiotic efflux in bacteria by the novel multidrug resistance inhibitors biricodar (VX-710) and timcodar (VX-853).

1 reference

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27 May 2018

Structural understanding of efflux-mediated drug resistance: potential routes to efflux inhibition

1 reference

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27 May 2018

The basis of differentiation of PPIs

1 reference

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27 May 2018

Synthesis, antimalarial activity, and molecular modeling of new pyrrolo[1,2-a]quinoxalines, bispyrrolo[1,2-a]quinoxalines, bispyrido[3,2-e]pyrrolo[1,2-a]pyrazines, and bispyrrolo[1,2-a]thieno[3,2-e]pyrazines

1 reference

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27 May 2018

The choice of proton pump inhibitor: does it matter?

1 reference

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27 May 2018

Efflux-mediated drug resistance in bacteria

1 reference

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27 May 2018

Antibiotic efflux pumps in prokaryotic cells: occurrence, impact on resistance and strategies for the future of antimicrobial therapy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Phenothiazines and thioxanthenes inhibit multidrug efflux pump activity in Staphylococcus aureus

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Expression of efflux pump gene pmrA in fluoroquinolone-resistant and -susceptible clinical isolates of Streptococcus pneumoniae

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

NorA functions as a multidrug efflux protein in both cytoplasmic membrane vesicles and reconstituted proteoliposomes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Efflux in bacteria: what do we really know about it?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Efflux pumps: their role in antibacterial drug discovery

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

In search of natural substrates and inhibitors of MDR pumps.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Improved high performance liquid chromatographic analysis of omeprazole in human plasma

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Synthesis of new 2-(aminomethyl)-4-phenylpyrrolo[1,2-a]-quinoxalines and their preliminary in-vivo central dopamine antagonist activity evaluation in mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Molecular properties of bacterial multidrug transporters

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

The proton-pump inhibitors: similarities and differences

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Multiple novel inhibitors of the NorA multidrug transporter of Staphylococcus aureus.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Introduction of a norA promoter region mutation into the chromosome of a fluoroquinolone-susceptible strain of Staphylococcus aureus using plasmid integration

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Effects of NorA inhibitors on in vitro antibacterial activities and postantibiotic effects of levofloxacin, ciprofloxacin, and norfloxacin in genetically related strains of Staphylococcus aureus

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Mechanisms of fluoroquinolone resistance in genetically related strains of Staphylococcus aureus

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Mutations affecting substrate specificity of the Bacillus subtilis multidrug transporter Bmr.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Proton-dependent multidrug efflux systems

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Hydrophilicity of quinolones is not an exclusive factor for decreased activity in efflux-mediated resistant mutants of Staphylococcus aureus

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Inducible NorA-mediated multidrug resistance in Staphylococcus aureus

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

Efflux-mediated fluoroquinolone resistance in Staphylococcus aureus

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

27 May 2018

2-[[(4-Amino-2-pyridyl)methyl]sulfinyl]benzimidazole H+/K+-ATPase inhibitors. The relationship between pyridine basicity, stability, and activity

1 reference

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Oral bioavailability of omeprazole before and after chronic therapy in patients with duodenal ulcer

1 reference

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27 May 2018

Uptake of sparfloxacin and norfloxacin by clinical isolates of Staphylococcus aureus

1 reference

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27 May 2018

64 The measurement of membrane potential and ΔpH in cells, organelles, and vesicles

1 reference

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27 May 2018

Synthesis of functionalized 2-aryl-5-nitro-1H-indoles and their activity as bacterial NorA efflux pump inhibitors

1 reference

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16 August 2018

Structural differences between paroxetine and femoxetine responsible for differential inhibition of Staphylococcus aureus efflux pumps

1 reference

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16 August 2018

Phenylpiperidine selective serotonin reuptake inhibitors interfere with multidrug efflux pump activity in Staphylococcus aureus

1 reference

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16 August 2018

A novel inhibitor of multidrug efflux pumps in Staphylococcus aureus

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1803156

16 August 2018

Comité de l'Antibiogramme de la Société Française de Microbiologie report 2003

1 reference

https://pubmed.ncbi.nlm.nih.gov/17101679

12 December 2020

based on heuristic

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Synthesis of 2-[[(4-fluoroalkoxy-2-pyridyl)methyl]sulfinyl]-1H- benzimidazoles as antiulcer agents

1 reference

https://pubmed.ncbi.nlm.nih.gov/17101679

12 December 2020

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Polyacylated oligosaccharides from medicinal Mexican morning glory species as antibacterials and inhibitors of multidrug resistance in Staphylococcus aureus

1 reference

https://pubmed.ncbi.nlm.nih.gov/17101679

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1128/AAC.01306-05

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

11 November 2017

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