(Q43333422)

19 November 2017

title

GSK962040: a small molecule motilin receptor agonist which increases gastrointestinal motility in conscious dogs (English)

1 reference

19 November 2017

S Leming

1

1 reference

19 November 2017

J Broad

2

1 reference

19 November 2017

S J Cozens

3

1 reference

19 November 2017

M Otterson

4

1 reference

19 November 2017

W Winchester

5

1 reference

19 November 2017

K Lee

6

1 reference

19 November 2017

G E Dukes

7

1 reference

19 November 2017

G J Sanger

8

1 reference

19 November 2017

publication date

5 September 2011

1 reference

Neurogastroenterology and Motility

19 November 2017

published in

1 reference

19 November 2017

volume

23

1 reference

19 November 2017

issue

10

1 reference

19 November 2017

page(s)

958-e410

1 reference

Development of drugs for gastrointestinal motor disorders: translating science to clinical need

19 November 2017

cites work

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Drug Insight: from disturbed motility to disordered movement--a review of the clinical benefits and medicolegal risks of metoclopramide

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Motilin, ghrelin and related neuropeptides as targets for the treatment of GI diseases.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

The use of erythromycin as a gastrointestinal prokinetic agent in adult critical care: benefits versus risks

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Therapeutic drugs that behave as mechanism-based inhibitors of cytochrome P450 3A4

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

The identification of and rationale for drugs which act at the motilin receptor.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Efficacy of mitemcinal, a motilin agonist, on gastrointestinal symptoms in patients with symptoms suggesting diabetic gastropathy: a randomized, multi-center, placebo-controlled trial

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Discovery of a potent and novel motilin agonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

GSK962040: a small molecule, selective motilin receptor agonist, effective as a stimulant of human and rabbit gastrointestinal motility

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Discovery of N-(3-fluorophenyl)-1-[(4-([(3S)-3-methyl-1-piperazinyl]methyl)phenyl)acetyl]-4-piperidinamine (GSK962040), the first small molecule motilin receptor agonist clinical candidate.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Stepwise loss of motilin and its specific receptor genes in rodents

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

The translational value of rodent gastrointestinal functions: a cautionary tale.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Molecular identification and characterization of the dog motilin receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Prokineticin-2, motilin, ghrelin and metoclopramide: prokinetic utility in mouse stomach and colon

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

The rabbit motilin receptor: molecular characterisation and pharmacology.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Effects of cholinoceptor and 5-hydroxytryptamine3 receptor antagonism on erythromycin-induced canine intestinal motility disruption and emesis

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Motilides accelerate regional gastrointestinal transit in the dog.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

Erythromycin induces migrating motor complex in human gastrointestinal tract.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1365-2982.2011.01770.X

10.1111/J.1365-2982.2011.01770.X

21 January 2018

Identifiers

DOI

1 reference

19 November 2017

1 reference