(Q43775734)

English

Efficacy of antipsychotic agents at human 5-HT(1A) receptors determined by [3H]WAY100,635 binding affinity ratios: relationship to efficacy for G-protein activation

scientific article published in October 2001

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Europe PubMed Central

PubMed publication ID

26 November 2017

Efficacy of antipsychotic agents at human 5-HT(1A) receptors determined by [3H]WAY100,635 binding affinity ratios: relationship to efficacy for G-protein activation (English)

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

Adrian Newman-Tancredi

1

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

author name string

Verrièle L

2

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

Touzard M

3

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

Millan MJ

4

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

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publication date

1 October 2001

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

European Journal of Pharmacology

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Europe PubMed Central

PubMed publication ID

26 November 2017

428

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

2

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

177-184

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

Prevention by (+/-)-8-hydroxy-2-(di-n-propylamino)tetralin of both catalepsy and the rises in rat striatal dopamine metabolism caused by haloperidol

1 reference

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7 January 2021

Correlation between low/high affinity ratios for 5-HT(1A) receptors and intrinsic activity

1 reference

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7 January 2021

A review of central 5-HT receptors and their function

1 reference

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Arrestin binding to the G protein-coupled N-formyl peptide receptor is regulated by the conserved "DRY" sequence

1 reference

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7 January 2021

[3H]WAYâ 100635 for 5â HT1A receptor autoradiography in human brain: a comparison with [3H]8â OHâ DPAT and demonstration of increased binding in the frontal cortex in schizophrenia

1 reference

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7 January 2021

Inverse agonism at heptahelical receptors: concept, experimental approach and therapeutic potential

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7 January 2021

5-HT1A receptor agonists: recent developments and controversial issues

1 reference

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7 January 2021

Electrophysiological, biochemical, neurohormonal and behavioural studies with WAY-100635, a potent, selective and silent 5-HT1A receptor antagonist

1 reference

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7 January 2021

Relative affinities of drugs acting at cholinoceptors in displacing agonist and antagonist radioligands: the NMS/Oxo-M ratio as an index of efficacy at cortical muscarinic receptors

1 reference

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7 January 2021

The selective 5-HT1A antagonist radioligand [3H]WAY 100635 labels both G-protein-coupled and free 5-HT1A receptors in rat brain membranes

1 reference

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7 January 2021

Alterations in the cortical serotonergic system in schizophrenia: a postmortem study

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7 January 2021

Augmentation with buspirone: a review

1 reference

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7 January 2021

Relationship between dopaminergic and serotonergic neuronal activity in the frontal cortex and the action of typical and atypical antipsychotic drugs

1 reference

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7 January 2021

The effect of serotonin(1A) receptor agonism on antipsychotic drug-induced dopamine release in rat striatum and nucleus accumbens

1 reference

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7 January 2021

5-HT(2A) and D(2) receptor blockade increases cortical DA release via 5-HT(1A) receptor activation: a possible mechanism of atypical antipsychotic-induced cortical dopamine release

1 reference

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7 January 2021

8-Hydroxy-2-(di-n-propylamino) tetralin, a selective serotonin1A receptor agonist, blocks haloperidol-induced catalepsy by an action on raphe nuclei medianus and dorsalis

1 reference

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7 January 2021

Pharmacological characterization of recombinant human 5-hydroxytryptamine1A receptors using a novel antagonist radioligand, [3H]WAY-100635.

1 reference

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7 January 2021

The molecular biology of serotonin receptors: therapeutic implications for the interface of mood and psychosis

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7 January 2021

Reversal of neuroleptic-induced catalepsy by novel aryl-piperazine anxiolytic drugs

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7 January 2021

S 14506: novel receptor coupling at 5-HT(1A) receptors.

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7 January 2021

Clozapine is a partial agonist at cloned, human serotonin 5-HT1A receptors.

1 reference

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7 January 2021

Inhibition of the constitutive activity of human 5-HT1A receptors by the inverse agonist, spiperone but not the neutral antagonist, WAY 100,635

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2801%2901344-9

7 January 2021

Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study

1 reference

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7 January 2021

Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2801%2901344-9

7 January 2021

Differential modulation by GTPgammaS of agonist and inverse agonist binding to h5-HT(1A) receptors revealed by [3H]-WAY100,635

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2801%2901344-9

7 January 2021

Binding of antipsychotic drugs to human brain receptors focus on newer generation compounds

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2801%2901344-9

7 January 2021

Clozapine increases dopamine release in prefrontal cortex by 5-HT1A receptor activation

1 reference

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7 January 2021

5-HT(1A) receptor agonist-antagonist binding affinity difference as a measure of intrinsic activity in recombinant and native tissue systems

1 reference

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7 January 2021

Identifiers

10.1016/S0014-2999(01)01344-9

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

26 November 2017

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