(Q43913062)

English

Specific labelling of serotonin 5-HT(1B) receptors in rat frontal cortex with the novel, phenylpiperazine derivative, [3H]GR125,743. A pharmacological characterization

scientific article published in April 2002

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Specific labelling of serotonin 5-HT(1B) receptors in rat frontal cortex with the novel, phenylpiperazine derivative, [3H]GR125,743. A pharmacological characterization (English)

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

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Adrian Newman-Tancredi

2

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Europe PubMed Central

PubMed publication ID

28 November 2017

author name string

Millan MJ

1

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Europe PubMed Central

PubMed publication ID

28 November 2017

Lochon S

3

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Europe PubMed Central

PubMed publication ID

28 November 2017

Touzard M

4

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Europe PubMed Central

PubMed publication ID

28 November 2017

Aubry S

5

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Europe PubMed Central

PubMed publication ID

28 November 2017

Audinot V

6

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Europe PubMed Central

PubMed publication ID

28 November 2017

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publication date

1 April 2002

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Pharmacology, Biochemistry and Behavior

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Europe PubMed Central

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28 November 2017

71

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Europe PubMed Central

PubMed publication ID

28 November 2017

4

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Europe PubMed Central

PubMed publication ID

28 November 2017

589-598

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

Binding profile of the novel 5-HT1B/1D receptor antagonist, [3H]GR 125,743, in guinea-pig brain: a comparison with [3H]5-carboxamidotryptamine

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Inverse agonist properties of antipsychotic agents at cloned, human (h) serotonin (5-HT)(1B) and h5-HT(1D) receptors

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Constitutive activity at serotonin 5-HT(1D) receptors: detection by homologous GTPgammaS versus [(35)S]-GTPgammaS binding isotherms.

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A review of central 5-HT receptors and their function

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L-694,247: a potent 5-HT1D receptor agonist

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Absence of cocaine-induced place conditioning in serotonin 1B receptor knock-out mice.

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Activation of 5-HT1B receptors suppresses low but not high frequency synaptic transmission in the rat subicular cortex in vitro

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Co-localization of 5-HT1B- and 5-HT1D receptor mRNA in serotonergic cell bodies in guinea pig dorsal raphé nucleus: a double labeling in situ hybridization histochemistry study.

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Humanization of mouse 5-hydroxytryptamine1B receptor gene by homologous recombination: in vitro and in vivo characterization.

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No contractile effect for 5-HT1D and 5-HT1F receptor agonists in human and bovine cerebral arteries: similarity with human coronary artery

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Dopamine release in the nucleus accumbens and latent inhibition in the rat following microinjections of a 5-HT1B agonist into the dorsal subiculum: implications for schizophrenia

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Key role of 5-HT1B receptors in the regulation of paradoxical sleep as evidenced in 5-HT1B knock-out mice.

1 reference

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Autoradiographic characterisation and localisation of 5-HT1D compared to 5-HT1B binding sites in rat brain.

1 reference

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3-(Piperazinylpropyl)indoles: selective, orally bioavailable h5-HT1D receptor agonists as potential antimigraine agents

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GR 127935 reduces basal locomotor activity and prevents RU 24969-, but not D -amphetamine-induced hyperlocomotion, in the Wistar-Kyoto Hyperactive (WKHA) rat

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Effects of PNU-109,291, a selective 5-HT1D receptor agonist, on electrically induced dural plasma extravasation and capsaicin-evoked c-fos immunoreactivity within trigeminal nucleus caudalis.

1 reference

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Effects of selected serotonin 5-HT(1) and 5-HT(2) receptor agonists on feeding behavior: possible mechanisms of action

1 reference

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Human 5-HT1B receptor stimulated inositol phospholipid hydrolysis in CHO cells: synergy with Gq-coupled receptors

1 reference

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7 January 2021

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5-HT1B receptor knockout, but not 5-HT1A receptor knockout mice, show reduced startle reactivity and footshock-induced sensitization, as measured with the acoustic startle response

1 reference

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7 January 2021

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Characterization of human serotonin 1D and 1B receptors using [3H]-GR-125743, a novel radiolabelled serotonin 5HT1D/1B receptor antagonist

1 reference

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Knockout mice reveal opposite roles for serotonin 1A and 1B receptors in prepulse inhibition

1 reference

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7 January 2021

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5-HT1A and 5-HT1B receptors control the firing of serotoninergic neurons in the dorsal raphe nucleus of the mouse: studies in 5-HT1B knock-out mice

1 reference

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7 January 2021

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Altered expression and functions of serotonin 5-HT1Aand 5-HT1Breceptors in knock-out mice lacking the 5-HT transporter

1 reference

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Activation of 5-HT1B receptors in the nucleus accumbens reduces amphetamine-induced enhancement of responding for conditioned reward.

1 reference

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Local infusion of the selective 5HT-1b agonist CP-93,129 facilitates striatal dopamine release in vivo

1 reference

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7 January 2021

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The selective 5-HT1B receptor inverse agonist 1'-methyl-5-[[2'-methyl-4'-(5-methyl-1,2, 4-oxadiazol-3-yl)biphenyl-4-yl]carbonyl]-2,3,6,7-tetrahydro- spiro[furo[2,3-f]indole-3,4'-piperidine] (SB-224289) potently blocks terminal 5-HT autoreceptor func

1 reference

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7 January 2021

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Functional characteristics of heterologously expressed 5-HT receptors

1 reference

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Serotonergic functions in arousal and motor activity

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Modulation of dialysate levels of dopamine, noradrenaline, and serotonin (5-HT) in the frontal cortex of freely-moving rats by (-)-pindolol alone and in association with 5-HT reuptake inhibitors: comparative roles of beta-adrenergic, 5-HT1A, and 5-H

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The ability of WAY100,635 to potentiate the neurochemical and functional actions of fluoxetine is enhanced by co-administration of SB224,289, but not BRL15572

1 reference

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Identification of an amino acid residue important for binding of methiothepin and sumatriptan to the human 5-HT(1B) receptor

1 reference

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7 January 2021

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5-HT 1D receptors mediate SKF 99101H-induced hypothermia in the guinea pig.

1 reference

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Species differences in the pharmacology of terminal 5-HT autoreceptors in mammalian brain

1 reference

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Immunolabeling of central serotonin 5-HT1D beta receptors in the rat, mouse, and guinea pig with a specific anti-peptide antiserum

1 reference

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7 January 2021

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Comparison of the vasoconstrictor effects of the selective 5-HT1D-receptor agonist L-775,606 with the mixed 5-HT1B/1D-receptor agonist sumatriptan and 5-HT in human isolated coronary artery

1 reference

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7 January 2021

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Absence of fenfluramine-induced anorexia and reduced c-Fos induction in the hypothalamus and central amygdaloid complex of serotonin 1B receptor knock-out mice.

1 reference

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7 January 2021

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5-HT1B receptor knock-out mice exhibit increased exploratory activity and enhanced spatial memory performance in the Morris water maze.

1 reference

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Acetylcholine release from rat hippocampal slices is modulated by 5-hydroxytryptamine

1 reference

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5-HT system and cognition

1 reference

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7 January 2021

based on heuristic

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The 5-HT1B receptors

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The induction of pain: an integrative review.

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Reciprocal autoreceptor and heteroreceptor control of serotonergic, dopaminergic and noradrenergic transmission in the frontal cortex: relevance to the actions of antidepressant agents

1 reference

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Quantitative autoradiography of 5-CT-sensitive (5-HT1D) and 5-CT-insensitive (5-HT1E) serotonin receptors in human brain

1 reference

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7 January 2021

based on heuristic

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The unique effect of methiothepin on the terminal serotonin autoreceptor in the rat hypothalamus could be an example of inverse agonism

1 reference

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7 January 2021

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The possible role of 5-HT(1B/D) receptors in psychiatric disorders and their potential as a target for therapy

1 reference

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7 January 2021

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Regulation of central synaptic transmission by 5-HT(1B) auto- and heteroreceptors.

1 reference

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7 January 2021

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Serotonergic lesioning differentially affects presynaptic and postsynaptic 5-HT1B receptor mRNA levels in rat brain.

1 reference

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7 January 2021

based on heuristic

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Inverse agonism and constitutive activity as functional correlates of serotonin h5-HT(1B) receptor/G-protein stoichiometry

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Differential modulation by GTPgammaS of agonist and inverse agonist binding to h5-HT(1A) receptors revealed by [3H]-WAY100,635

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

[3H]-5-carboxamidotryptamine labels 5-HT1D binding sites in bovine substantia nigra

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

A single amino-acid difference confers major pharmacological variation between human and rodent 5-HT1B receptors

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

5-HT1D receptors regulate 5-HT release in the rat raphe nuclei. In vivo voltammetry and in vitro superfusion studies

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Cellular and subcellular localization of 5-hydroxytryptamine1B receptors in the rat central nervous system: immunocytochemical, autoradiographic and lesion studies

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Enhanced aggressive behavior in mice lacking 5-HT1B receptor.

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Effects of the 5-HT1D receptor antagonist GR127935 on extracellular levels of 5-HT in the guinea-pig frontal cortex as measured by microdialysis.

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

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1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Enhanced 5-HT metabolism and synthesis rate by the new selective r5-HT1B receptor antagonist, NAS-181 in the rat brain

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Triptans in migraine: a comparative review of pharmacology, pharmacokinetics and efficacy

1 reference

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7 January 2021

based on heuristic

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Characterization and distribution of putative 5-ht7 receptors in guinea-pig brain

1 reference

https://api.crossref.org/works/10.1016%2FS0091-3057%2801%2900716-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Autoradiographic visualisation of [3H]5-carboxamidotryptamine binding sites in the guinea pig and rat brain

1 reference

https://api.crossref.org/works/10.1016%2FS0091-3057%2801%2900716-X

7 January 2021

based on heuristic

inferred from DOI database lookup

GR127935 acts as a partial agonist at recombinant human 5-HT1D alpha and 5-HT1D beta receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0091-3057%2801%2900716-X

7 January 2021

based on heuristic

inferred from DOI database lookup

5-HT1B receptor-mediated contractions in human temporal artery: evidence from selective antagonists and 5-HT receptor mRNA expression

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

5-Hydroxytryptamine-induced outward currents mediated via 5-HT(1A) receptors in neurons of the rat dorsolateral septal nucleus

1 reference

https://api.crossref.org/works/10.1016%2FS0091-3057%2801%2900716-X

7 January 2021

based on heuristic

inferred from DOI database lookup

The 5-HT1D receptor antagonist GR-127,935 prevents inhibitory effects of sumatriptan but not CP-122,288 and 5-CT on neurogenic plasma extravasation within guinea pig dura mater

1 reference

https://api.crossref.org/works/10.1016%2FS0091-3057%2801%2900716-X

7 January 2021

based on heuristic

inferred from DOI database lookup

Native 5-HT1B receptors expressed in OK cells display dual coupling to elevation of intracellular calcium concentrations and inhibition of adenylate cyclase

1 reference

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7 January 2021

based on heuristic

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Identifiers

10.1016/S0091-3057(01)00716-X

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

28 November 2017

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