(Q43978611)

28 November 2017

title

Progress in the proxifan class: heterocyclic congeners as novel potent and selective histamine H(3)-receptor antagonists (English)

1 reference

28 November 2017

author

Jean-Charles Schwartz

7

object named as

Jean-Charles Schwartz

0 references

Sven Grassmann

1

object named as

Sven Grassmann

1 reference

28 November 2017

3

Xavier Ligneau

1 reference

28 November 2017

4

Sigurd Elz

1 reference

28 November 2017

6

Jean-Michel Arrang

1 reference

28 November 2017

Bassem Sadek

2

1 reference

28 November 2017

C Robin Ganellin

5

1 reference

28 November 2017

Holger Stark

8

1 reference

28 November 2017

Walter Schunack

9

1 reference

28 November 2017

language of work or name

English

0 references

publication date

1 May 2002

1 reference

European Journal of Pharmaceutical Sciences

28 November 2017

published in

1 reference

28 November 2017

volume

15

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28 November 2017

issue

4

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28 November 2017

page(s)

367-378

1 reference

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

28 November 2017

cites work

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Highly potent and selective ligands for histamine H3-receptors

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Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors

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Studies in detoxication. 75. Further observations on the metabolism of hydrazides of aromatic acids

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A novel series of (phenoxyalkyl)imidazoles as potent H3-receptor histamine antagonists.

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Iodoaminopotentidine and related compounds: a new class of ligands with high affinity and selectivity for the histamine H2 receptor.

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Ciproxifan and chemically related compounds are highly potent and selective histamine H3-receptor antagonists

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4-Alkynylphenyl imidazolylpropyl ethers as selective histamine H3-receptor antagonists with high oral central nervous system activity

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The Use of Diethyl Azodicarboxylate and Triphenylphosphine in Synthesis and Transformation of Natural Products

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High constitutive activity of native H3 receptors regulates histamine neurons in brain.

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Inhibition of histamine versus acetylcholine metabolism as a mechanism of tacrine activity.

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Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes

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Neuronal histamine deficit in Alzheimer's disease

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New histamine H(3)-receptor ligands of the proxifan series: imoproxifan and other selective antagonists with high oral in vivo potency.

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Benzophenone derivatives and related compounds as potent histamine H3-receptor antagonists and potential PET/SPECT ligands

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7 January 2021

The moderate affinity of clozapine at H3 receptors is not shared by its two major metabolites and by structurally related and unrelated atypical neuroleptics.

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7 January 2021

Novel histamine H3 receptor antagonists: affinities in an H3 receptor binding assay and potencies in two functional H3 receptor models

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7 January 2021

Histaminergic transmission in the mammalian brain

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7 January 2021

[125I]iodoproxyfan and related compounds: a reversible radioligand and novel classes of antagonists with high affinity and selectivity for the histamine H3 receptor.

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7 January 2021

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7 January 2021

Analogues and derivatives of ciproxifan, a novel prototype for generating potent histamine H3-receptor antagonists.

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7 January 2021

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7 January 2021

Novel 5-HT3 antagonists. Indole oxadiazoles

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7 January 2021

Cloning and cerebral expression of the guinea pig histamine H3 receptor: evidence for two isoforms

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7 January 2021

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7 January 2021

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Identifiers

DOI

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/k5h3z5gu35c23dzmduudnjl5oy

30 July 2022

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Fatcat ID

release_k5h3z5gu35c23dzmduudnjl5oy

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Fatcat

https://api.fatcat.wiki/v0/release/k5h3z5gu35c23dzmduudnjl5oy

30 July 2022

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https://api.fatcat.wiki/v0/release/k5h3z5gu35c23dzmduudnjl5oy

1 reference

30 July 2022