(Q43979326)

28 November 2017

title

Interaction of 1,2,4-substituted piperazines, new serotonin receptor ligands, with 5-HT1A and 5-HT2A receptors (English)

1 reference

28 November 2017

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9

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28 November 2017

1

Zdzisław Chilmonczyk

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Ewa Chojnacka-Wójcik

4

object named as

Ewa Chojnacka-Wójcik

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28 November 2017

5

Ewa Tatarczyńska

1 reference

28 November 2017

3

Joanna Iskra-Jopa

1 reference

28 November 2017

Aleksandra Kłodzińska

6

object named as

Aleksandra Kłodzińska

1 reference

28 November 2017

Marcin Cybulski

2

1 reference

28 November 2017

Andrzej Leś

7

1 reference

28 November 2017

Agnieszka Bronowska

8

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28 November 2017

publication date

1 April 2002

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28 November 2017

number of pages

17

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based on heuristic

inferred from page(s)

published in

Il Farmaco

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28 November 2017

volume

57

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28 November 2017

issue

4

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28 November 2017

page(s)

285-301

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Characterization of MDL 73005EF as a 5-HT1A selective ligand and its effects in animal models of anxiety: comparison with buspirone, 8-OH-DPAT and diazepam

28 November 2017

cites work

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5-HT1A receptor agonists: recent developments and controversial issues

7 January 2021

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Antidepressant-like activity of compounds with varying efficacy at 5-HT1A receptors

7 January 2021

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Buspirone Analogs as Ligands of the 5-HT1A Receptor. 1. The Molecular Structure of Buspirone and Its Two Analogs

7 January 2021

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Conformational flexibility of serotonin1A receptor ligands from crystallographic data. Updated model of the receptor pharmacophore.

7 January 2021

1 reference

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8-Hydroxy-2-(di-n-propylamino)-tetralin discriminates between subtypes of the 5-HT1 recognition site

7 January 2021

1 reference

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Involvement of 5-HT1C-receptors in drug-induced penile erections in rats

7 January 2021

1 reference

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The involvement of subtypes of the 5-HT1 receptor and of catecholaminergic systems in the behavioural response to 8-hydroxy-2-(di-n-propylamino)tetralin in the rat.

7 January 2021

1 reference

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Molecular dynamics of buspirone analogues interacting with the 5-HT1A and 5-HT2A serotonin receptors

7 January 2021

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Molecular dynamics of 5-HT1A and 5-HT2A serotonin receptors with methylated buspirone analogues.

7 January 2021

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A theoretical study of the dielectric constant of protein.

7 January 2021

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The ligand-binding site of buspirone analogues at the 5-HT1A receptor.

7 January 2021

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Crystal structure of rhodopsin: A G protein-coupled receptor

7 January 2021

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Projection structure of rhodopsin

7 January 2021

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Low resolution structure of bovine rhodopsin determined by electron cryo-microscopy.

7 January 2021

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The probable arrangement of the helices in G protein-coupled receptors.

7 January 2021

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An alpha-carbon template for the transmembrane helices in the rhodopsin family of G-protein-coupled receptors

7 January 2021

1 reference

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Primary structure of the human platelet serotonin 5-HT2A receptor: identify with frontal cortex serotonin 5-HT2A receptor

7 January 2021

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Requirement of rigid-body motion of transmembrane helices for light activation of rhodopsin

7 January 2021

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Molecular mechanisms involved in muscarinic acetylcholine receptor-mediated G protein activation studied by insertion mutagenesis

7 January 2021

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Ligand induced conformational states of the 5-HT(1A) receptor

7 January 2021

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Ab InitioModeling and Molecular Dynamics Simulation of the α1b-Adrenergic Receptor Activation

7 January 2021

1 reference

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The role of conserved aspartate and serine residues in ligand binding and in function of the 5-HT1A receptor: a site-directed mutation study

7 January 2021

1 reference

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Identification of conserved aromatic residues essential for agonist binding and second messenger production at 5-hydroxytryptamine2A receptors

7 January 2021

1 reference

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Identification, expression, and pharmacology of a Cys23-Ser23 substitution in the human 5-HT2c receptor gene (HTR2C)

7 January 2021

1 reference

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Five-transmembrane domains appear sufficient for a G protein-coupled receptor: functional five-transmembrane domain chemokine receptors

7 January 2021

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Transducin activation by rhodopsin without a covalent bond to the 11-cis-retinal chromophore

7 January 2021

1 reference

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Involvement of Asn-293 in stereospecific agonist recognition and in activation of the beta 2-adrenergic receptor

7 January 2021

1 reference

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Agonists induce conformational changes in transmembrane domains III and VI of the beta2 adrenoceptor

7 January 2021

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How receptors talk to trimeric G proteins

7 January 2021

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Identification of a receptor/G-protein contact site critical for signaling specificity and G-protein activation

7 January 2021

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7 January 2021

1 reference

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Characterization of N- and C-terminal deletion mutants of the rat serotonin HT2 receptor in Xenopus laevis oocytes.

7 January 2021

1 reference

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Identification of a Gs coupling domain in the amino terminus of the third intracellular loop of the alpha 2A-adrenergic receptor. Evidence for distinct structural determinants that confer Gs versus Gi coupling

7 January 2021

1 reference

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Mapping the binding site pocket of the serotonin 5-Hydroxytryptamine2A receptor. Ser3.36(159) provides a second interaction site for the protonated amine of serotonin but not of lysergic acid diethylamide or bufotenin

7 January 2021

1 reference

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Site-directed mutagenesis of a single residue changes the binding properties of the serotonin 5-HT2 receptor from a human to a rat pharmacology

7 January 2021

1 reference

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Depletion of brain serotonin differently affects behaviors induced by 5HT1A, 5HT1C, and 5HT2 receptor activation in rats

7 January 2021

1 reference

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Structure-activity relationship studies of central nervous system agents. 13. 4-[3-(Benzotriazol-1-yl)propyl]-1-(2-methoxyphenyl)piperazine, a new putative 5-HT1A receptor antagonist, and its analogs

7 January 2021

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The pharmacology of the hypothermic response in mice to 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT). A model of presynaptic 5-HT1 function

7 January 2021

1 reference

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8-[4-[2-(1,2,3,4-Tetrahydroisoquinolinyl]butyl-8-azaspiro[4.5]decane-7,9-dione: a new 5-HT1A receptor ligand with the same activity profile as buspirone.

7 January 2021

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Differential effects of 5-hydroxytryptamine1a selective drugs on the 5-HT behavioral syndrome

7 January 2021

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Pharmacodynamic and pharmacokinetic studies in rats of S-8-(2-Furyl)- and R-8-phenyl-2-(di-n-propylamino) tetralin, two novel 5-HT1A receptor agonists in-vitro with different properties in-vivo

7 January 2021

1 reference

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Structure-activity relationship studies of central nervous system agents. 5. Effect of the hydrocarbon chain on the affinity of 4-substituted 1-(3-chlorophenyl)piperazines for 5-HT1A receptor site

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-827X%2802%2901205-3

Functional correlates of serotonin 5-HT1 recognition sites

7 January 2021

1 reference

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10.1016/S0014-827X(02)01205-3

7 January 2021

Identifiers

DOI

1 reference

release_6nekntyiujbaneaveiao3rcnwm

28 November 2017

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/6nekntyiujbaneaveiao3rcnwm

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference