(Q44022781)

29 November 2017

title

Piperidino-hydrocarbon compounds as novel non-imidazole histamine H(3)-receptor antagonists (English)

1 reference

29 November 2017

author

Jean-Charles Schwartz

5

object named as

Jean-Charles Schwartz

0 references

Xavier Ligneau

2

object named as

Xavier Ligneau

1 reference

29 November 2017

3

Heinz H Pertz

1 reference

29 November 2017

1

Galina Meier

1 reference

29 November 2017

C Robin Ganellin

4

1 reference

29 November 2017

Walter Schunack

6

1 reference

29 November 2017

Holger Stark

7

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29 November 2017

language of work or name

English

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publication date

1 August 2002

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Bioorganic & Medicinal Chemistry

29 November 2017

published in

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29 November 2017

volume

10

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29 November 2017

issue

8

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29 November 2017

page(s)

2535-2542

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Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

29 November 2017

cites work

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Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors

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Cloning and functional expression of the human histamine H3 receptor

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Identification of rat H3 receptor isoforms with different brain expression and signaling properties.

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Genomic organization and characterization of splice variants of the human histamine H3 receptor

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High constitutive activity of native H3 receptors regulates histamine neurons in brain.

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Inhibition of histamine versus acetylcholine metabolism as a mechanism of tacrine activity

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7 January 2021

Effects of thioperamide, a histamine H3-receptor antagonist, on a scopolamine-induced learning deficit using an elevated plus-maze test in mice

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7 January 2021

Inhibition of cortical acetylcholine release and cognitive performance by histamine H3 receptor activation in rats

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7 January 2021

Improvement by FUB 181, a novel histamine H3-receptor antagonist, of learning and memory in the elevated plus-maze test in mice

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Therapeutic potential of histamine H3 receptor agonists and antagonists.

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High antagonist potency of GT-2227 and GT-2331, new histamine H3 receptor antagonists, in two functional models

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7 January 2021

General construction pattern of histamine H3-receptor antagonists: change of a paradigm

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7 January 2021

Synthesis of potent non-imidazole histamine H3-receptor antagonists

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7 January 2021

Non-imidazole histamine H3 ligands. Part I. Synthesis of 2-(1-piperazinyl)- and 2-(hexahydro-1H-1,4-diazepin-1-yl)benzothiazole derivatives as H3-antagonists with H1 blocking activities

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7 January 2021

Non-imidazole histamine H3 ligands, Part 2: New 2-substituted benzothiazoles as histamine H3 antagonists

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7 January 2021

Influence of imidazole replacement in different structural classes of histamine H(3)-receptor antagonists

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Novel histamine H(3)-receptor antagonists with carbonyl-substituted 4-(3-(phenoxy)propyl)-1H-imidazole structures like ciproxifan and related compounds

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7 January 2021

New acetylene based histamine H3 receptor antagonists derived from the marine natural product verongamine

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7 January 2021

In-vitro pharmacology of sarpogrelate and the enantiomers of its major metabolite: 5-HT2A receptor specificity, stereoselectivity and modulation of ritanserin-induced depression of 5-HT contractions in rat tail artery

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7 January 2021

Effects of histamine H3-receptor ligands on various biochemical indices of histaminergic neuron activity in rat brain

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7 January 2021

Novel partial agonists for the histamine H(3) receptor with high in vitro and in vivo activity

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7 January 2021

Effects of selected histamine H3 receptor antagonists on tele-methylhistamine levels in rat cerebral cortex

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7 January 2021

A synthetic method for formyl→ethynyl conversion (RCHO→RCCH or RCCR′)

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7 January 2021

Study of the contractile effect of 5-hydroxytryptamine (5-HT) in the isolated longitudinal muscle strip from guinea-pig ileum. Evidence for two distinct release mechanisms.

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7 January 2021

Novel histamine H3 receptor antagonists: affinities in an H3 receptor binding assay and potencies in two functional H3 receptor models

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7 January 2021

Sensitive radioimmunoassays for histamine and tele-methylhistamine in the brain

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7 January 2021

10.1016/S0968-0896(02)00115-3

Identifiers

DOI

1 reference

29 November 2017

1 reference