(Q44061384)

English

2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356.

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scholarly article

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Europe PubMed Central

PubMed publication ID

29 November 2017

2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. (English)

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Europe PubMed Central

PubMed publication ID

29 November 2017

3

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29 November 2017

author name string

Markus Bergauer

1

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Europe PubMed Central

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29 November 2017

Harald Hübner

2

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29 November 2017

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publication date

1 August 2002

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29 November 2017

Bioorganic & Medicinal Chemistry Letters

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29 November 2017

12

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29 November 2017

15

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29 November 2017

1937-1940

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29 November 2017

Cloning of the gene for a human dopamine D4 receptor with high affinity for the antipsychotic clozapine

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Evidence for linkage of a tandem duplication polymorphism upstream of the dopamine D4 receptor gene (DRD4) with attention deficit hyperactivity disorder (ADHD).

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A hypervariable segment in the human dopamine receptor D4 (DRD4) gene.

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3-((4-(4-Chlorophenyl)piperazin-1-yl)-methyl)-1H-pyrrolo-2,3-b-pyridine: an antagonist with high affinity and selectivity for the human dopamine D4 receptor

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Azaindole derivatives with high affinity for the dopamine D4 receptor: Synthesis, ligand binding studies and comparison of molecular electrostatic potential maps

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Cyanoindole derivatives as highly selective dopamine D(4) receptor partial agonists: solid-phase synthesis, binding assays, and functional experiments

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Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213).

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2-Phenyl-4(5)-[[4-(pyrimidin-2-yl)piperazin-1-yl]methyl]imidazole. A highly selective antagonist at cloned human D4 receptors

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NGD 94-1 as an agonist at human recombinant dopamine D4.4 receptors expressed in HEK293 cells

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Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPC synthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179).

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2,2-dicyanovinyl as a nonaromatic aryl bioisostere: synthesis, binding experiments and SAR studies of highly selective dopamine D4 receptor ligands

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Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptor

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Modulation of Intracellular Cyclic AMP Levels by Different Human Dopamine D4 Receptor Variants

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Conjugated enynes as nonaromatic catechol bioisosteres: synthesis, binding experiments, and computational studies of novel dopamine receptor agonists recognizing preferentially the D(3) subtype

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Pramipexole binding and activation of cloned and expressed dopamine D2, D3 and D4 receptors

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Identifiers

10.1016/S0960-894X(02)00316-5

1 reference

Europe PubMed Central

PubMed publication ID

29 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

29 November 2017

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