(Q44424814)

English

Synthesis and Biological Evaluation of Thiol-Based Inhibitors of Glutamate Carboxypeptidase II: Discovery of an Orally Active GCP II Inhibitor

scientific article published on May 8, 2003

In more languages

Statements

scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Synthesis and biological evaluation of thiol-based inhibitors of glutamate carboxypeptidase II: discovery of an orally active GCP II inhibitor (English)

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Synthesis and Biological Evaluation of Thiol-Based Inhibitors of Glutamate Carboxypeptidase II: Discovery of an Orally Active GCP II Inhibitor (English)

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

molecular medicine

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

1

object named as

Pavel Majer

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

author name string

Greg Delahanty

3

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Yao-Sen Ko

5

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Weixing Li

6

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Qun Liu

7

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Jana Poláková

9

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Doris Stoermer

11

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Dilrukshi Vitharana

12

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Eric Yanjun Wang

13

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Anthony Zakrzewski

14

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Camilo Rojas

15

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Eric Burak

18

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Tharin Limsakun

19

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Takashi Tsukamoto

20

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Paul F. Jackson

2

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12723961

29 December 2023

Brian S. Grella

4

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12723961

29 December 2023

Keith M. Maclin

8

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12723961

29 December 2023

Kathryn A. Shaffer

10

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12723961

29 December 2023

Barbara S. Slusher

16

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12723961

29 December 2023

Krystyna M. Wozniak

17

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12723961

29 December 2023

language of work or name

0 references

publication date

1 May 2003

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

8 May 2003

1 reference

National Center for Biotechnology Information

PubMed publication ID

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=12723961

29 December 2023

full work available at URL

https://pubs.acs.org/doi/pdf/10.1021/jm020515w

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Journal of Medicinal Chemistry

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

46

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

10

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

1989-1996

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

l-glutamate as a central neurotransmitter: looking back

1

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Amino acids are still as exciting as ever

2

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Current approaches to multiple parallel synthesis

5

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Design and pharmacological activity of phosphinic acid based NAALADase inhibitors

6

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Competitive inhibition of N-acetylated-alpha-linked acidic dipeptidase activity by N-acetyl-L-aspartyl-beta-linked L-glutamate.

7

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Synthesis of acyclic and dehydroaspartic acid analogues of Ac-Asp-Glu-OH and their inhibition of rat brain N-acetylated alpha-linked acidic dipeptidase (NAALA dipeptidase).

8

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Journal of Medicinal Chemistry

9

43

774

author name string

Nan F.

publication date

2000

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Design of remarkably simple, yet potent urea-based inhibitors of glutamate carboxypeptidase II (NAALADase)

10

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Phosphonate and phosphinate analogues of N-acylated gamma-glutamylglutamate. potent inhibitors of glutamate carboxypeptidase II.

12

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Design, synthesis, and biological activity of a potent inhibitor of the neuropeptidase N-acetylated alpha-linked acidic dipeptidase

13

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Kinetics and inhibition of glutamate carboxypeptidase II using a microplate assay

14

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Selective inhibition of NAALADase, which converts NAAG to glutamate, reduces ischemic brain injury

15

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

GCPII (NAALADase) inhibition prevents long-term diabetic neuropathy in type 1 diabetic BB/Wor rats

16

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Design of angiotensin converting enzyme inhibitors.

18

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Journal of Organic Chemistry

20

67

7368

author name string

Hin B.

publication date

2002

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Inhibition of .gamma.-butyrobetaine hydroxylase by cyclopropyl-substituted .gamma.-butyrobetaines

21

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Design of potent competitive inhibitors of angiotensin-converting enzyme. Carboxyalkanoyl and mercaptoalkanoyl amino acids

23

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Design of potent and specific inhibitors of carboxypeptidases A and B

24

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Structure of membrane glutamate carboxypeptidase.

25

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Design of NAALADase inhibitors: a novel neuroprotective strategy

26

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Journal of Medicinal Chemistry

28

45

4152

author name string

Rong S. B.

publication date

2002

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Captopril: pharmacology, metabolism and disposition

29

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

A peripheral mononeuropathy in rat that produces disorders of pain sensation like those seen in man.

30

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Substrate specificity, inhibition and enzymological analysis of recombinant human glutamate carboxypeptidase II.

31

1 reference

10.1021/JM020515W

https://api.crossref.org/works/10.1021/JM020515W

29 December 2023

Identifiers

10.1021/JM020515W

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Sitelinks

Wikipedia(0 entries)

Wikibooks(0 entries)

Wikinews(0 entries)

Wikiquote(0 entries)

Wikisource(0 entries)

Wikiversity(0 entries)

Wikivoyage(0 entries)

Wiktionary(0 entries)

Multilingual sites(0 entries)

Retrieved from "https://www.wikidata.org/w/index.php?title=Q44424814&oldid=2039676418"