(Q44443061)

3 December 2017

title

Design, synthesis and biological evaluation of new endocannabinoid transporter inhibitors (English)

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3 December 2017

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2

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3 December 2017

Silvia Ortega-Gutiérrez

3

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3 December 2017

Eva de Lago

6

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María L López-Rodríguez

object named as

María L López-Rodríguez

1

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author name string

Christopher J Fowler

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3 December 2017

Gunnar Tiger

5

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3 December 2017

Javier Fernández-Ruiz

7

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3 December 2017

José A Ramos

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3 December 2017

publication date

1 April 2003

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European Journal of Medicinal Chemistry

3 December 2017

published in

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3 December 2017

volume

38

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3 December 2017

issue

4

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3 December 2017

page(s)

403-412

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Isolation, Structure, and Partial Synthesis of an Active Constituent of Hashish

3 December 2017

cites work

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The neurobiology and evolution of cannabinoid signalling

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Cannabinoid receptor ligands: clinical and neuropharmacological considerations, relevant to future drug discovery and development

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7 January 2021

Structure of a cannabinoid receptor and functional expression of the cloned cDNA

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7 January 2021

Molecular characterization of a peripheral receptor for cannabinoids

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7 January 2021

Isolation and structure of a brain constituent that binds to the cannabinoid receptor

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7 January 2021

2-Arachidonoylglycerol: a possible endogenous cannabinoid receptor ligand in brain

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7 January 2021

2-arachidonyl glyceryl ether, an endogenous agonist of the cannabinoid CB1 receptor

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7 January 2021

Characterization of a novel endocannabinoid, virodhamine, with antagonist activity at the CB1 receptor

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7 January 2021

Functional role of high-affinity anandamide transport, as revealed by selective inhibition

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7 January 2021

The fatty acid amide hydrolase (FAAH).

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7 January 2021

The endogenous cannabinoid system and brain development

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7 January 2021

Endogenous cannabinoids mediate retrograde signalling at hippocampal synapses

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7 January 2021

Leptin-regulated endocannabinoids are involved in maintaining food intake

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7 January 2021

The endocannabinoid system: a physiological perspective on its role in psychomotor control

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7 January 2021

Endocannabinoids and fatty acid amides in cancer, inflammation and related disorders

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Bidirectional control of airway responsiveness by endogenous cannabinoids

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7 January 2021

Cannabinoids control spasticity and tremor in a multiple sclerosis model

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7 January 2021

Anti-tumoral action of cannabinoids: involvement of sustained ceramide accumulation and extracellular signal-regulated kinase activation

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7 January 2021

Cannabinoids and brain injury: therapeutic implications

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7 January 2021

Endocannabinoids control spasticity in a multiple sclerosis model

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7 January 2021

Alleviation of motor hyperactivity and neurochemical deficits by endocannabinoid uptake inhibition in a rat model of Huntington's disease.

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7 January 2021

Structural determinants for recognition and translocation by the anandamide transporter

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7 January 2021

Structure-activity relationships among N-arachidonylethanolamine (Anandamide) head group analogues for the anandamide transporter

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7 January 2021

Overlap between the ligand recognition properties of the anandamide transporter and the VR1 vanilloid receptor: inhibitors of anandamide uptake with negligible capsaicin-like activity

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7 January 2021

The anandamide transport inhibitor AM404 activates vanilloid receptors.

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7 January 2021

Anandamide: an endogenous activator of the vanilloid receptor

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7 January 2021

Design, synthesis and biological evaluation of novel arachidonic acid derivatives as highly potent and selective endocannabinoid transporter inhibitors.

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7 January 2021

UCM707, a potent and selective inhibitor of endocannabinoid uptake, potentiates hypokinetic and antinociceptive effects of anandamide

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7 January 2021

2-amino-4H-3,1-benzoxazin-4-ones as inhibitors of C1r serine protease

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7 January 2021

A New synthesis of 4,5,6,7-tetrahydrofuro[2,3-c]pyridines and furo[2,3-c]pyrrolidines

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7 January 2021

Synthesis and evaluation of radioiodinated 2-(2(RS)-aminopropyl)-5-iodothiophenes as brain imaging agents

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7 January 2021

Proteins regulating the biosynthesis and inactivation of neuromodulatory fatty acid amides

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7 January 2021

The cellular uptake of anandamide is coupled to its breakdown by fatty-acid amide hydrolase

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7 January 2021

A non-pungent triprenyl phenol of fungal origin, scutigeral, stimulates rat dorsal root ganglion neurons via interaction at vanilloid receptors

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7 January 2021

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

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7 January 2021

Arachidonoyl ethanolamide-[1,2-14C] as a substrate for anandamide amidase.

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7 January 2021

Effects of homologues and analogues of palmitoylethanolamide upon the inactivation of the endocannabinoid anandamide

1 reference

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7 January 2021

Extrapyramidal and neuroendocrine effects of AM404, an inhibitor of the carrier-mediated transport of anandamide

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7 January 2021

Nefopam reduces thermal hypersensitivity in acute and postoperative pain models in the rat.

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7 January 2021

10.1016/S0223-5234(03)00045-X

Identifiers

DOI

1 reference

3 December 2017

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