(Q44466648)

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Synthesis of a [6-pyridinyl-18F]-labelled fluoro derivative of WAY-100635 as a candidate radioligand for brain 5-HT1A receptor imaging with PET.

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Europe PubMed Central

PubMed publication ID

3 December 2017

Synthesis of a [6-pyridinyl-18F]-labelled fluoro derivative of WAY-100635 as a candidate radioligand for brain 5-HT1A receptor imaging with PET. (English)

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

Christer Halldin

6

object named as

Christer Halldin

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

author name string

Mylène Karramkam

1

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

Françoise Hinnen

2

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

Myriam Berrehouma

3

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

Christophe Hlavacek

4

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

Françoise Vaufrey

5

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

Julie A McCarron

7

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

Victor W Pike

8

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

Frédéric Dollé

9

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

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publication date

1 July 2003

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Europe PubMed Central

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3 December 2017

Bioorganic & Medicinal Chemistry

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Europe PubMed Central

PubMed publication ID

3 December 2017

11

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Europe PubMed Central

PubMed publication ID

3 December 2017

13

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

2769-2782

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Europe PubMed Central

PubMed publication ID

3 December 2017

Brain Serotonin1A Receptor Binding Measured by Positron Emission Tomography With [11C]WAY-100635

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Pindolol binding to 5-HT1A receptors in the human brain confirmed with positron emission tomography

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Pindolol augmentation of selective serotonin reuptake inhibitors: PET evidence that the dose used in clinical trials is too low.

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Evaluation of EMD 128 130 occupancy of the 5-HT1A and the D2 receptor: a human PET study with [11C]WAY-100635 and [11C]raclopride

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PET-Determination of robalzotan (NAD-299) induced 5-HT(1A) receptor occupancy in the monkey brain

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Exquisite delineation of 5-HT1A receptors in human brain with PET and [carbonyl-11C]WAY-100635

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PET-characterization of [carbonyl-11C]WAY-100635 binding to 5-HT1A receptors in the primate brain.

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Radioligands for the study of brain 5-HT1A receptors in vivo.

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Characterisation of the appearance of radioactive metabolites in monkey and human plasma from the 5-HT1A receptor radioligand, [carbonyl-11C]WAY-100635--explanation of high signal contrast in PET and an aid to biomathematical modelling.

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PET evaluation of [(18)F]FCWAY, an analog of the 5-HT(1A) receptor antagonist, WAY-100635.

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Development of fluorine-18-labeled 5-HT1A antagonists

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High-yield radiosynthesis and preliminary in vivo evaluation of p-[18F]MPPF, a fluoro analog of WAY-100635.

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[18F]p-MPPF: A Radiolabeled Antagonist for the Study of 5-HT1A Receptors with PET

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Tissue distribution, autoradiography, and metabolism of 4-(2'-methoxyphenyl)-1-[2' -[N-2"-pyridinyl)-p-[(18)F]fluorobenzamido]ethyl]piperazine (p-[(18)F]MPPF), a new serotonin 5-HT(1A) antagonist for positron emission tomography: An In vivo study in

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Quantitative imaging of 5-HT(1A) receptor binding in healthy volunteers with [(18)f]p-MPPF

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7 January 2021

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In vivo characterization of p-[(18)F]MPPF, a fluoro analog of WAY-100635 for visualization of 5-HT(1a) receptors

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Quantifying drug-related 5-HT1A receptor occupancy with

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Modeling [18 F]MPPF positron emission tomography kinetics for the determination of 5-hydroxytryptamine(1A) receptor concentration with multiinjection.

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Effect of endogenous serotonin on the binding of the 5-hT1A PET ligand 18F-MPPF in the rat hippocampus: kinetic beta measurements combined with microdialysis

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7 January 2021

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Short and efficient syntheses of analogues of WAY-100635: new and potent 5-HT1A receptor antagonists

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7 January 2021

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New halogenated [11C]WAY analogues, [11C]6FPWAY and [11C]6BPWAY--radiosynthesis and assessment as radioligands for the study of brain 5-HT1A receptors in living monkey

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7 January 2021

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Mapping nicotinic acetylcholine receptors with PET.

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Synthesis of a fluorine-18 labeled derivative of epibatidine for in vivo nicotinic acetylcholine receptor PET imaging

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Synthesis and nicotinic acetylcholine receptor binding properties of exo-2-(2'-fluoro-5'-pyridinyl)-7-azabicyclo-[2.2.1]heptane: a new positron emission tomography ligand for nicotinic receptors.

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Synthesis and nicotinic acetylcholine receptor in vivo binding properties of 2-fluoro-3-[2(S)-2-azetidinylmethoxy]pyridine: a new positron emission tomography ligand for nicotinic receptors

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1-Polyfluoroalkylbenzodiazepines; 1

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Stereochemical influence on the stability of radio-metal complexes in vivo. Synthesis and evaluation of the four stereoisomers of 2-(p-nitrobenzyl)-trans-CyDTPA

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Identifiers

10.1016/S0968-0896(03)00225-6

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

3 December 2017

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