(Q44570479)

4 December 2017

title

Synthesis and structure-activity relationships of 1-arylmethyl-3-(2-aminopropyl)-5-aryl-6-methyluracils as potent GnRH receptor antagonists (English)

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4 December 2017

Zhiqiang Guo

1

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4 December 2017

Yun-Fei Zhu

2

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4 December 2017

Fabio C Tucci

3

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4 December 2017

Yinghong Gao

4

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4 December 2017

R Scott Struthers

5

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4 December 2017

John Saunders

6

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4 December 2017

Timothy D Gross

7

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4 December 2017

Qiu Xie

8

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4 December 2017

Greg J Reinhart

9

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4 December 2017

Chen Chen

10

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4 December 2017

language of work or name

English

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publication date

1 October 2003

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Bioorganic & Medicinal Chemistry Letters

4 December 2017

published in

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4 December 2017

volume

13

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4 December 2017

issue

19

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4 December 2017

page(s)

3311-3315

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Gonadotropin-releasing-hormone-receptor antagonists

4 December 2017

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Structure of the porcine LH- and FSH-releasing hormone. I. The proposed amino acid sequence

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Purification, amino acid composition and N-terminus of the hypothalamic luteinizing hormone releasing factor (LRF) of ovine origin

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Synthetic analogs of luteinizing hormone releasing hormone (LH-RH) substituted in position 6 and 10.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Discovery of a novel, potent, and orally active nonpeptide antagonist of the human luteinizing hormone-releasing hormone (LHRH) receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Orally bioavailable, indole-based nonpeptide GnRH receptor antagonists with high potency and functional activity

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Substituted indole-5-carboxamides and -acetamides as potent nonpeptide GnRH receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Potent nonpeptide GnRH receptor antagonists derived from substituted indole-5-carboxamides and -acetamides bearing a pyridine side-chain terminus

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Initial structure-activity relationship of a novel class of nonpeptidyl GnRH receptor antagonists: 2-arylindoles

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

SAR studies of novel 5-substituted 2-arylindoles as nonpeptidyl GnRH receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Initial structure-activity relationship studies of a novel series of pyrrolo[1,2-a]pyrimid-7-ones as GnRH receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

A novel synthesis of 2-arylpyrrolo[1,2-a]pyrimid-7-ones and their structure-activity relationships as potent GnRH receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Synthesis and initial structure-activity relationships of a novel series of imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Design, synthesis and structure-activity relationships of novel imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Design and Structure−Activity Relationships of 2-Alkyl-3-aminomethyl-6-(3-methoxyphenyl)-7-methyl-8-(2-fluorobenzyl)imidazolo[1,2-a]pyrimid-5-ones as Potent GnRH Receptor Antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Identification of 1-Arylmethyl-3- (2-aminoethyl)-5-aryluracil as Novel Gonadotropin-Releasing Hormone Receptor Antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

Synthesis and structure-activity relationships of deazaxanthines: analogs of potent A1- and A2-adenosine receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900620-6

7 January 2021

10.1016/S0960-894X(03)00620-6

Identifiers

DOI

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4 December 2017

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