(Q44650646)

English

Pharmacological and Genetic Characterization of Two Selective Serotonin Transporter Ligands: 2-[2-(Dimethylaminomethylphenylthio)]-5-fluoromethylphenylamine (AFM) and 3-Amino-4-[2-(dimethylaminomethyl-phenylthio)]benzonitrile (DASB)

scientific article published on November 10, 2003

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scholarly article

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Europe PubMed Central

PubMed publication ID

5 December 2017

Pharmacological and Genetic Characterization of Two Selective Serotonin Transporter Ligands: 2-[2-(Dimethylaminomethylphenylthio)]-5-fluoromethylphenylamine (AFM) and 3-Amino-4-[2-(dimethylaminomethyl-phenylthio)]benzonitrile (DASB) (English)

1 reference

10.1124/JPET.103.058636

https://api.crossref.org/works/10.1124/JPET.103.058636

31 March 2024

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nerve tissue protein

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14610240

31 March 2024

1 reference

10.1124/JPET.103.058636

https://api.crossref.org/works/10.1124/JPET.103.058636

31 March 2024

molecular medicine

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10.1124/JPET.103.058636

https://api.crossref.org/works/10.1124/JPET.103.058636

31 March 2024

author name string

Qian Li

1

1 reference

Europe PubMed Central

PubMed publication ID

5 December 2017

Li Ma

2

1 reference

Europe PubMed Central

PubMed publication ID

5 December 2017

Nicholas Seneca

4

1 reference

Europe PubMed Central

PubMed publication ID

5 December 2017

Masanori Ichise

5

1 reference

Europe PubMed Central

PubMed publication ID

5 December 2017

Henry Huang

6

1 reference

Europe PubMed Central

PubMed publication ID

5 December 2017

Marc Laruelle

7

1 reference

Europe PubMed Central

PubMed publication ID

5 December 2017

Robert B. Innis

3

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14610240

31 March 2024

Dennis L. Murphy

8

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14610240

31 March 2024

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publication date

10 November 2003

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PubMed publication ID

5 December 2017

full work available at URL

https://syndication.highwire.org/content/doi/10.1124/jpet.103.058636

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10.1124/JPET.103.058636

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31 March 2024

Journal of Pharmacology and Experimental Therapeutics

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5 December 2017

308

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5 December 2017

2

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5 December 2017

481-486

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Europe PubMed Central

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5 December 2017

Pharmacologic profile of MDMA (3,4-methylenedioxymethamphetamine) at various brain recognition sites

1

1 reference

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Functional consequences of central serotonin depletion produced by repeated fenfluramine administration in rats.

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High-affinity binding of [125I]RTI-55 to dopamine and serotonin transporters in rat brain

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Comparative affinity of duloxetine and venlafaxine for serotonin and norepinephrine transporters in vitro and in vivo, human serotonin receptor subtypes, and other neuronal receptors

5

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Influence of life stress on depression: moderation by a polymorphism in the 5-HTT gene

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Further evidence of Ca(2+)-dependent, exocytotic-like serotonin release induced by D-fenfluramine

7

1 reference

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Carrier-mediated serotonin release induced by d-fenfluramine: studies with human neuroblastoma cells transfected with a rat serotonin transporter

8

1 reference

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31 March 2024

Importance of duration of drug action in the antagonism of p-chloroamphetamine depletion of brain serotonin—comparison of fluoxetine and chlorimipramine

11

1 reference

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31 March 2024

[11C]-DASB, a tool for in vivo measurement of SSRI-induced occupancy of the serotonin transporter: PET characterization and evaluation in cats

12

1 reference

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31 March 2024

Imaging the serotonin transporter with positron emission tomography: initial human studies with [11C]DAPP and [11C]DASB.

13

1 reference

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31 March 2024

Regulation of high- and low-affinity [3H]imipramine recognition sites in rat brain by chronic treatment with antidepressants

14

1 reference

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31 March 2024

Comparative evaluation in nonhuman primates of five PET radiotracers for imaging the serotonin transporters: [11C]McN 5652, [11C]ADAM, [11C]DASB, [11C]DAPA, and [11C]AFM.

16

1 reference

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31 March 2024

Synthesis and pharmacological characterization of a new PET ligand for the serotonin transporter: [11C]5-bromo-2-[2-(dimethylaminomethylphenylsulfanyl)]phenylamine ([11C]DAPA).

17

1 reference

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Chirality and drugs used in psychiatry: nice to know or need to know?

18

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Association of anxiety-related traits with a polymorphism in the serotonin transporter gene regulatory region

19

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Carrier-mediated release of neurotransmitters

20

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Endocrine and receptor pharmacology of serotonergic anxiolytics, antipsychotics and antidepressants

21

1 reference

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Fluoxetine gradually increases [125I]DOI-labelled 5-HT2A/2C receptors in the hypothalamus without changing the levels of Gq- and G11-proteins

22

1 reference

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Protein measurement with the Folin phenol reagent

23

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Genetic perspectives on the serotonin transporter

25

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Interactions of selective serotonin reuptake inhibitors with the serotonin 5-HT2c receptor

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Applications of positron emission tomography in psychiatry

28

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Serotonin releasing agents. Neurochemical, therapeutic and adverse effects

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p-Chloroamphetamine induces serotonin release through serotonin transporters

30

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31 March 2024

Molecular Pharmacology

31

43

271

publication date

1993

1 reference

10.1124/JPET.103.058636

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31 March 2024

Biological Psychiatry

33

35

644

publication date

1994

1 reference

10.1124/JPET.103.058636

https://api.crossref.org/works/10.1124/JPET.103.058636

31 March 2024

In vitro and in vivo characterisation of [11C]-DASB: a probe for in vivo measurements of the serotonin transporter by positron emission tomography.

34

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Novel radiotracers for imaging the serotonin transporter by positron emission tomography: synthesis, radiosynthesis, and in vitro and ex vivo evaluation of (11)C-labeled 2-(phenylthio)araalkylamines

35

1 reference

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Prozac (fluoxetine, Lilly 110140), the first selective serotonin uptake inhibitor and an antidepressant drug: twenty years since its first publication

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31 March 2024

Identifiers

10.1124/JPET.103.058636

1 reference

Europe PubMed Central

PubMed publication ID

5 December 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

5 December 2017

ResearchGate publication ID

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