(Q45059765)

9 December 2017

title

Binding mode of TMC-95A analogues to eukaryotic 20S proteasome (English)

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9 December 2017

3

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9 December 2017

9

Robert Huber

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9 December 2017

Markus Kaiser

1

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9 December 2017

Michael Groll

2

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9 December 2017

Irmgard Assfalg-Machleidt

4

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9 December 2017

Elisabeth Weyher

5

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9 December 2017

Jun Kohno

6

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9 December 2017

Alexander G Milbradt

7

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9 December 2017

Christian Renner

8

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9 December 2017

Luis Moroder

10

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9 December 2017

publication date

1 September 2004

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9 December 2017

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9 December 2017

volume

5

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9 December 2017

issue

9

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9 December 2017

page(s)

1256-1266

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Degradation of cell proteins and the generation of MHC class I-presented peptides

9 December 2017

cites work

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Proteasome inhibition: a novel approach to cancer therapy

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Crystal structure of the 20S proteasome from the archaeon T. acidophilum at 3.4 A resolution

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Structure of 20S proteasome from yeast at 2.4 A resolution

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A gated channel into the proteasome core particle

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Molecular shredders: how proteasomes fulfill their role

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The active sites of the eukaryotic 20 S proteasome and their involvement in subunit precursor processing

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Cleavage motifs of the yeast 20S proteasome beta subunits deduced from digests of enolase 1.

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The catalytic sites of 20S proteasomes and their role in subunit maturation: a mutational and crystallographic study

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Catalytic activities of the 20 S proteasome, a multicatalytic proteinase complex

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Crystal structure of the 20 S proteasome:TMC-95A complex: a non-covalent proteasome inhibitor

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Probing structural determinants distal to the site of hydrolysis that control substrate specificity of the 20S proteasome.

21 January 2018

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The ubiquitin-proteasome pathway and proteasome inhibitors

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Not just research tools--proteasome inhibitors offer therapeutic promise

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A new structural class of selective and non-covalent inhibitors of the chymotrypsin-like activity of the 20S proteasome

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Structure-based optimisation of 2-aminobenzylstatine derivatives: potent and selective inhibitors of the chymotrypsin-like activity of the human 20S proteasome

21 January 2018

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The core structure of TMC-95A is a promising lead for reversible proteasome inhibition

21 January 2018

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Inhibitors of the proteasome block the degradation of most cell proteins and the generation of peptides presented on MHC class I molecules

21 January 2018

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Substrate binding and sequence preference of the proteasome revealed by active-site-directed affinity probes

21 January 2018

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Synthesis of beta-(1-azulenyl)-L-alanine as a potential blue-colored fluorescent tryptophan analog and its use in peptide synthesis

21 January 2018

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The total synthesis of proteasome inhibitors TMC-95A and TMC-95B: discovery of a new method to generate cis-propenyl amides

21 January 2018

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Simplified synthetic TMC-95A/B analogues retain the potency of proteasome inhibitory activity

21 January 2018

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The structure of the mammalian 20S proteasome at 2.75 A resolution

21 January 2018

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The Entropic Cost of Bound Water in Crystals and Biomolecules

21 January 2018

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Structure and energetics of ligand binding to proteins: Escherichia coli dihydrofolate reductase-trimethoprim, a drug-receptor system.

21 January 2018

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Structure of form III crystals of bovine pancreatic trypsin inhibitor

21 January 2018

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TMC-95A analogues with endocyclic biphenyl ether group as proteasome inhibitors.

21 January 2018

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Protein secondary structure templates derived from bioactive natural products. Combinatorial chemistry meets structure-based design

21 January 2018

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Determination of three-dimensional structures of proteins from interproton distance data by dynamical simulated annealing from a random array of atoms. Circumventing problems associated with folding

21 January 2018

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https://api.crossref.org/works/10.1002%2FCBIC.200400096

Epitope tagging of yeast genes using a PCR-based strategy: more tags and improved practical routines

21 January 2018

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High efficiency transformation of intact yeast cells using single stranded nucleic acids as a carrier

21 January 2018

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Crystallography & NMR System: A New Software Suite for Macromolecular Structure Determination

21 January 2018

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TMC-95A, B, C, and D, novel proteasome inhibitors produced by Apiospora montagnei Sacc. TC 1093. Taxonomy, production, isolation, and biological activities.

21 January 2018

1 reference

12 April 2024

https://opencitations.net/index/api/v1/citations/10.7164/ANTIBIOTICS.53.105

Identifiers

DOI

10.1002/CBIC.200400096

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9 December 2017

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