(Q45579688)

English

Discovery of N-benzyl-2-[(4S)-4-(1H-indol-3-ylmethyl)-5-oxo-1-phenyl-4,5-dihydro-6H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-6-yl]-N-isopropylacetamide, an orally active, gut-selective CCK1 receptor agonist for the potential treatment of obesity

scientific article published on 28 September 2010

Statements

Discovery of N-benzyl-2-[(4S)-4-(1H-indol-3-ylmethyl)-5-oxo-1-phenyl-4,5-dihydro-6H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-6-yl]-N-isopropylacetamide, an orally active, gut-selective CCK1 receptor agonist for the potential treatment of obesity (English)
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Richard L Elliott
Kimberly O Cameron
Janice E Chin
Jeremy A Bartlett
Elena E Beretta
Yue Chen
Paul Da Silva Jardine
Jeffrey S Dubins
Melissa L Gillaspy
Diane M Hargrove
Amit S Kalgutkar
Janet A LaFlamme
Mary E Lame
Kelly A Martin
Tristan S Maurer
Nancy A Nardone
Robert M Oliver
Dexue Sun
Andrew G Swick
Catherine E Trebino
Yingxin Zhang
28 September 2010
6797-6801

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