(Q46077676)

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Analytical method for simultaneously measuring ex vivo drug receptor occupancy and dissociation rate: application to (R)-dimethindene occupancy of central histamine H1 receptors.

scientific article published in January 2009

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scholarly article

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

Analytical method for simultaneously measuring ex vivo drug receptor occupancy and dissociation rate: application to (R)-dimethindene occupancy of central histamine H1 receptors (English)

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

Lisa M Hernández

2

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

author name string

Siobhan Malany

1

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

William F Smith

3

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

Paul D Crowe

4

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

Sam R J Hoare

5

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

publication date

1 January 2009

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

Journal of Receptors and Signal Transduction

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

29

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

2

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24 January 2020

84-93

1 reference

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24 January 2020

Drug-target residence time and its implications for lead optimization

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Models and methods for studying insurmountable antagonism

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Slow antagonist dissociation and long-lasting in vivo receptor protection

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Quantifying the association and dissociation rates of unlabelled antagonists at the muscarinic M3 receptor.

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Kinetics of nonpeptide antagonist binding to the human gonadotropin-releasing hormone receptor: Implications for structure-activity relationships and insurmountable antagonism

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Changes in pH differently affect the binding properties of histamine H1 receptor antagonists

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Structure-activity relationships of dimethindene derivatives as new M2-selective muscarinic receptor antagonists

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

3HDoxepin interactions with histamine H1-receptors and other sites in guinea pig and rat brain homogenates

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Histamine H1 receptors in human brain labelled with [3H]Doxepin

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Sedation and histamine H1-receptor antagonism: studies in man with the enantiomers of chlorpheniramine and dimethindene

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

A review of the evidence from comparative studies of levocetirizine and desloratadine for the symptoms of allergic rhinitis

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Biochemical characterization of desloratadine, a potent antagonist of the human histamine H(1) receptor

1 reference

https://api.crossref.org/works/10.1080%2F10799890902721339

21 January 2018

Identifiers

10.1080/10799890902721339

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19308787%20AND%20SRC:MED&resulttype=core&format=json

24 January 2020

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