(Q46354297)

21 December 2017

title

Binding of the novel radioligand [(3)H]UFP-101 to recombinant human and native rat nociceptin/orphanin FQ receptors (English)

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21 December 2017

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5

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21 December 2017

author name string

Massimo Ibba

1

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21 December 2017

Masato Kitayama

2

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21 December 2017

John McDonald

3

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21 December 2017

Girolamo Calo

4

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21 December 2017

Judit Farkas

6

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21 December 2017

Geza Toth

7

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21 December 2017

David G Lambert

8

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21 December 2017

publication date

21 September 2008

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21 December 2017

Naunyn-Schmiedeberg's Archives of Pharmacology

published in

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21 December 2017

volume

378

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21 December 2017

issue

6

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21 December 2017

page(s)

553-561

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21 December 2017

UFP-101, a peptide antagonist selective for the nociceptin/orphanin FQ receptor.

cites work

1 reference

Crossref

https://api.crossref.org/works/10.1007%2FS00210-008-0350-3

Binding of dynorphin A and related peptides to kappa- and mu-opioid receptors: sensitivity to Na+ ions and Gpp(NH)p

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1007%2FS00210-008-0350-3

Nociceptin/orphanin FQ and its receptor--potential targets for pain therapy?

21 January 2018

1 reference

12 December 2020

UFP-101, a high affinity antagonist for the nociceptin/orphanin FQ receptor: radioligand and GTPgamma(35)S binding studies.

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12 December 2020

Highly potent nociceptin analog containing the Arg-Lys triple repeat

1 reference

12 December 2020

Cellular actions of nociceptin: transduction mechanisms.

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12 December 2020

N- and C-terminal modifications of nociceptin/orphanin FQ generate highly potent NOP receptor ligands.

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12 December 2020

Orphanin FQ/nociceptin receptor binding studies

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12 December 2020

Nociceptin receptor binding in mouse forebrain membranes: thermodynamic characteristics and structure activity relationships

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12 December 2020

Fluorescent labeling of purified beta 2 adrenergic receptor. Evidence for ligand-specific conformational changes

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12 December 2020

[Nphe1,Arg14,Lys15]nociceptin-NH2, a novel potent and selective antagonist of the nociceptin/orphanin FQ receptor.

1 reference

12 December 2020

Comparison of the binding of [(3)H]nociceptin/orphaninFQ(1-13)NH(2), [(3)H]nociceptin/orphaninFQ(1-17)OH and [(125)I]Tyr(14)nociceptin/orphaninFQ(1-17)OH to recombinant human and native rat cerebrocortical nociceptin/orphanin FQ receptors.

1 reference

12 December 2020

Nociceptin/orphanin FQ peptide receptors: pharmacology and clinical implications

1 reference

12 December 2020

[Arg(14),Lys(15)]nociceptin, a highly potent agonist of the nociceptin/orphanin FQ receptor: in vitro and in vivo studies

1 reference

12 December 2020

Interaction of [3H]orphanin FQ and 125I-Tyr14-orphanin FQ with the orphanin FQ receptor: kinetics and modulation by cations and guanine nucleotides

1 reference

12 December 2020

Opiate agonists and antagonists discriminated by receptor binding in brain

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12 December 2020

Isolation and structure of the endogenous agonist of opioid receptor-like ORL1 receptor

1 reference

12 December 2020

Nociceptin (orphanin FQ): high-affinity and high-capacity binding site coupled to low-potency stimulation of guanylyl-5'-O-(gamma-thio)-triphosphate binding in rat brain membranes

1 reference

12 December 2020

Cardiac muscarinic cholinergic receptor binding is regulated by Na+ and guanyl nucleotides

1 reference

12 December 2020

Orphanin FQ: a neuropeptide that activates an opioidlike G protein-coupled receptor.

1 reference

12 December 2020

A single residue, aspartic acid 95, in the delta opioid receptor specifies selective high affinity agonist binding.

1 reference

12 December 2020

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

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12 December 2020

The nociceptin/orphanin FQ receptor: a target with broad therapeutic potential

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12 December 2020

Pharmacological profile of the cyclic nociceptin/orphanin FQ analogues c[Cys10,14]N/OFQ(1-14)NH2 and c[Nphe1,Cys10,14]N/OFQ(1-14)NH2.

1 reference

12 December 2020

An aspartate conserved among G-protein receptors confers allosteric regulation of alpha 2-adrenergic receptors by sodium

1 reference

12 December 2020

The ORL1 receptor: molecular pharmacology and signalling mechanisms

1 reference

12 December 2020

Antidepressant- and anxiolytic-like effects of nociceptin/orphanin FQ receptor ligands.

1 reference

12 December 2020

Pivotal role for aspartate-80 in the regulation of dopamine D2 receptor affinity for drugs and inhibition of adenylyl cyclase

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12 December 2020

Ligand-selective receptor conformations revisited: the promise and the problem

1 reference

12 December 2020

Characterization of nociceptin/orphanin FQ binding sites in dog brain membranes

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12 December 2020

The molecular and behavioral pharmacology of the orphanin FQ/nociceptin peptide and receptor family

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12 December 2020

Identification of an achiral analogue of J-113397 as potent nociceptin/orphanin FQ receptor antagonist.

1 reference

12 December 2020

Structure-activity relationship of [Nphe1]-NC-(1-13)-NH2, a pure and selective nociceptin/orphanin FQ receptor antagonist

1 reference

12 December 2020

Protein measurement with the Folin phenol reagent

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12 December 2020

Characterization of [Nphe(1)]nociceptin(1-13)NH(2), a new selective nociceptin receptor antagonist

1 reference

12 December 2020

Reciprocal modulation of agonist and antagonist binding to muscarinic cholinergic receptor by guanine nucleotide

1 reference

12 December 2020

[3H]ac-RYYRWK-NH2, a novel specific radioligand for the nociceptin/orphanin FQ receptor.

1 reference

12 December 2020

Address and message sequences for the nociceptin receptor: a structure-activity study of nociceptin-(1-13)-peptide amide.

1 reference

12 December 2020

Pharmacology of nociceptin and its receptor: a novel therapeutic target

1 reference

12 December 2020

Functional coupling of the nociceptin/orphanin FQ receptor in dog brain membranes.

1 reference

12 December 2020

Sodium ions and GTP decrease the potency of [Nphe1]N/OFQ(1-13)NH2 in blocking nociceptin/orphanin FQ receptors coupled to cyclic AMP in N1E-115 neuroblastoma cells and rat olfactory bulb

1 reference

12 December 2020

10.1007/S00210-008-0350-3

Identifiers

DOI

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21 December 2017

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21 December 2017