(Q46482843)

22 December 2017

title

Design, synthesis, and biological evaluation of HSP90 inhibitors based on conformational analysis of radicicol and its analogues (English)

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22 December 2017

author

Nicolas Winssinger

5

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22 December 2017

Martin Karplus

4

object named as

Martin Karplus

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22 December 2017

Emilie Moulin

1

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author name string

Vincent Zoete

2

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22 December 2017

Sofia Barluenga

3

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22 December 2017

language of work or name

English

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publication date

1 May 2005

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22 December 2017

Journal of the American Chemical Society

published in

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22 December 2017

volume

127

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22 December 2017

issue

19

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22 December 2017

page(s)

6999-7004

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22 December 2017

Synthesis and activity of a new generation of ruthenium-based olefin metathesis catalysts coordinated with 1,3-dimesityl-4,5-dihydroimidazol-2-ylidene ligands

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Halohydrin and oxime derivatives of radicicol: synthesis and antitumor activities

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Polymer-assisted, multi-step solution phase synthesis and biological screening of histone deacetylase inhibitors

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The heat shock protein 90 antagonist novobiocin interacts with a previously unrecognized ATP-binding domain in the carboxyl terminus of the chaperone

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A time-resolved fluorescence resonance energy transfer-based HTS assay and a surface plasmon resonance-based binding assay for heat shock protein 90 inhibitors

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Heat shock protein 90 as a molecular target for cancer therapeutics

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Structure-activity relationships in purine-based inhibitor binding to HSP90 isoforms

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Targeting wide-range oncogenic transformation via PU24FCl, a specific inhibitor of tumor Hsp90.

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Conformational analysis of drug-like molecules bound to proteins: an extensive study of ligand reorganization upon binding

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Synthesis and antitumor activity of novel O-carbamoylmethyloxime derivatives of radicicol

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SPANphos: a C2-symmetric trans-coordinating diphosphane ligand

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Do active site conformations of small ligands correspond to low free-energy solution structures?

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The Clinical Applications of Heat Shock Protein Inhibitors in Cancer - Present and Future

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Structure and functional relationships of Hsp90.

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11 October 2022

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Development of Purine-Scaffold Small Molecule Inhibitors of Hsp90

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11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JA043101W

Evidence that the novobiocin-sensitive ATP-binding site of the heat shock protein 90 (hsp90) is necessary for its autophosphorylation

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Pochonins A-F, new antiviral and antiparasitic resorcylic acid lactones from Pochonia chlamydosporia var. catenulata

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Synthesis of Functionalized Olefins by Cross and Ring-Closing Metatheses

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Identifiers

DOI

10.1021/JA043101W

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22 December 2017

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22 December 2017