(Q46638358)

23 December 2017

title

Cyclothiazide: a subunit-specific inhibitor of GABAC receptors (English)

1 reference

23 December 2017

3

Harris Ripps

1 reference

23 December 2017

author name string

An Xie

series ordinal

1

1 reference

23 December 2017

Xiangqian Song

series ordinal

2

1 reference

23 December 2017

Haohua Qian

series ordinal

4

1 reference

23 December 2017

language of work or name

English

0 references

publication date

17 April 2008

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23 December 2017

published in

Journal of Physiology

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23 December 2017

volume

586

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23 December 2017

issue

11

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23 December 2017

page(s)

2743-2752

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23 December 2017

Streptozotocin-induced diabetes modulates GABA receptor activity of rat retinal neurons

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1 reference

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A single amino acid in the second transmembrane domain of GABA rho receptors regulates channel conductance

29 September 2018

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Rat alpha6beta2delta GABAA receptors exhibit two distinct and separable agonist affinities

29 September 2018

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Targeting AMPA receptor gating processes with allosteric modulators and mutations

29 September 2018

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Picrotoxin accelerates relaxation of GABAC receptors

29 September 2018

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Cyclothiazide potently inhibits γ-aminobutyric acid type A receptors in addition to enhancing glutamate responses

29 September 2018

1 reference

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Expression and dendritic mRNA localization of GABAC receptor rho1 and rho2 subunits in developing rat brain and spinal cord

29 September 2018

1 reference

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Mechanism of glutamate receptor desensitization

29 September 2018

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The GABAC receptors of retinal neurons

29 September 2018

1 reference

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Mechanisms underlying presynaptic facilitatory effect of cyclothiazide at the calyx of Held of juvenile rats

29 September 2018

1 reference

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Structure and function of GABA(C) receptors: a comparison of native versus recombinant receptors

29 September 2018

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A novel presynaptic inhibitory mechanism underlies paired pulse depression at a fast central synapse.

29 September 2018

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A single amino acid in the second transmembrane domain of GABA rho subunits is a determinant of the response kinetics of GABAC receptors

29 September 2018

1 reference

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The glutamate receptor ion channels

29 September 2018

1 reference

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GABAC receptor rho subunits are heterogeneously expressed in the human CNS and form homo- and heterooligomers with distinct physical properties

29 September 2018

1 reference

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Molecular and pharmacological properties of GABA-rho subunits from white perch retina

29 September 2018

1 reference

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Distribution of GABA receptor rho subunit transcripts in the rat brain

29 September 2018

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Use-dependent and use-independent blocking actions of picrotoxin and zinc at the GABAC receptor in retinal horizontal cells

29 September 2018

1 reference

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AMPA receptor flip/flop mutants affecting deactivation, desensitization, and modulation by cyclothiazide, aniracetam, and thiocyanate.

29 September 2018

1 reference

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New developments in the molecular pharmacology of alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionate and kainate receptors

29 September 2018

1 reference

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Cloning of a gamma-aminobutyric acid type C receptor subunit in rat retina with a methionine residue critical for picrotoxinin channel block

29 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2536589

A single amino acid in gamma-aminobutyric acid rho 1 receptors affects competitive and noncompetitive components of picrotoxin inhibition

29 September 2018

1 reference

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Benzothiadiazides inhibit rapid glutamate receptor desensitization and enhance glutamatergic synaptic currents.

29 September 2018

1 reference

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Modulation of AMPA/kainate receptors by analogues of diazoxide and cyclothiazide in thin slices of rat hippocampus.

29 September 2018

1 reference

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Structural determinants of allosteric regulation in alternatively spliced AMPA receptors.

29 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2536589

Desensitization of AMPA receptors upon multiquantal neurotransmitter release

29 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2536589

Asynchronous release of synaptic vesicles determines the time course of the AMPA receptor-mediated EPSC

29 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2536589

Selective modulation of desensitization at AMPA versus kainate receptors by cyclothiazide and concanavalin A.

29 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2536589

The antihypertensive effect of cyclothiazide, a double blind study

29 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/18420703

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1113/JPHYSIOL.2008.153346

1 reference

23 December 2017

PMC publication ID

2536589

0 references

1 reference

23 December 2017