(Q46890983)

26 December 2017

title

Linking agonist binding to histamine H1 receptor activation (English)

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26 December 2017

author

Leonardo Pardo

6

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26 December 2017

author name string

Aldo Jongejan

1

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26 December 2017

Martijn Bruysters

2

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26 December 2017

Juan A Ballesteros

3

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26 December 2017

Eric Haaksma

4

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26 December 2017

Remko A Bakker

5

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26 December 2017

Rob Leurs

7

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26 December 2017

publication date

19 June 2005

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26 December 2017

published in

Nature Chemical Biology

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26 December 2017

volume

1

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26 December 2017

issue

2

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26 December 2017

page(s)

98-103

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26 December 2017

https://scigraph.springernature.com/pub.10.1038/nchembio714

exact match

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Mapping the binding site pocket of the serotonin 5-Hydroxytryptamine2A receptor. Ser3.36(159) provides a second interaction site for the protonated amine of serotonin but not of lysergic acid diethylamide or bufotenin

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7 January 2021

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7 January 2021

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7 January 2021

Serine and threonine residues bend alpha-helices in the chi(1) = g(-) conformation.

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7 January 2021

Modifications of vectors pEF-BOS, pcDNA1 and pcDNA3 result in improved convenience and expression

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7 January 2021

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7 January 2021

Identifiers

DOI

10.1038/NCHEMBIO714

1 reference

26 December 2017

PubMed ID

16408006

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26 December 2017