(Q47111058)

http://europepmc.org/abstract/PMC/5642017

8 January 2018

title

6-Cyano Analogues of Bedaquiline as Less Lipophilic and Potentially Safer Diarylquinolines for Tuberculosis (English)

1 reference

http://europepmc.org/abstract/PMC/5642017

8 January 2018

1 reference

1 reference

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

Daniel Conole

15

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

8

Christopher B Cooper

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

13

William A Denny

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

11

Scott G Franzblau

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

4

Hamish S Sutherland

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

1

Amy S T Tong

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

14

Brian D Palmer

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

6

Jerome Guillemont

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

7

Magali Motte

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

9

Koen Andries

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

3

Adrian Blaser

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

author name string

Sophia K Y Tsang

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

Walter Van den Broeck

10

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

Anna M Upton

12

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

publication date

22 September 2017

1 reference

http://europepmc.org/abstract/PMC/5642017

8 January 2018

published in

ACS Medicinal Chemistry Letters

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

volume

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

issue

10

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

page(s)

1019-1024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

Structure of the mycobacterial ATP synthase Fo rotor ring in complex with the anti-TB drug bedaquiline

5 June 2020

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

Bactericidal activity of pyrazinamide and clofazimine alone and in combinations with pretomanid and bedaquiline

23 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

Rifampicin and rifapentine significantly reduce concentrations of bedaquiline, a new anti-TB drug

23 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

Bedaquiline for the treatment of resistant tuberculosis: promises and pitfalls

23 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

Randomized pilot trial of eight weeks of bedaquiline (TMC207) treatment for multidrug-resistant tuberculosis: long-term outcome, tolerability, and effect on emergence of drug resistance.

23 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

Diarylquinolines, synthesis pathways and quantitative structure--activity relationship studies leading to the discovery of TMC207.

23 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

Challenges associated with current and future TB treatment

23 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

Diarylquinolines target subunit c of mycobacterial ATP synthase

23 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

QT prolongation through hERG K(+) channel blockade: current knowledge and strategies for the early prediction during drug development

23 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

Microplate alamar blue assay versus BACTEC 460 system for high-throughput screening of compounds against Mycobacterium tuberculosis and Mycobacterium avium

23 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5642017

Catalytic asymmetric synthesis of R207910

23 May 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/29057044

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ACSMEDCHEMLETT.7B00196

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29057044%20AND%20SRC:MED&resulttype=core&format=json

5 June 2020

PubMed publication ID

29057044

1 reference