(Q55715063)

22 July 2018

title

FIKK Kinase, a Ser/Thr Kinase Important to Malaria Parasites, Is Inhibited by Tyrosine Kinase Inhibitors. (English)

1 reference

22 July 2018

serine/threonine protein kinase, FIKK family

main subject

malaria

0 references

1 reference

14 December 2018

Gabriel S Brandt

10

0 references

author name string

Benjamin C Lin

1

1 reference

22 July 2018

Darcy R Harris

2

1 reference

22 July 2018

Lucy M D Kirkman

3

1 reference

22 July 2018

Astrid M Perez

4

1 reference

22 July 2018

Yiwen Qian

5

1 reference

22 July 2018

Janse T Schermerhorn

6

1 reference

22 July 2018

Min Y Hong

7

1 reference

22 July 2018

Dennis S Winston

8

1 reference

22 July 2018

Lingyin Xu

9

1 reference

22 July 2018

publication date

11 October 2017

1 reference

22 July 2018

published in

ACS Omega

1 reference

22 July 2018

volume

2

1 reference

22 July 2018

issue

10

1 reference

22 July 2018

page(s)

6605-6612

1 reference

22 July 2018

Stromal Fibroblasts from the Interface Zone of Triple Negative Breast Carcinomas Induced Epithelial-Mesenchymal Transition and its Inhibition by Emodin

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1 reference

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A novel FIKK kinase regulates the development of mosquito and liver stages of the malaria

27 July 2018

1 reference

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27 July 2018

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How Do Protein Kinases Take a Selfie (Autophosphorylate)?

27 July 2018

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27 July 2018

1 reference

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The FIKK kinase of Toxoplasma gondii is not essential for the parasite's lytic cycle

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

Classification of small molecule protein kinase inhibitors based upon the structures of their drug-enzyme complexes

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

Biochemical characterization of FIKK8--A unique protein kinase from the malaria parasite Plasmodium falciparum and other apicomplexans

27 July 2018

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The structural basis for control of eukaryotic protein kinases

27 July 2018

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Plant and animal sensors of conserved microbial signatures

27 July 2018

1 reference

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Plasmodium falciparum FIKK kinase members target distinct components of the erythrocyte membrane

27 July 2018

1 reference

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27 July 2018

1 reference

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Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum

27 July 2018

1 reference

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27 July 2018

1 reference

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Tyrphostins and other tyrosine kinase inhibitors

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

Features of selective kinase inhibitors

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

A new Apicomplexa-specific protein kinase family: multiple members in Plasmodium falciparum, all with an export signature

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

Protein kinases of the human malaria parasite Plasmodium falciparum: the kinome of a divergent eukaryote

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

Emodin, a protein tyrosine kinase inhibitor from Polygonum cuspidatum

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

Discovery and structure activity relationship of the first potent cryptosporidium FIKK kinase inhibitor.

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

A structural atlas of kinases inhibited by clinically approved drugs

12 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

An exported kinase (FIKK4.2) that mediates virulence-associated changes in Plasmodium falciparum-infected red blood cells

12 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

Dematin, a human erythrocyte cytoskeletal protein, is a substrate for a recombinant FIKK kinase from Plasmodium falciparum

12 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

Pseudokinases from a structural perspective

12 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

The evolution of protein kinase inhibitors from antagonists to agonists of cellular signaling

12 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

A novel protein kinase family in Plasmodium falciparum is differentially transcribed and secreted to various cellular compartments of the host cell

12 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

ApiDB: integrated resources for the apicomplexan bioinformatics resource center

12 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

A phosphorylation-induced conformation change in dematin headpiece.

12 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

The replacement of ATP by the competitive inhibitor emodin induces conformational modifications in the catalytic site of protein kinase CK2

12 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6044879

T7 vectors with modified T7lac promoter for expression of proteins in Escherichia coli

12 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/30023525

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Assay of protein kinases using radiolabeled ATP: a protocol

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/30023525

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ACSOMEGA.7B00997

1 reference

22 July 2018

PMC publication ID

6044879

1 reference

22 July 2018

PubMed publication ID

30023525

1 reference

22 July 2018