(Q59033724)

English

Synthesis, benzodiazepine receptor affinity and in vivo testing of 3-aryl-4,7-dihydro-6-(N1′-alkylpyrazol-3′ - or 5′-yl)pyrazolo[1,5-a]pyrimidin-7-ones

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scholarly article

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Synthesis, benzodiazepine receptor affinity and in vivo testing of 3-aryl-4,7-dihydro-6-(N1′-alkylpyrazol-3′ - or 5′-yl)pyrazolo[1,5-a]pyrimidin-7-ones (English)

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object named as

L Giusti

7

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Claudia Martini

object named as

C Martini

9

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author name string

S Selleri

1

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F Bruni

2

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A Costanzo

3

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G Guerrini

4

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M.L. Casilli

5

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C Costagli

6

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A Lucacchini

8

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P Malmberg Aiello

10

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C Lamberti

11

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publication date

December 1998

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European Journal of Medicinal Chemistry

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32

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12

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941-953

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Proconvulsant effects in baboons of β-carboline, a putative endogenous ligand for benzodiazepine receptors

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7 January 2021

based on heuristic

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2-Arylpyrazolo[4,3-c]quinolin-3-ones: a novel agonist, a partial agonist and an antagonist of benzodiazepines

1 reference

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7 January 2021

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Methyl-beta-carboline-induced convulsions are antagonized by Ro 15-1788 and by propyl-beta-carboline

1 reference

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7 January 2021

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Structure-activity relationship studies at the benzodiazepine receptor (BZR): a comparison of the substitutent effects of pyrazoloquinolinone analogs.

1 reference

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7 January 2021

based on heuristic

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Thienylpyrazoloquinolines with high affinity to benzodiazepine receptors: continuous shift from inverse agonist to agonist properties depending on the size of the alkyl substituent

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7 January 2021

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A new thienylpyrazoloquinoline: a potent and orally active inverse agonist to benzodiazepine receptors

1 reference

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7 January 2021

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The rapidly expanding range of neuronal benzodiazepine receptor ligands

1 reference

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7 January 2021

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Antagonist, partial agonist, and full agonist imidazo[1,5-a]quinoxaline amides and carbamates acting through the GABAA/benzodiazepine receptor

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7 January 2021

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Novel anxiolytics that act as partial agonists at benzodiazepine receptors

1 reference

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7 January 2021

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Inhibition of [3H]diazepam and [3H]3-carboethoxy-beta-carboline binding by irazepine: evidence for multiple "domains" of the benzodiazepine receptor

1 reference

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7 January 2021

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Synthesis of benzo-fused benzodiazepines employed as probes of the agonist pharmacophore of benzodiazepine receptors

1 reference

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7 January 2021

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Synthetic and computer assisted analysis of the pharmacophore for agonists at benzodiazepine receptors

1 reference

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7 January 2021

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The agonist pharmacophore of the benzodiazepine receptor. Synthesis of a selective anticonvulsant/anxiolytic

1 reference

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7 January 2021

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Structural requirements for agonist actions at the benzodiazepine receptor: studies with analogues of 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester

1 reference

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Synthesis of substituted 7,12-dihydropyrido[3,2-b:5,4-b']diindoles: rigid planar benzodiazepine receptor ligands with inverse agonist/antagonist properties

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Synthetic and computer-assisted analyses of the pharmacophore for the benzodiazepine receptor inverse agonist site

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2897%2989638-9

7 January 2021

based on heuristic

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Synthesis of some 2-aryl-1,2,4-triazolo[1,5-c][1,3]benzoxazin-5-ones as tools to define the essential pharmacophoric descriptors of a benzodiazepine receptor ligand

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2897%2989638-9

7 January 2021

based on heuristic

inferred from DOI database lookup

Behavioural evidence for partial agonist properties of RO 15-1788, a benzodiazepine receptor antagonist.

1 reference

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7 January 2021

based on heuristic

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Flumazenil as an anti-epileptic agent

1 reference

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7 January 2021

based on heuristic

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Anticonvulsant activity of flumazenil in rats during ontogenetic development.

1 reference

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7 January 2021

based on heuristic

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Structure-activity relationships of 1,2,4-triazolo[1,5-a] quinoxalines and their 1-deaza analogues imidazo[1,2-a]quinoxalines at the benzodiazepine receptor

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

GABA and the behavioral effects of anxiolytic drugs

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Benzodiazepine receptor ligands with positive and negative efficacy

1 reference

https://api.crossref.org/works/10.1016%2FS0223-5234%2897%2989638-9

7 January 2021

based on heuristic

inferred from DOI database lookup

A comparison of the antinociceptive responses to the GABA-receptor agonists THIP and baclofen

1 reference

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7 January 2021

based on heuristic

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Identifiers

10.1016/S0223-5234(97)89638-9

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