(Q62648677)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16489544%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

title

Development of a QSAR model for binding of tripeptides and tripeptidomimetics to the human intestinal di-/tripeptide transporter hPEPT1 (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16489544%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

0 references

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pharmaceutical science

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author

Flemming Steen Jørgensen

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16489544%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

Jon Våbenø

4

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17 January 2020

Carsten Uhd Nielsen

6

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17 January 2020

Bente Steffansen

7

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17 January 2020

author name string

Rikke Andersen

1

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16489544%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

Lars Olsen

3

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17 January 2020

Karina Thorn

5

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17 January 2020

publication date

26 February 2006

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17 January 2020

published in

Pharmaceutical Research

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17 January 2020

volume

23

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17 January 2020

issue

3

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17 January 2020

page(s)

483-492

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Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in the human intestinal Caco-2 cell line.

17 January 2020

cites work

1 reference

12 December 2020

Mechanism of intestinal absorption and renal reabsorption of an orally active ace inhibitor: uptake and transport of fosinopril in cell cultures

1 reference

12 December 2020

VolSurf: a new tool for the pharmacokinetic optimization of lead compounds

1 reference

12 December 2020

The intestinal H+/peptide symporter PEPT1: structure-affinity relationships

1 reference

12 December 2020

The role of water in sequence-independent ligand binding by an oligopeptide transporter protein

1 reference

12 December 2020

How to Make Drugs Orally Active: A Substrate Template for Peptide Transporter PepT1

1 reference

12 December 2020

Intestinal absorption of peptides

1 reference

12 December 2020

Passive and carrier-mediated intestinal absorption components of two angiotensin converting enzyme (ACE) inhibitor prodrugs in rats: enalapril and fosinopril

1 reference

12 December 2020

Expression cloning of a mammalian proton-coupled oligopeptide transporter

1 reference

12 December 2020

Color test for detection of free terminal amino groups in the solid-phase synthesis of peptides

1 reference

12 December 2020

Just add water! The effect of water on the specificity of protein-ligand binding sites and its potential application to drug design

1 reference

12 December 2020

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

12 December 2020

Predicting blood-brain barrier permeation from three-dimensional molecular structure.

1 reference

12 December 2020

Three-dimensional quantitative structure-activity relationship analyses of peptide substrates of the mammalian H+/peptide cotransporter PEPT1.

1 reference

12 December 2020

Three-dimensional quantitative structure-activity relationship analyses of beta-lactam antibiotics and tripeptides as substrates of the mammalian H+/peptide cotransporter PEPT1.

1 reference

12 December 2020

A novel inhibitor of the mammalian peptide transporter PEPT1.

1 reference

12 December 2020

Conformational restrictions in ligand binding to the human intestinal di-/tripeptide transporter: implications for design of hPEPT1 targeted prodrugs

1 reference

12 December 2020

Transport of peptidomimetic drugs by the intestinal Di/tri-peptide transporter, PepT1.

1 reference

12 December 2020

PEPT1 as a paradigm for membrane carriers that mediate electrogenic bidirectional transport of anionic, cationic, and neutral substrates

1 reference

12 December 2020

Intestinal transport of beta-lactam antibiotics: analysis of the affinity at the H+/peptide symporter (PEPT1), the uptake into Caco-2 cell monolayers and the transepithelial flux

1 reference

12 December 2020

Angiotensin-converting enzyme (ACE) inhibitor transport in human intestinal epithelial (Caco-2) cells

1 reference

12 December 2020

Model based on GRID-derived descriptors for estimating CYP3A4 enzyme stability of potential drug candidates

1 reference

12 December 2020

Molecular modeling study of structural requirements for the oligopeptide transporter

1 reference

12 December 2020

Mapping the binding site of the small intestinal peptide carrier (PepT1) using comparative molecular field analysis

1 reference

12 December 2020

Stoichiometry and pH dependence of the rabbit proton-dependent oligopeptide transporter PepT1.

1 reference

12 December 2020

Functional roles of histidine and tyrosine residues in the H(+)-peptide transporter PepT1.

1 reference

12 December 2020

10.1007/S11095-006-9462-Y

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16489544%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

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