(Q77965515)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10395100%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

title

Insurmountable angiotensin AT1 receptor antagonists: the role of tight antagonist binding (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10395100%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

author name string

F L Fierens

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10395100%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

P M Vanderheyden

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10395100%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

J P De Backer

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10395100%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

G Vauquelin

4

1 reference

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9 December 2019

publication date

1 May 1999

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10395100%20AND%20SRC:MED&resulttype=core&format=json

European Journal of Pharmacology

9 December 2019

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10395100%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

volume

372

1 reference

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9 December 2019

issue

2

1 reference

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9 December 2019

page(s)

199-206

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10395100%20AND%20SRC:MED&resulttype=core&format=json

The conformational change responsible for AT1 receptor activation is dependent upon two juxtaposed asparagine residues on transmembrane helices III and VII.

9 December 2019

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Pharmacology of LR-B/081, a new highly potent, selective and orally active, nonpeptide angiotensin II AT1 receptor antagonist

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Internalization of the rat AT1a and AT1b receptors: pharmacological and functional requirements

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Processing of angiotensin II (A-II) and (Sar1,Ala8)A-II by cultured bovine adrenocortical cells

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Dimerization of the delta opioid receptor: implication for a role in receptor internalization

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

BMS-180560, an insurmountable inhibitor of angiotensin II-stimulated responses: comparison with losartan and EXP3174.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Desensitization, two-state receptors and pharmacological parameters

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Kinetic studies on the interaction of nonlabeled antagonists with the angiotensin II receptor

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

The two-state model of receptor activation

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Evidence that the apparent complexity of receptor antagonism by angiotensin II analogues is due to a reversible and syntopic action

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Polar residues in the transmembrane domains of the type 1 angiotensin II receptor are required for binding and coupling. Reconstitution of the binding site by co-expression of two deficient mutants.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Inhibition of rabbit aortic angiotensin II (AII) receptor by CV-11974, a new nonpeptide AII antagonist

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Candesartan (CV-11974) dissociates slowly from the angiotensin AT1 receptor

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Non-peptide angiotensin agonist. Functional and molecular interaction with the AT1 receptor.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

The kinetics of action of acetylcholine antagonists in smooth muscle

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Molecular pharmacology of LR-B/081, a new non-peptide angiotensin AT1 receptor antagonist

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Pharmacological profile of GR117289 in vitro: a novel, potent and specific non-peptide angiotensin AT1 receptor antagonist

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Agonist-antagonist interactions at angiotensin receptors: application of a two-state receptor model

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Nonpeptide angiotensin II receptor antagonists

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Angiotensin II receptor subtypes

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Distinction between surmountable and insurmountable selective AT1 receptor antagonists by use of CHO-K1 cells expressing human angiotensin II AT1 receptors

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

Pharmacological characterization of the novel nonpeptide angiotensin II receptor antagonist, BIBR 277

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0014-2999%2899%2900205-8

10.1016/S0014-2999(99)00205-8

7 January 2021

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10395100%20AND%20SRC:MED&resulttype=core&format=json

9 December 2019

1 reference