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Adenophostins: High-Affinity Agonists of IP(3) Receptors
scientific article published on 25 July 2010
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Europe PubMed Central
PubMed publication ID
22353482
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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
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23 January 2020
title
Adenophostins: High-Affinity Agonists of IP(3) Receptors
(English)
1 reference
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Europe PubMed Central
PubMed publication ID
22353482
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
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23 January 2020
author
Colin W Taylor
series ordinal
4
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Europe PubMed Central
PubMed publication ID
22353482
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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
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23 January 2020
author name string
Ana M Rossi
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1
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Europe PubMed Central
PubMed publication ID
22353482
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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
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23 January 2020
Andrew M Riley
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2
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Europe PubMed Central
PubMed publication ID
22353482
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
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23 January 2020
Barry V L Potter
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3
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Europe PubMed Central
PubMed publication ID
22353482
reference URL
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23 January 2020
publication date
25 July 2010
1 reference
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Europe PubMed Central
PubMed publication ID
22353482
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
retrieved
23 January 2020
published in
Current Topics in Membranes
1 reference
stated in
Europe PubMed Central
PubMed publication ID
22353482
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
retrieved
23 January 2020
volume
66
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Europe PubMed Central
PubMed publication ID
22353482
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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
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23 January 2020
page(s)
209-233
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Europe PubMed Central
PubMed publication ID
22353482
reference URL
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23 January 2020
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Inositol 1,4,5-trisphosphate receptors are downregulated in mouse oocytes in response to sperm or adenophostin A but not to increases in intracellular Ca(2+) or egg activation.
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Binding of inositol 1,4,5-trisphosphate (IP3) and adenophostin A to the N-terminal region of the IP3 receptor: thermodynamic analysis using fluorescence polarization with a novel IP3 receptor ligand.
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Inframolecular studies of the protonation of adenophostin A: comparison with 1-D-myo-inositol 1,4,5-trisphosphate
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Evidence for the involvement of a small subregion of the endoplasmic reticulum in the inositol trisphosphate receptor-induced activation of Ca2+ inflow in rat hepatocytes
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Isoforms of the inositol 1,4,5-trisphosphate receptor are expressed in bovine oocytes and ovaries: the type-1 isoform is down-regulated by fertilization and by injection of adenophostin A.
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Down-regulation of the inositol 1,4,5-trisphosphate receptor in mouse eggs following fertilization or parthenogenetic activation
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7 January 2021
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Adenophostin A and inositol 1,4,5-trisphosphate differentially activate Cl- currents in Xenopus oocytes because of disparate Ca2+ release kinetics.
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ATP-dependent adenophostin activation of inositol 1,4,5-trisphosphate receptor channel gating: kinetic implications for the durations of calcium puffs in cells
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Disaccharide polyphosphates based upon adenophostin A activate hepatic D-myo-inositol 1,4,5-trisphosphate receptors.
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7 January 2021
based on heuristic
inferred from DOI database lookup
Rapid activation and partial inactivation of inositol trisphosphate receptors by inositol trisphosphate
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Contribution of the adenine base to the activity of adenophostin A investigated using a base replacement strategy.
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Simplification of adenophostin A defines a minimal structure for potent glucopyranoside-based mimics of D-myo-inositol 1,4,5-trisphosphate
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Cation-pi interactions in aromatics of biological and medicinal interest: electrostatic potential surfaces as a useful qualitative guide
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Functional properties of the type-3 InsP3 receptor in 16HBE14o- bronchial mucosal cells
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Synthesis of adenophostin A analogues conjugating an aromatic group at the 5'-position as potent IP3 receptor ligands.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Determinants of adenophostin A binding to inositol trisphosphate receptors
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Structural analogues of D-myo-inositol-1,4,5-trisphosphate and adenophostin A: recognition by cerebellar and platelet inositol-1,4,5-trisphosphate receptors.
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Selective recognition of inositol phosphates by subtypes of the inositol trisphosphate receptor
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Store-operated calcium channels
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Adenophostin A and ribophostin, but not inositol 1,4,5-trisphosphate or manno-adenophostin, activate the Ca2+ release-activated Ca2+ current, I(CRAC), in weak intracellular Ca2+ buffer
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
STIM1 clusters and activates CRAC channels via direct binding of a cytosolic domain to Orai1
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Clustering of InsP3 receptors by InsP3 retunes their regulation by InsP3 and Ca2+.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Synthesis and Ca2+-Mobilizing Activity of Purine-Modified Mimics of Adenophostin A: A Model for the Adenophostin−Ins(1,4,5)P3 Receptor Interaction
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Xylopyranoside-based agonists of D-myo-inositol 1,4,5-trisphosphate receptors: synthesis and effect of stereochemistry on biological activity
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Selective determinants of inositol 1,4,5-trisphosphate and adenophostin A interactions with type 1 inositol 1,4,5-trisphosphate receptors.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Synthetic partial agonists reveal key steps in IP3 receptor activation
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Adenophostin, a potent agonist of the inositol 1,4,5-trisphosphate receptor, is useful for fertilization of mouse oocytes injected with round spermatids leading to normal offspring.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Total synthesis of nucleobase-modified adenophostin A mimics
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Imaging the quantal substructure of single IP3R channel activity during Ca2+ puffs in intact mammalian cells
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Activation of IP(3) receptors by synthetic bisphosphate ligands
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Guanophostin A: Synthesis and evaluation of a high affinity agonist of the d-myo-inositol 1,4,5-trisphosphate receptor
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
2-Position base-modified analogues of adenophostin A as high-affinity agonists of the D-myo-inositol trisphosphate receptor: in vitro evaluation and molecular modeling.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Functional properties of Drosophila inositol trisphosphate receptors
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Adenophostins A and B: Potent agonists of inositol-1,4,5-trisphosphate receptor produced by Penicillium brevicompactum. Taxonomy, fermentation, isolation, physico-chemical and biological properties.
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Adenophostins A and B: potent agonists of inositol-1,4,5-trisphosphate receptor produced by Penicillium brevicompactum. Structure elucidation
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
IP(3) receptors: the search for structure.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Discrimination of intracellular calcium store subcompartments using TRPV1 (transient receptor potential channel, vanilloid subfamily member 1) release channel activity.
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Ca2+ and calmodulin differentially modulate myo-inositol 1,4, 5-trisphosphate (IP3)-binding to the recombinant ligand-binding domains of the various IP3 receptor isoforms
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
New developments in the molecular pharmacology of the myo-inositol 1,4,5-trisphosphate receptor
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reference URL
https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Role of two series of Ca2+ oscillations in activation of ascidian eggs.
1 reference
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https://api.crossref.org/works/10.1016%2FS1063-5823%2810%2966010-3
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7 January 2021
based on heuristic
inferred from DOI database lookup
Identifiers
DOI
10.1016/S1063-5823(10)66010-3
1 reference
stated in
Europe PubMed Central
PubMed publication ID
22353482
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
retrieved
23 January 2020
PubMed publication ID
22353482
1 reference
stated in
Europe PubMed Central
PubMed publication ID
22353482
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22353482%20AND%20SRC:MED&resulttype=core&format=json
retrieved
23 January 2020
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