(Q24685243)

2

0 references

Selena Schreiber

3

0 references

Mia Defino

4

0 references

Steven C Kwan

5

0 references

Shuang Li

6

0 references

Charles Chavkin

Journal of Biological Chemistry

7

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language of work or name

English

0 references

publication date

12 October 2007

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published in

0 references

volume

282

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issue

41

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page(s)

29803-11

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cites work

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7 April 2017

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Mu and kappa opioid receptors activate ERK/MAPK via different protein kinase C isoforms and secondary messengers in astrocytes

7 April 2017

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Kappa opioid receptor antagonism and prodynorphin gene disruption block stress-induced behavioral responses

7 April 2017

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Mitogenic signaling via endogenous kappa-opioid receptors in C6 glioma cells: evidence for the involvement of protein kinase C and the mitogen-activated protein kinase signaling cascade

7 April 2017

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Functional Selectivity and Classical Concepts of Quantitative Pharmacology

7 April 2017

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Differential effects of the novel kappa opioid receptor antagonist, JDTic, on reinstatement of cocaine-seeking induced by footshock stressors vs cocaine primes and its antidepressant-like effects in rats

7 April 2017

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Kappa-opioid receptor signals through Src and focal adhesion kinase to stimulate c-Jun N-terminal kinases in transfected COS-7 cells and human monocytic THP-1 cells

7 April 2017

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SP600125, an anthrapyrazolone inhibitor of Jun N-terminal kinase

7 April 2017

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Phosphorylation of a carboxyl-terminal serine within the kappa-opioid receptor produces desensitization and internalization

7 April 2017

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Ubiquitin and ubiquitin-like proteins as multifunctional signals

7 April 2017

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Convenient synthesis and in vitro pharmacological activity of 2-thioanalogs of salvinorins A and B.

9 May 2017

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Risperidone irreversibly binds to and inactivates the h5-HT7 serotonin receptor

28 September 2017

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Pharmacological properties of JDTic: a novel kappa-opioid receptor antagonist

28 September 2017

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Principles: receptor theory in pharmacology

28 September 2017

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Targeting the JNK MAPK cascade for inhibition: basic science and therapeutic potential.

28 September 2017

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Prolonged kappa opioid receptor phosphorylation mediated by G-protein receptor kinase underlies sustained analgesic tolerance

28 September 2017

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Identification of (3R)-7-hydroxy-N-((1S)-1-[[(3R,4R)-4-(3-hydroxyphenyl)- 3,4-dimethyl-1-piperidinyl]methyl]-2-methylpropyl)-1,2,3,4-tetrahydro- 3-isoquinolinecarboxamide as a novel potent and selective opioid kappa receptor antagonist.

28 September 2017

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Antidepressant-like effects of kappa-opioid receptor antagonists in the forced swim test in rats

28 September 2017

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Kappa opioid antagonist effects of the novel kappa antagonist 5'-guanidinonaltrindole (GNTI) in an assay of schedule-controlled behavior in rhesus monkeys

28 September 2017

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Identification of the first trans-(3R,4R)- dimethyl-4-(3-hydroxyphenyl)piperidine derivative to possess highly potent and selective opioid kappa receptor antagonist activity

28 September 2017

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G-protein-coupled receptors and signaling networks: emerging paradigms.

28 September 2017

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5'-Guanidinonaltrindole, a highly selective and potent kappa-opioid receptor antagonist

28 September 2017

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Intracisternal nor-binaltorphimine distinguishes central and peripheral kappa-opioid antinociception in rhesus monkeys

28 September 2017

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Pseudo-noncompetitive antagonism of M1, M3, and M5 muscarinic receptor-mediated Ca2+ mobilization by muscarinic antagonists

28 September 2017

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Opioid modulation of extracellular signal-regulated protein kinase activity is ras-dependent and involves Gbetagamma subunits

28 September 2017

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Activation of the cloned human kappa opioid receptor by agonists enhances [35S]GTPgammaS binding to membranes: determination of potencies and efficacies of ligands.

28 September 2017

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Functional analysis of cloned opioid receptors in transfected cell lines.

28 September 2017

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Reinforcing and discriminative stimulus properties of mixed agonist-antagonist opioids

28 September 2017

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Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonists

28 September 2017

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Nor-binaltorphimine, a highly selective kappa-opioid antagonist in analgesic and receptor binding assays

28 September 2017

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A peptide c-Jun N-terminal kinase (JNK) inhibitor blocks mechanical allodynia after spinal nerve ligation: respective roles of JNK activation in primary sensory neurons and spinal astrocytes for neuropathic pain development and maintenance.

28 September 2017

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Autoradiography of opioid and ORL1 ligands in opioid receptor triple knockout mice

30 May 2018

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Buprenorphine: differential interaction with opiate receptor subtypes in vivo

30 May 2018

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Dynorphin Is a Specific Endogenous Ligand of the κ Opioid Receptor

30 May 2018

1 reference

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Bimorphinans as highly selective, potent kappa opioid receptor antagonists

30 May 2018

1 reference

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Nor-binaltorphimine is a reversible, noncompetitive opioid antagonist in the mouse vas deferens with high affinity for kappa receptors in monkey brain membranes

30 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2096775

Long term kappa-opioid receptor blockade following nor-binaltorphimine

30 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2096775

Differential effects of systemically administered nor-binaltorphimine (nor-BNI) on kappa-opioid agonists in the mouse writhing assay

30 May 2018

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Retention of heroin and morphine-6 beta-glucuronide analgesia in a new line of mice lacking exon 1 of MOR-1.

21 January 2018

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Importance of phenolic address groups in opioid kappa receptor selective antagonists

21 January 2018

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Synthetic studies of neoclerodane diterpenes from Salvia divinorum: preparation and opioid receptor activity of salvinicin analogues

21 January 2018

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Synthesis and in vitro pharmacological evaluation of salvinorin A analogues modified at C(2).

21 January 2018

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Nor-binaltorphimine: an ultra-long acting kappa-opioid antagonist in pigeons

21 January 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2096775

Kappa opioid antagonist effects of systemically administered nor-binaltorphimine in a thermal antinociception assay in rhesus monkeys.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2096775

Extremely long-lasting antagonistic actions of nor-binaltorphimine (nor-BNI) in the mouse tail-flick test

28 November 2018

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