(Q27662332)

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Critical Roles of Hydrophobicity and Orientation of Side Chains for Inactivation of Sarcoplasmic Reticulum Ca2+-ATPase with Thapsigargin and Thapsigargin Analogs

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20551329%20AND%20SRC:MED&resulttype=core&format=json

5 February 2020

Critical roles of hydrophobicity and orientation of side chains for inactivation of sarcoplasmic reticulum Ca2+-ATPase with thapsigargin and thapsigargin analogs (English)

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5 February 2020

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5 February 2020

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5 February 2020

Carl Erik Olsen

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5 February 2020

Søren Brøgger Christensen

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5 February 2020

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Huizhen Liu

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5 February 2020

Yonathan Sonntag

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5 February 2020

Marc le Maire

5

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5 February 2020

Helmer Soehoel

6

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5 February 2020

Jesper V Møller

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5 February 2020

Anne-Marie L Winther

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5 February 2020

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15 June 2010

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5 February 2020

Journal of Biological Chemistry

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5 February 2020

285

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5 February 2020

37

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5 February 2020

28883-28892

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5 February 2020

Crystal structure of the sodium-potassium pump at 2.4 A resolution

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20 March 2017

Cyclopiazonic Acid Is Complexed to a Divalent Metal Ion When Bound to the Sarcoplasmic Reticulum Ca2+-ATPase

1 reference

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20 March 2017

Crystal structure of the sodium–potassium pump

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

20 March 2017

MolProbity: all-atom contacts and structure validation for proteins and nucleic acids

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

20 March 2017

Interdomain communication in calcium pump as revealed in the crystal structures with transmembrane inhibitors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

20 March 2017

The molecular basis for cyclopiazonic acid inhibition of the sarcoplasmic reticulum calcium pump

1 reference

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20 March 2017

Structural changes in the calcium pump accompanying the dissociation of calcium

1 reference

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20 March 2017

Coot: model-building tools for molecular graphics

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20 March 2017

PRODRG: a tool for high-throughput crystallography of protein-ligand complexes

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20 March 2017

Crystallography & NMR System: A New Software Suite for Macromolecular Structure Determination

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20 March 2017

Improved methods for building protein models in electron density maps and the location of errors in these models

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

20 March 2017

The versatility and universality of calcium signalling

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

7 April 2017

BAX and BAK regulation of endoplasmic reticulum Ca2+: a control point for apoptosis

1 reference

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7 April 2017

Databases in protein crystallography

1 reference

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7 April 2017

STIM and Orai: dynamic intermembrane coupling to control cellular calcium signals.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

A Trojan horse in drug development: targeting of thapsigargins towards prostate cancer cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

Crystal structure of the plasma membrane proton pump.

1 reference

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29 September 2017

Fragment-based approaches to enzyme inhibition

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

Natural products as starting materials for development of second-generation SERCA inhibitors targeted towards prostate cancer cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

Structural role of countertransport revealed in Ca(2+) pump crystal structure in the absence of Ca(2+)

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

Unlocking the secrets of cell signaling

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

The SERCA pump as a therapeutic target: making a "smart bomb" for prostate cancer

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

Lipid-protein interactions in biological membranes: a structural perspective

1 reference

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29 September 2017

Calcium signaling: a tale for all seasons

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

Specific substitutions at amino acid 256 of the sarcoplasmic/endoplasmic reticulum Ca2+ transport ATPase mediate resistance to thapsigargin in thapsigargin-resistant hamster cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

Specific and efficient peptide substrates for assaying the proteolytic activity of prostate-specific antigen.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

29 September 2017

Kinetic characterization of the normal and detergent-perturbed reaction cycles of the sarcoplasmic reticulum calcium pump. Rate-limiting step(s) under different conditions.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

2 June 2018

Characterization of the inhibition of intracellular Ca2+ transport ATPases by thapsigargin

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

2 June 2018

Enzyme kinetics and substrate stabilization of detergent-solubilized and membraneous (Ca2+ + Mg2+)-activated ATPase from sarcoplasmic reticulum. Effect of protein-protein interactions.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2937915

2 June 2018

Thapsigargin and dimethyl sulfoxide activate medium P(i)<-->HOH oxygen exchange catalyzed by sarcoplasmic reticulum Ca2+-ATPase

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M110.136242

21 January 2018

Dephosphorylation of the calcium pump coupled to counterion occlusion

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M110.136242

21 January 2018

A tool coming of age: thapsigargin as an inhibitor of sarco-endoplasmic reticulum Ca(2+)-ATPases

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M110.136242

21 January 2018

Prostate-specific antigen-activated thapsigargin prodrug as targeted therapy for prostate cancer

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M110.136242

21 January 2018

Total synthesis of two novel subpicomolar sarco/endoplasmatic reticulum Ca2+-ATPase inhibitors designed by an analysis of the binding site of thapsigargin

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M110.136242

21 January 2018

Calcium transport by sarcoplasmic reticulum Ca(2+)-ATPase. Role of the A domain and its C-terminal link with the transmembrane region.

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M110.136242

21 January 2018

Specific structural requirements for the inhibitory effect of thapsigargin on the Ca2+ ATPase SERCA.

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M110.136242

21 January 2018

Design, synthesis, and pharmacological evaluation of thapsigargin analogues for targeting apoptosis to prostatic cancer cells

1 reference

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21 January 2018

Molecular determinants of thapsigargin binding by SERCA Ca2+-ATPase: a computational docking study

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M110.136242

21 January 2018

Kinetic characterization of the perturbation by dodecylmaltoside of sarcoplasmic reticulum Ca(2+)-ATPase

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M110.136242

21 January 2018

Annular and non-annular binding sites on the (Ca2+ + Mg2+)-ATPase.

1 reference

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21 January 2018

Perturbation of the structure and function of a membranous Ca2+-ATPase by non-solubilizing concentrations of a non-ionic detergent

1 reference

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12 December 2020

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inferred from PubMed ID database lookup

Competition between cholesterol and phosphatidylcholine for the hydrophobic surface of sarcoplasmic reticulum calcium(2+) ATPase

1 reference

https://pubmed.ncbi.nlm.nih.gov/20551329

12 December 2020

based on heuristic

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Inhibition of the sarcoplasmic reticulum Ca2+ transport ATPase by thapsigargin at subnanomolar concentrations

1 reference

https://pubmed.ncbi.nlm.nih.gov/20551329

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The inhibitors thapsigargin and 2,5-di(tert-butyl)-1,4-benzohydroquinone favour the E2 form of the Ca2+,Mg(2+)-ATPase

1 reference

https://pubmed.ncbi.nlm.nih.gov/20551329

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The importance of the hydroxyl moieties for inhibition of the Ca(2+)-ATPase by trilobolide and 2,5-di(tert-butyl)-1,4-benzohydroquinone

1 reference

https://pubmed.ncbi.nlm.nih.gov/20551329

12 December 2020

based on heuristic

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Identifiers

10.1074/JBC.M110.136242

2 references

Consolidated OpenCitations Corpus – April 2017

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5 February 2020

OpenCitations bibliographic resource ID

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

PMC publication ID

2 references

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20551329%20AND%20SRC:MED&resulttype=core&format=json

5 February 2020

PubMed publication ID

2 references

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20551329%20AND%20SRC:MED&resulttype=core&format=json

5 February 2020

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