(Q27667675)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

title

Two distinct conformations of helix 6 observed in antagonist-bound structures of a beta1-adrenergic receptor (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

Christopher G. Tate

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

Gebhard Schertler

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

author name string

Rouslan Moukhametzianov

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

Patricia C Edwards

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

Maria J Serrano-Vega

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

Andrew G W Leslie

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

language of work or name

English

0 references

publication date

3 May 2011

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

Proceedings of the National Academy of Sciences of the United States of America

30 January 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

volume

108

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

page(s)

8228-8232

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

issue

20

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

Structure of the Human Dopamine D3 Receptor in Complex with a D2/D3 Selective Antagonist

30 January 2020

cites work

1 reference

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Structures of the CXCR4 chemokine GPCR with small-molecule and cyclic peptide antagonists

20 March 2017

1 reference

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Conserved Binding Mode of Human β 2 Adrenergic Receptor Inverse Agonists and Antagonist Revealed by X-ray Crystallography

20 March 2017

1 reference

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Identification of two distinct inactive conformations of the beta2-adrenergic receptor reconciles structural and biochemical observations

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist

20 March 2017

1 reference

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Crystal structure of opsin in its G-protein-interacting conformation

20 March 2017

1 reference

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Structure of a beta1-adrenergic G-protein-coupled receptor

20 March 2017

1 reference

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Crystal structure of the ligand-free G-protein-coupled receptor opsin

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

A Specific Cholesterol Binding Site Is Established by the 2.8 Å Structure of the Human β2-Adrenergic Receptor

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

High-resolution crystal structure of an engineered human beta2-adrenergic G protein-coupled receptor

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Crystal structure of the human beta2 adrenergic G-protein-coupled receptor

20 March 2017

2 references

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

20 March 2017

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Crystal structure of rhodopsin: A G protein-coupled receptor

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Phasercrystallographic software

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Scaling and assessment of data quality

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Refinement of macromolecular structures by the maximum-likelihood method

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

PHENIX: building new software for automated crystallographic structure determination

20 March 2017

2 references

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

20 March 2017

https://api.crossref.org/works/10.1073%2FPNAS.1100185108

A G protein-coupled receptor at work: the rhodopsin model.

22 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Engineering G protein-coupled receptors to facilitate their structure determination.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

High-resolution distance mapping in rhodopsin reveals the pattern of helix movement due to activation

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

New G-protein-coupled receptor crystal structures: insights and limitations

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Conformational thermostabilization of the beta1-adrenergic receptor in a detergent-resistant form

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Activation of G protein-coupled receptors

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Conformational complexity of G-protein-coupled receptors

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Constitutive activity of muscarinic acetylcholine receptors

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Recent developments in constitutive receptor activity and inverse agonism, and their potential for GPCR drug discovery

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Historical review: Negative efficacy and the constitutive activity of G-protein-coupled receptors.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

International Union of Pharmacology. XLVI. G protein-coupled receptor list.

29 September 2017

1 reference

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Structure of bovine rhodopsin in a trigonal crystal form.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Expression and purification of truncated, non-glycosylated turkey beta-adrenergic receptors for crystallization.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Activation of the beta 2-adrenergic receptor involves disruption of an ionic lock between the cytoplasmic ends of transmembrane segments 3 and 6.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Somatic mutations in the thyrotropin receptor gene cause hyperfunctioning thyroid adenomas

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Antagonists with negative intrinsic activity at delta opioid receptors coupled to GTP-binding proteins

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Constitutive activation of the alpha 1B-adrenergic receptor by all amino acid substitutions at a single site. Evidence for a region which constrains receptor activation

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

Functional role of a conserved motif in TM6 of the rat mu opioid receptor: constitutively active and inactive receptors result from substitutions of Thr6.34(279) with Lys and Asp.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3100933

The repertoire of G-protein-coupled receptors in fully sequenced genomes

2 June 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.1100185108

The retinal conformation and its environment in rhodopsin in light of a new 2.2 A crystal structure

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.1100185108

Structural biology: A moving story of receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.1100185108

Development and crystallization of a minimal thermostabilised G protein-coupled receptor.

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.1100185108

The Ile164 beta(2)-adrenoceptor polymorphism alters salmeterol exosite binding and conventional agonist coupling to G(s).

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.1100185108

Role of the third intracellular loop for the activation of gonadotropin receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.1100185108

21 January 2018

Identifiers

DOI

10.1073/PNAS.1100185108

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

0 references

release_35iv5y2ui5ehdba6qgukioedte

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/35iv5y2ui5ehdba6qgukioedte

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21540331%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

2 references