(Q27667834)

English

Discovery and characterization of small molecule inhibitors of the BET family bromodomains

scientific article

Discovery and Characterization of Small Molecule Inhibitors of the BET Family Bromodomains

In more languages

edit

Statements

instance of

scholarly article

0 references

title

Discovery and characterization of small molecule inhibitors of the BET family bromodomains (English)

0 references

12

Helen Flynn

0 references

Robert Burns Woodward

series ordinal

9

object named as

Robert Woodward

0 references

Olivier Mirguet

object named as

Olivier Mirguet

series ordinal

4

0 references

Julia H. White

series ordinal

3

object named as

Julia H White

0 references

Iain Uings

series ordinal

21

object named as

Iain J Uings

0 references

author name string

Chun-Wa Chung

series ordinal

1

0 references

Herve Coste

series ordinal

2

0 references

Jonathan Wilde

series ordinal

5

0 references

Romain L Gosmini

series ordinal

6

0 references

Chris Delves

series ordinal

7

0 references

Sylvie M Magny

series ordinal

8

0 references

Stephen A Hughes

series ordinal

10

0 references

Eric V Boursier

series ordinal

11

0 references

Anne M Bouillot

series ordinal

13

0 references

Jean-Marie G Brusq

series ordinal

15

0 references

Francoise J Gellibert

series ordinal

16

0 references

Emma J Jones

series ordinal

17

0 references

Alizon M Riou

series ordinal

18

0 references

Paul Homes

series ordinal

19

0 references

Sandrine L Martin

series ordinal

20

0 references

Jerome Toum

series ordinal

22

0 references

Catherine A Clement

series ordinal

23

0 references

Anne-Benedicte Boullay

series ordinal

24

0 references

Rachel L Grimley

series ordinal

25

0 references

Florence M Blandel

series ordinal

26

0 references

Rab K Prinjha

series ordinal

27

0 references

Kevin Lee

series ordinal

28

0 references

Jorge Kirilovsky

series ordinal

29

0 references

Edwige Nicodeme

series ordinal

30

0 references

language of work or name

English

0 references

publication date

9 June 2011

0 references

published in

Journal of Medicinal Chemistry

0 references

volume

54

0 references

issue

11

0 references

page(s)

3827-38

0 references

cites work

A quantitative high-throughput screen identifies potential epigenetic modulators of gene expression

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

The CCP4 suite: programs for protein crystallography

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Antiinflammatory properties of HDL.

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Chemical genetic modifier screens: small molecule trichostatin suppressors as probes of intracellular histone and tubulin acetylation

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Probability-based protein identification by searching sequence databases using mass spectrometry data

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Structural Basis for Acetylated Histone H4 Recognition by the Human BRD2 Bromodomain

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

The double bromodomain proteins Brd2 and Brd3 couple histone acetylation to transcription

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Coot: model-building tools for molecular graphics

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

The double bromodomain-containing chromatin adaptor Brd4 and transcriptional regulation

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Solution structure of the second bromodomain of Brd2 and its specific interaction with acetylated histone tails

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Selective small molecules blocking HIV-1 Tat and coactivator PCAF association

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

The structural basis for the recognition of acetylated histone H4 by the bromodomain of histone acetyltransferase gcn5p

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

E mu-BRD2 transgenic mice develop B-cell lymphoma and leukemia.

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

How chromatin-binding modules interpret histone modifications: lessons from professional pocket pickers

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Suppression of inflammation by a synthetic histone mimic

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Rationalizing the chemical space of protein-protein interaction inhibitors

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Epigenetics: a landscape takes shape

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Selective inhibition of BET bromodomains

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Chromatin modifications and their function

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Structures of the Dual Bromodomains of the P-TEFb-activating Protein Brd4 at Atomic Resolution

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Cooperative binding of two acetylation marks on a histone tail by a single bromodomain

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Enzymatic and structural insights for substrate specificity of a family of jumonji histone lysine demethylases

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Effect of chain length on transfection properties of spermine-based gemini surfactants

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Acetylation-dependent chromatin reorganization by BRDT, a testis-specific bromodomain-containing protein

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Crystal structure of the human BRD2 bromodomain: insights into dimerization and recognition of acetylated histone H4.

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Structure and acetyl-lysine recognition of the bromodomain

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Target structure-based discovery of small molecules that block human p53 and CREB binding protein association

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

A quantitative high-throughput screen for modulators of IL-6 signaling: a model for interrogating biological networks using chemical libraries

1 reference

11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JM200108T

Interaction of the bovine papillomavirus E2 protein with Brd4 tethers the viral DNA to host mitotic chromosomes

(Q27667834)

Discovery and characterization of small molecule inhibitors of the BET family bromodomains

Statements

Identifiers

Sitelinks

Wikipedia(0 entries)

Wikibooks(0 entries)

Wikinews(0 entries)

Wikiquote(0 entries)

Wikisource(0 entries)

Wikiversity(0 entries)

Wikivoyage(0 entries)

Wiktionary(0 entries)

Multilingual sites(0 entries)