(Q27679284)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23899692%20AND%20SRC:MED&resulttype=core&format=json

6 March 2020

title

Discovery of a potent and selective DDR1 receptor tyrosine kinase inhibitor (English)

1 reference

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6 March 2020

author name string

Hyung-Gu Kim

1

1 reference

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6 March 2020

Li Tan

2

1 reference

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6 March 2020

Ellen L Weisberg

3

1 reference

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6 March 2020

Feiyang Liu

4

1 reference

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6 March 2020

Hwan Geun Choi

6

1 reference

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6 March 2020

Scott A Ezell

7

1 reference

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6 March 2020

Hong Wu

8

1 reference

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6 March 2020

Zheng Zhao

9

1 reference

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6 March 2020

Jinhua Wang

10

1 reference

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6 March 2020

Anna Mandinova

11

1 reference

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6 March 2020

James D Griffin

12

1 reference

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6 March 2020

Alex N Bullock

13

1 reference

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6 March 2020

Qingsong Liu

14

1 reference

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6 March 2020

Sam W Lee

15

1 reference

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6 March 2020

publication date

13 August 2013

1 reference

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6 March 2020

1 reference

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6 March 2020

volume

8

1 reference

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6 March 2020

issue

10

1 reference

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6 March 2020

page(s)

2145-2150

1 reference

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Cell signaling by receptor tyrosine kinases

6 March 2020

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Expression and mutation analysis of the discoidin domain receptors 1 and 2 in non-small cell lung carcinoma

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Consistent and selective expression of the discoidin domain receptor-1 tyrosine kinase in human brain tumors

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Discoidin domain receptor 1 (DDR1) signaling in PC12 cells: activation of juxtamembrane domains in PDGFR/DDR/TrkA chimeric receptors

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Comprehensive analysis of kinase inhibitor selectivity

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Discovery and optimization of 3-(2-(Pyrazolo[1,5-a]pyrimidin-6-yl)ethynyl)benzamides as novel selective and orally bioavailable discoidin domain receptor 1 (DDR1) inhibitors

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Discoidin domain receptor tyrosine kinases: new players in cancer progression

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

DDR1 receptor tyrosine kinase promotes prosurvival pathway through Notch1 activation

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Inhibition of collagen-induced discoidin domain receptor 1 and 2 activation by imatinib, nilotinib and dasatinib

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Somatic mutations and germline sequence variants in the expressed tyrosine kinase genes of patients with de novo acute myeloid leukemia

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Overexpression of discoidin domain receptor 1 increases the migration and invasion of hepatocellular carcinoma cells in association with matrix metalloproteinase.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Quantitative chemical proteomics reveals mechanisms of action of clinical ABL kinase inhibitors

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Identification of expressed genes characterizing long-term survival in malignant glioma patients

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Somatic mutations of the protein kinase gene family in human lung cancer

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Overexpression of the cell adhesion molecules DDR1, Claudin 3, and Ep-CAM in metaplastic ovarian epithelium and ovarian cancer.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

p53 induction and activation of DDR1 kinase counteract p53-mediated apoptosis and influence p53 regulation through a positive feedback loop

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Phosphotyrosine mediated protein interactions of the discoidin domain receptor 1.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

A general framework for inhibitor resistance in protein kinases.

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Chemical proteomic profiles of the BCR-ABL inhibitors imatinib, nilotinib, and dasatinib reveal novel kinase and nonkinase targets

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

A general strategy for creating "inactive-conformation" abl inhibitors

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

Expression analysis of genes involved in brain tumor progression driven by retroviral insertional mutagenesis in mice.

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3800496

27 November 2018

Identifiers

DOI

10.1021/CB400430T

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23899692%20AND%20SRC:MED&resulttype=core&format=json

6 March 2020

1 reference

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23899692%20AND%20SRC:MED&resulttype=core&format=json

6 March 2020

PubMed publication ID

23899692

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23899692%20AND%20SRC:MED&resulttype=core&format=json