(Q27684146)

English

Novel Carboxamide-Based Allosteric MEK Inhibitors: Discovery and Optimization Efforts toward XL518 (GDC-0973)

scientific article

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Novel Carboxamide-Based Allosteric MEK Inhibitors: Discovery and Optimization Efforts toward XL518 (GDC-0973) (English)
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Kenneth D Rice
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Naing Aay
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Neel K Anand
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Charles M Blazey
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Owen J Bowles
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Joerg Bussenius
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Simona Costanzo
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Jeffry K Curtis
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Steven C Defina
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Larisa Dubenko
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Stefan Engst
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Anagha A Joshi
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Abigail R Kennedy
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Angie I Kim
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Elena S Koltun
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Julie C Lougheed
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Jean-Claire L Manalo
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Jean-Francois Martini
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John M Nuss
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Csaba J Peto
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Tsze H Tsang
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Peiwen Yu
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Stuart Johnston
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10 May 2012
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3
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5
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416-21
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