(Q27684637)

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Selective small molecule probes for the hypoxia inducible factor (HIF) prolyl hydroxylases

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Selective small molecule probes for the hypoxia inducible factor (HIF) prolyl hydroxylases (English)

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13

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Rasheduzzaman Chowdhury

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1

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Christopher J. Schofield

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18

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Nathan R Rose

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Nathan R Rose

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9

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Michael A McDonough

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Michael A McDonough

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7

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Peter J. Ratcliffe

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Peter J Ratcliffe

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17

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Ya-Min Tian

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6

object named as

Ya-Min Tian

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Christopher J A Pugh

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16

object named as

Christopher W Pugh

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Ana Conejo-García

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10

object named as

Ana Conejo-Garcia

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Kar Kheng Yeoh

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5

object named as

Kar Kheng Yeoh

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Anthony Tumber

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8

object named as

Anthony Tumber

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Mun Chiang Chan

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3

object named as

Mun Chiang Chan

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Marina Demetriades

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11

object named as

Marina Demetriades

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author name string

José Ignacio Candela-Lena

series ordinal

2

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David Jeremy Greenald

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4

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Sinnakaruppan Mathavan

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12

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Myung Kyu Lee

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14

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Freek van Eeden

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15

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publication date

19 July 2013

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published in

ACS Chemical Biology

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volume

8

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issue

7

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page(s)

1488-96

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1,3,8-Triazaspiro[4.5]decane-2,4-diones as efficacious pan-inhibitors of hypoxia-inducible factor prolyl hydroxylase 1-3 (HIF PHD1-3) for the treatment of anemia

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Dipeptidyl-quinolone derivatives inhibit hypoxia inducible factor-1α prolyl hydroxylases-1, -2, and -3 with altered selectivity.

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C. elegans EGL-9 and mammalian homologs define a family of dioxygenases that regulate HIF by prolyl hydroxylation

(Q27684637)

Selective small molecule probes for the hypoxia inducible factor (HIF) prolyl hydroxylases

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