(Q33456441)

English

Evaluation of the P-glycoprotein (Abcb1) affinity status of a series of morphine analogs: comparative study with meperidine analogs to identify opioids with minimal P-glycoprotein interactions

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

Evaluation of the P-glycoprotein (Abcb1) affinity status of a series of morphine analogs: comparative study with meperidine analogs to identify opioids with minimal P-glycoprotein interactions (English)

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

author name string

Hazem E Hassan

1

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

Susan L Mercer

2

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

Christopher W Cunningham

3

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

Andrew Coop

4

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

Natalie D Eddington

5

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

language of work or name

0 references

publication date

5 April 2009

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

International Journal of Pharmaceutics

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

375

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

1-2

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

48-54

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

Differential involvement of P-glycoprotein (ABCB1) in permeability, tissue distribution, and antinociceptive activity of methadone, buprenorphine, and diprenorphine: in vitro and in vivo evaluation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Opioids and efflux transporters. Part 1: P-glycoprotein substrate activity of N-substituted analogs of meperidine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Use of loperamide as a phenotypic probe of mdr1a status in CF-1 mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Compounds related to pethidine-IV. New general chemical methods of increasing the analgesic activity of pethidine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Role of P-glycoprotein in pharmacokinetics: clinical implications

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Passive permeability and P-glycoprotein-mediated efflux differentiate central nervous system (CNS) and non-CNS marketed drugs.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Interaction of morphine, fentanyl, sufentanil, alfentanil, and loperamide with the efflux drug transporter P-glycoprotein

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Rational use of in vitro P-glycoprotein assays in drug discovery

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Co-administration of sub-antinociceptive doses of oxycodone and morphine produces marked antinociceptive synergy with reduced CNS side-effects in rats

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

P-glycoprotein in the blood-brain barrier of mice influences the brain penetration and pharmacological activity of many drugs

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Dose-ranging study of oxycodone for chronic pain in advanced cancer

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Biochemistry of multidrug resistance mediated by the multidrug transporter

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Absence of the mdr1a P-Glycoprotein in mice affects tissue distribution and pharmacokinetics of dexamethasone, digoxin, and cyclosporin A.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Novel analgesics and molecular rearrangements in the morphine-thebaine group. II. Alcohols derived from 6,14-endo-etheno- and 6,14-endo-ethanotetrahydrothebaine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Multidrug resistance gene family and chemical carcinogens

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Deoxymorphines: role of the phenolic hydroxyl in antinociception and opiate receptor interactions

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Studies in the (+)-morphinan series. 5. Synthesis and biological properties of (+)-naloxone

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Comparisons of the Analgesic Effects of Oral and Intramuscular Oxymorphone and of Intramuscular Oxymorphone and Morphine in Patients with Cancer

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

21 June 2018

Oxycodone induces overexpression of P-glycoprotein (ABCB1) and affects paclitaxel's tissue distribution in Sprague Dawley rats

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

Hepatobiliary disposition of the metabolically stable opioid peptide [D-Pen2, D-Pen5]-enkephalin (DPDPE): pharmacokinetic consequences of the interplay between multiple transport systems

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

Variable modulation of opioid brain uptake by P-glycoprotein in mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

Effects of ABCB1 (multidrug resistance transporter) gene mutations on disposition and central nervous effects of loperamide in healthy volunteers

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

Drug-drug interaction mediated by inhibition and induction of P-glycoprotein

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

Opiate-induced analgesia is increased and prolonged in mice lacking P-glycoprotein

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

P-glycoprotein-mediated transport of morphine in brain capillary endothelial cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

Effects of a potent and specific P-glycoprotein inhibitor on the blood-brain barrier distribution and antinociceptive effect of morphine in the rat.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

Enhanced antinociception of the model opioid peptide [D-penicillamine] enkephalin by P-glycoprotein modulation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

Synthetic and natural opiates interact with P-glycoprotein in multidrug-resistant cells.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401594

31 October 2018

Methods to compare dissolution profiles and a rationale for wide dissolution specifications for metoprolol tartrate tablets

1 reference

https://pubmed.ncbi.nlm.nih.gov/19481690

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effect of GF120918, a potent P-glycoprotein inhibitor, on morphine pharmacokinetics and pharmacodynamics in the rat

1 reference

https://pubmed.ncbi.nlm.nih.gov/19481690

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Comparative studies of 6-substituted delta 6-desoxymorphines and morphine with special reference to 6-methyl-delta6-desoxymorphine

1 reference

https://pubmed.ncbi.nlm.nih.gov/19481690

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Increased brain P-glycoprotein in morphine tolerant rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/19481690

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Morphine antinociception is enhanced in mdr1a gene-deficient mice

1 reference

https://pubmed.ncbi.nlm.nih.gov/19481690

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Incomplete, asymmetric, and route-dependent cross-tolerance between oxycodone and morphine in the Dark Agouti rat

1 reference

https://pubmed.ncbi.nlm.nih.gov/19481690

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Antinociceptive activity and toxicity of meperidine and normeperidine in mice

1 reference

https://pubmed.ncbi.nlm.nih.gov/19481690

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Multidrug resistance

1 reference

https://pubmed.ncbi.nlm.nih.gov/19481690

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Cyclosporin A treatment induces overexpression of P-glycoprotein in the kidney and other tissues

1 reference

https://pubmed.ncbi.nlm.nih.gov/19481690

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.IJPHARM.2009.03.037

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

26 July 2017

ResearchGate publication ID

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