(Q33604021)

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Discovery of potent small-molecule inhibitors of multidrug-resistant Plasmodium falciparum using a novel miniaturized high-throughput luciferase-based assay

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

Discovery of potent small-molecule inhibitors of multidrug-resistant Plasmodium falciparum using a novel miniaturized high-throughput luciferase-based assay (English)

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

Plasmodium falciparum

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multiple drug resistance

1 reference

based on heuristic

inferred from title

Rajesh Chandramohanadas

object named as

Rajesh Chandramohanadas

5

0 references

object named as

Hyunil Jo

3

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Giancarlo Biagini

object named as

Giancarlo A Biagini

10

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William DeGrado

11

object named as

William F DeGrado

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

1 reference

ORCID Public Data File 2021

7

object named as

Alison E Shone

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

4

object named as

Andrew D Napper

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Europe PubMed Central

PubMed publication ID

28 July 2017

author name string

Edinson Lucumi

1

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

Claire Darling

2

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Europe PubMed Central

PubMed publication ID

28 July 2017

Nicholas Fisher

6

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

Huiyan Jing

8

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

Stephen A Ward

9

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

Scott L Diamond

12

1 reference

Europe PubMed Central

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28 July 2017

Doron C Greenbaum

13

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Europe PubMed Central

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28 July 2017

language of work or name

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publication date

14 June 2010

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Europe PubMed Central

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28 July 2017

Antimicrobial Agents and Chemotherapy

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Europe PubMed Central

PubMed publication ID

28 July 2017

54

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Europe PubMed Central

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28 July 2017

9

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28 July 2017

3597-3604

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

Chemical genetics of Plasmodium falciparum

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Chapter 17 Type II NADH: quinone oxidoreductases of Plasmodium falciparum and Mycobacterium tuberculosis kinetic and high-throughput assays.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen

1 reference

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21 June 2018

Plasmodium falciparum: development of a transgenic line for screening antimalarials using firefly luciferase as the reporter

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Kinetic characterization and molecular docking of a novel, potent, and selective slow-binding inhibitor of human cathepsin L

1 reference

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21 June 2018

Acridinediones: selective and potent inhibitors of the malaria parasite mitochondrial bc1 complex

1 reference

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21 June 2018

Target assessment for antiparasitic drug discovery

1 reference

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21 June 2018

High-throughput screening assays for the identification of chemical probes

1 reference

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21 June 2018

The malaria parasite type II NADH:quinone oxidoreductase: an alternative enzyme for an alternative lifestyle

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Assessment and continued validation of the malaria SYBR green I-based fluorescence assay for use in malaria drug screening

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

High-throughput Plasmodium falciparum growth assay for malaria drug discovery

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Searching for new antimalarial therapeutics amongst known drugs

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

A clinical drug library screen identifies astemizole as an antimalarial agent

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Functional characterization and target validation of alternative complex I of Plasmodium falciparum mitochondria

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

A Comparison of Assay Performance Measures in Screening Assays: Signal Window, Z' Factor, and Assay Variability Ratio

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

The global distribution of clinical episodes of Plasmodium falciparum malaria

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Simple and inexpensive fluorescence-based technique for high-throughput antimalarial drug screening.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Human disease-related mutations in cytochrome b studied in yeast

1 reference

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21 June 2018

The past, present and future of childhood malaria mortality in Africa

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Mutations in Plasmodium falciparum cytochrome b that are associated with atovaquone resistance are located at a putative drug-binding site

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Mutations in the cytochrome b gene of Plasmodium berghei conferring resistance to atovaquone

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Resistance mutations reveal the atovaquone-binding domain of cytochrome b in malaria parasites

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Mutations in dihydropteroate synthase are responsible for sulfone and sulfonamide resistance in Plasmodium falciparum

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

N-Dialkylaminoalkylbiphenylamines as antimalarial and antischistosomal agents

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Thin sow syndrome (TSS): the effect of amperozide

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Quantitative assessment of antimalarial activity in vitro by a semiautomated microdilution technique

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

21 June 2018

Pharmacological evaluation of cimetidine, a new histamine H2-receptor antagonist, in healthy man

1 reference

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21 June 2018

Development and validation of flow cytometric measurement for parasitemia in cultures of P. falciparum vitally stained with YOYO-1.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

30 October 2018

Plasmodium falciparum var genes are regulated by two regions with separate promoters, one upstream of the coding region and a second within the intron

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2934977

30 October 2018

Studies on cytochrome oxidase. 8. Preparation and some properties of cardiac cytochrome oxidase

1 reference

https://pubmed.ncbi.nlm.nih.gov/20547797

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

2-(Aminomethyl)phenols, a new class of saluretic agents. 1. Effects of nuclear substitution

1 reference

https://pubmed.ncbi.nlm.nih.gov/20547797

12 December 2020

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Modulation of morphine antinociception by the brain-penetrating H2 antagonist zolantidine: detailed characterization in five nociceptive test systems

1 reference

https://pubmed.ncbi.nlm.nih.gov/20547797

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Site of action of the antimalarial hydroxynaphthoquinone, 2-[trans-4-(4'-chlorophenyl) cyclohexyl]-3- hydroxy-1,4-naphthoquinone (566C80)

1 reference

https://pubmed.ncbi.nlm.nih.gov/20547797

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Aminoalkylphenols as antimalarials (heterocyclicamino)-alpha-amino-o-cresols; the synthesis of camoquin

1 reference

https://pubmed.ncbi.nlm.nih.gov/20547797

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1128/AAC.00431-10

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

28 July 2017

ResearchGate publication ID

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