(Q33630509)

28 July 2017

title

Biotin analogues with antibacterial activity are potent inhibitors of biotin protein ligase (English)

1 reference

Tatiana P. Soares da Costa

28 July 2017

author

1

Tatiana P Soares da Costa

0 references

William Tieu

William Tieu

2

0 references

Steven W Polyak

Steven W Polyak

11

0 references

Andrew D Abell

10

Andrew D Abell

1 reference

28 July 2017

Min Y Yap

3

1 reference

28 July 2017

Ondrej Zvarec

4

1 reference

28 July 2017

Jan M Bell

5

1 reference

28 July 2017

John D Turnidge

6

1 reference

28 July 2017

John C Wallace

7

1 reference

28 July 2017

Grant W Booker

8

1 reference

28 July 2017

Matthew C J Wilce

9

1 reference

28 July 2017

publication date

23 May 2012

1 reference

ACS Medicinal Chemistry Letters

28 July 2017

published in

1 reference

28 July 2017

volume

3

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28 July 2017

issue

6

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28 July 2017

page(s)

509-514

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Selective inhibition of Biotin Protein Ligase from Staphylococcus aureus

28 July 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025796

Structure, function and selective inhibition of bacterial acetyl-coa carboxylase

21 June 2018

1 reference

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Bisubstrate Adenylation Inhibitors of Biotin Protein Ligase from Mycobacterium tuberculosis

21 June 2018

1 reference

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Is bacterial fatty acid synthesis a valid target for antibacterial drug discovery?

21 June 2018

1 reference

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Fix the antibiotics pipeline.

21 June 2018

1 reference

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High burden of antimicrobial resistance in Asia

21 June 2018

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Burden of endemic health-care-associated infection in developing countries: systematic review and meta-analysis

21 June 2018

1 reference

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Structure, mechanism and regulation of pyruvate carboxylase

21 June 2018

1 reference

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Purification, crystallization and preliminary crystallographic analysis of biotin protein ligase from Staphylococcus aureus.

21 June 2018

1 reference

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Microbial biotin protein ligases aid in understanding holocarboxylase synthetase deficiency

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025796

Conservation of the biotin regulon and the BirA regulatory signal in Eubacteria and Archaea.

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025796

A biotin analog inhibits acetyl-CoA carboxylase activity and adipogenesis

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025796

The C-terminal domain of biotin protein ligase from E. coli is required for catalytic activity

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025796

Biotin protein ligase from Saccharomyces cerevisiae. The N-terminal domain is required for complete activity

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025796

Evidence for distinct ligand-bound conformational states of the multifunctional Escherichia coli repressor of biotin biosynthesis.

21 June 2018

1 reference

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Mechanism of the antibiotic action of alpha-dehydrobiotin

21 June 2018

1 reference

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A novel molecular mechanism to explain biotin-unresponsive holocarboxylase synthetase deficiency

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025796

Biotin sensing at the molecular level

30 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025796

Naturally Occurring Antimetabolite Antibiotic Related to Biotin

30 October 2018

1 reference

12 December 2020

Inhibition of biotin carboxylase by a reaction intermediate analog: implications for the kinetic mechanism

1 reference

12 December 2020

Synthesis of a reaction intermediate analogue of biotin-dependent carboxylases via a selective derivatization of biotin

1 reference

12 December 2020

Synthesis of norbiotinamine and its derivatives

1 reference

12 December 2020

Identifiers

DOI

10.1021/ML300106P

1 reference

28 July 2017

1 reference

28 July 2017

1 reference