(Q33828724)

29 July 2017

title

Structure and ligand recognition of class C GPCRs (English)

1 reference

G protein-coupled receptor

29 July 2017

main subject

0 references

author name string

Lei Chun

series ordinal

1

1 reference

29 July 2017

Wen-hua Zhang

series ordinal

2

1 reference

29 July 2017

Jian-feng Liu

series ordinal

3

1 reference

29 July 2017

publication date

30 January 2012

1 reference

Acta Pharmacologica Sinica

29 July 2017

published in

1 reference

29 July 2017

volume

33

1 reference

29 July 2017

issue

3

1 reference

29 July 2017

page(s)

312-323

1 reference

Interdomain movements in metabotropic glutamate receptor activation

29 July 2017

cites work

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Ronacaleret, a calcium-sensing receptor antagonist, has no significant effect on radial fracture healing time: results of a randomized, double-blinded, placebo-controlled Phase II clinical trial

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28 July 2018

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28 July 2018

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A virtual screening hit reveals new possibilities for developing group III metabotropic glutamate receptor agonists

28 July 2018

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Molecular mechanism of the sweet taste enhancers

28 July 2018

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Ligand-induced rearrangements of the GABA(B) receptor revealed by fluorescence resonance energy transfer

28 July 2018

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28 July 2018

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Agonists and allosteric modulators of the calcium-sensing receptor and their therapeutic applications

28 July 2018

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28 July 2018

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Optical measurement of mGluR1 conformational changes reveals fast activation, slow deactivation, and sensitization.

28 July 2018

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Evolution of the class C GPCR Venus flytrap modules involved positive selected functional divergence

28 July 2018

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Metabotropic receptors for glutamate and GABA in pain.

28 July 2018

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Allosteric modulators of GPCRs: a novel approach for the treatment of CNS disorders

28 July 2018

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Molecular mechanism for the umami taste synergism

28 July 2018

1 reference

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Activation of metabotropic glutamate receptors as a novel approach for the treatment of schizophrenia

28 July 2018

1 reference

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Characterization of (R,S)-5,7-di-tert-butyl-3-hydroxy-3-trifluoromethyl-3H-benzofuran-2-one as a positive allosteric modulator of GABAB receptors

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Transposition of three amino acids transforms the human metabotropic glutamate receptor (mGluR)-3-positive allosteric modulation site to mGluR2, and additional characterization of the mGluR2-positive allosteric modulation site

28 July 2018

1 reference

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Functioning of the dimeric GABA(B) receptor extracellular domain revealed by glycan wedge scanning.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Structural diversity of G protein-coupled receptors and significance for drug discovery

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

N-{4-Chloro-2-[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)methyl]phenyl}-2-hydroxybenzamide (CPPHA) acts through a novel site as a positive allosteric modulator of group 1 metabotropic glutamate receptors

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Activation of a dimeric metabotropic glutamate receptor by intersubunit rearrangement.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Activation of mGlu2/3 receptors as a new approach to treat schizophrenia: a randomized Phase 2 clinical trial

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Molecular diversity, trafficking and subcellular localization of GABAB receptors

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Dual signaling is differentially activated by different active states of the metabotropic glutamate receptor 1alpha

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

GABAB receptor: a site of therapeutic benefit

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Lactisole interacts with the transmembrane domains of human T1R3 to inhibit sweet taste.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Metabotropic glutamate receptors as novel targets for anxiety and stress disorders

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Don't worry 'B' happy!: a role for GABA(B) receptors in anxiety and depression.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

A region in the seven-transmembrane domain of the human Ca2+ receptor critical for response to Ca2+.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

The cysteine-rich region of T1R3 determines responses to intensely sweet proteins

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Closed state of both binding domains of homodimeric mGlu receptors is required for full activity.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

The heptahelical domain of GABA(B2) is activated directly by CGP7930, a positive allosteric modulator of the GABA(B) receptor

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Positive and negative allosteric modulators of the Ca2+-sensing receptor interact within overlapping but not identical binding sites in the transmembrane domain

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Molecular determinants involved in the allosteric control of agonist affinity in the GABAB receptor by the GABAB2 subunit.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Heptahelical domain of metabotropic glutamate receptor 5 behaves like rhodopsin-like receptors.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Allosteric modulation of group III metabotropic glutamate receptor 4: A potential approach to Parkinson's disease treatment

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Modeling and Mutagenesis of the Binding Site of Calhex 231, a Novel Negative Allosteric Modulator of the Extracellular Ca2+-sensing Receptor

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Mutational Analysis and Molecular Modeling of the Binding Pocket of the Metabotropic Glutamate 5 Receptor Negative Modulator 2-Methyl-6-(phenylethynyl)-pyridine

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Evolution, structure, and activation mechanism of family 3/C G-protein-coupled receptors

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

The metabotropic glutamate receptors: structure, activation mechanism and pharmacology

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Anxiolytic effects of a novel group II metabotropic glutamate receptor agonist (LY354740) in the fear-potentiated startle paradigm in humans

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Identification of acidic residues in the extracellular loops of the seven-transmembrane domain of the human Ca2+ receptor critical for response to Ca2+ and a positive allosteric modulator

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Closure of the Venus flytrap module of mGlu8 receptor and the activation process: Insights from mutations converting antagonists into agonists

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Three adjacent serines in the extracellular domains of the CaR are required for L-amino acid-mediated potentiation of receptor function

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Function of GB1 and GB2 subunits in G protein coupling of GABA(B) receptors

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Positive allosteric modulation of native and recombinant gamma-aminobutyric acid(B) receptors by 2,6-Di-tert-butyl-4-(3-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) and its aldehyde analog CGP13501

28 July 2018

2 references

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

28 July 2018

https://api.crossref.org/works/10.1038%2FAPS.2011.186

7 January 2021

inferred from DOI database lookup

Positive allosteric modulators of metabotropic glutamate 1 receptor: characterization, mechanism of action, and binding site

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Mammalian sweet taste receptors

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

A candidate taste receptor gene near a sweet taste locus

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Covalent and noncovalent interactions mediate metabotropic glutamate receptor mGlu5 dimerization.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Cys-140 is critical for metabotropic glutamate receptor-1 dimerization

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Cryptic dimer interface and domain organization of the extracellular region of metabotropic glutamate receptor subtype 1.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Human Ca2+ receptor cysteine-rich domain. Analysis of function of mutant and chimeric receptors

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Calcium sensing properties of the GABA(B) receptor.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Identification of the cysteine residues in the amino-terminal extracellular domain of the human Ca(2+) receptor critical for dimerization. Implications for function of monomeric Ca(2+) receptor

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

The agonist-binding domain of the calcium-sensing receptor is located at the amino-terminal domain

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Mutagenesis and modeling of the GABAB receptor extracellular domain support a venus flytrap mechanism for ligand binding

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

CPCCOEt, a noncompetitive metabotropic glutamate receptor 1 antagonist, inhibits receptor signaling without affecting glutamate binding

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

GABA(B)-receptor subtypes assemble into functional heteromeric complexes.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Domains involved in the specificity of G protein activation in phospholipase C-coupled metabotropic glutamate receptors.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

G-protein-coupled receptor oligomerization and its potential for drug discovery

28 July 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Allosteric modulation of family C G-protein-coupled receptors: from molecular insights to therapeutic perspectives

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Pharmacology and functions of metabotropic glutamate receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

GABA(B) receptors function as a heteromeric assembly of the subunits GABA(B)R1 and GABA(B)R2.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Phospho-dependent functional modulation of GABA(B) receptors by the metabolic sensor AMP-dependent protein kinase.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Ischemic preconditioning ameliorates excitotoxicity by shifting glutamate/gamma-aminobutyric acid release and biosynthesis

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

GABAB receptor activation protects neurons from apoptosis via IGF-1 receptor transactivation.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Clinical lessons from the calcium-sensing receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Future therapeutic targets in osteoporosis

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Anti-parathyroid and anti-calcium sensing receptor antibodies in autoimmune hypoparathyroidism

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Structural views of the ligand-binding cores of a metabotropic glutamate receptor complexed with an antagonist and both glutamate and Gd3+.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Locking the dimeric GABA(B) G-protein-coupled receptor in its active state.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Structures of the extracellular regions of the group II/III metabotropic glutamate receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Ligand-induced rearrangement of the dimeric metabotropic glutamate receptor 1alpha.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Dimerization of the extracellular calcium-sensing receptor (CaR) on the cell surface of CaR-transfected HEK293 cells.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Structure, pharmacology and therapeutic prospects of family C G-protein coupled receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Mutational analysis and molecular modeling of the allosteric binding site of a novel, selective, noncompetitive antagonist of the metabotropic glutamate 1 receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Identification of the cyclamate interaction site within the transmembrane domain of the human sweet taste receptor subunit T1R3.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Determination of key amino acids implicated in the actions of allosteric modulation by 3,3'-difluorobenzaldazine on rat mGlu5 receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

A novel class of positive allosteric modulators of metabotropic glutamate receptor subtype 1 interact with a site distinct from that of negative allosteric modulators

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

The antibody-capture [(35)S]GTPgammaS scintillation proximity assay: a powerful emerging technique for analysis of GPCR pharmacology

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Dominant role of GABAB2 and Gbetagamma for GABAB receptor-mediated-ERK1/2/CREB pathway in cerebellar neurons.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

N,N'-Dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine (GS39783) and structurally related compounds: novel allosteric enhancers of gamma-aminobutyric acidB receptor function.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Arylalkylamines are a novel class of positive allosteric modulators at GABA(B) receptors in rat neocortex

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Potentiation of metabotropic GABAB receptors by l-amino acids and dipeptides in rat neocortex

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Delineating a Ca2+ binding pocket within the venus flytrap module of the human calcium-sensing receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

A novel calcium-sensing receptor antagonist transiently stimulates parathyroid hormone secretion in vivo

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2011.186

Ca(2+) requirement for high-affinity gamma-aminobutyric acid (GABA) binding at GABA(B) receptors: involvement of serine 269 of the GABA(B)R1 subunit

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4077135

Coupling of agonist binding to effector domain activation in metabotropic glutamate-like receptors

29 October 2018

1 reference

12 December 2020

Amino-pyrrolidine tricarboxylic acids give new insight into group III metabotropic glutamate receptor activation mechanism

1 reference

12 December 2020

Virtual screening workflow development guided by the "receiver operating characteristic" curve approach. Application to high-throughput docking on metabotropic glutamate receptor subtype 4

1 reference

12 December 2020

The non-competitive antagonists 2-methyl-6-(phenylethynyl)pyridine and 7-hydroxyiminocyclopropan[b]chromen-1a-carboxylic acid ethyl ester interact with overlapping binding pockets in the transmembrane region of group I metabotropic glutamate recepto

1 reference

12 December 2020

The second cytoplasmic loop of metabotropic glutamate receptor functions at the third loop position of rhodopsin

1 reference

12 December 2020

Identifiers

DOI

10.1038/APS.2011.186

1 reference

Dimensions Publication ID

29 July 2017

0 references

1 reference

29 July 2017

1 reference