(Q34419702)

2 August 2017

1 reference

title

The estradiol pharmacophore: ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site (English)

1 reference

2 August 2017

Anstead GM

1

1 reference

PubMed ID

9071738

2 August 2017

Carlson KE

series ordinal

2

1 reference

PubMed ID

9071738

2 August 2017

Katzenellenbogen JA

series ordinal

3

1 reference

2 August 2017

1 March 1997

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2 August 2017

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2 August 2017

62

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2 August 2017

3

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2 August 2017

268-303

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https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

2 August 2017

1 reference

7 January 2021

Hormonal treatment of postmenopausal women

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Radiolabeled steroidal estrogens in cancer research

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The steroid and thyroid hormone receptor superfamily

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Full-length sequence and in vitro expression of rainbow trout estrogen receptor cDNA.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Molecular cloning and characterization of rat estrogen receptor cDNA.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Structural organization and expression of the mouse estrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Human oestrogen receptor cDNA: sequence, expression and homology to v-erb-A

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Sequence and expression of human estrogen receptor complementary DNA

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The C-terminal half of the porcine estradiol receptor contains no post-translational modification: determination of the primary structure

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

DNA recognition by the oestrogen receptor: from solution to the crystal.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Crystal structure of the ligand-binding domain of the human nuclear receptor RXR-alpha

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Crystal structure of the RAR-gamma ligand-binding domain bound to all-trans retinoic acid

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

A structural role for hormone in the thyroid hormone receptor.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

A canonical structure for the ligand-binding domain of nuclear receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Tripartite steroid hormone receptor pharmacology: interaction with multiple effector sites as a basis for the cell- and promoter-specific action of these hormones

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Nuclear hormone receptors: ligand-activated regulators of transcription and diverse cell responses

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Benz[a]anthracene diols: predicted carcinogenicity and structure-estrogen receptor binding affinity relationships

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Do thermodynamic studies provide information on both the binding to and the activation of dopaminergic and other receptors?

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

11.beta.-Methoxy-, 11.beta.-ethyl, and 17.alpha.-ethynyl-substituted 16.alpha.-fluoroestradiols: receptor-based imaging agents with enhanced uptake efficiency and selectivity

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Torsionally and hydrophobically modified 2,3-diarylindenes as estrogen receptor ligands

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The crystal and molecular structure of diethylstilbestrol

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Molecular conformation, receptor binding, and hormone action of natural and synthetic estrogens and antiestrogens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Development and use of quantum mechanical molecular models. 76. AM1: a new general purpose quantum mechanical molecular model

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Molecular modeling of steroidal estrogens: novel conformations and their role in biological activity

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Functional group contributions to drug-receptor interactions.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Kinetics of the hormone-receptor interaction competition experiments with slowly equilibrating ligands

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The relevance of kinetic parameters in the determination of specific binding to the estrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

11 beta-chloromethyl-[3H]estradiol-17 beta: a very high affinity, reversible ligand for the estrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Equilibrium hormone binding to human estrogen receptors in highly diluted cell extracts is non-cooperative and has a Kd of approximately 10 pM.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Interaction of 17β-estradiol and its specific uterine receptor. Evidence for complex kinetic and equilibrium behavior

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Methyl and bromo derivatives of estradiol are agonistic ligands for the estrogen receptor of MCF-7 breast cancer cells

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Binding characteristics of estrone, estradiol and estriol to the human myometrial estrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The synthesis and study of some potential affinity labeling reagents for estrogen receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The relationship between estrogenic action and chemical constitution in a group of azomethine derivatives

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Correspondence factor analysis of steroid libraries

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Steroid flexibility and receptor specificity

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Hydrogen bonding in globular proteins

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Estrogenic steroids. 3. The crystal and molecular structure of estriol

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

A series of optical structural and isomeric analogs of estradiol: a comparative study of the biological activity and affinity to cytosol receptor of rabbit uterus

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Ligand-mediated modulation of estrogen receptor conformation by estradiol analogs

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

2-Arylindenes and 2-arylindenones: molecular structures and considerations in the binding orientation of unsymmetrical nonsteroidal ligands to the estrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Hydrogen bonding and biological specificity analysed by protein engineering

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Quantitation of long-range effects in steroids by molecular orbital calculations

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Crystal structure of human estrogenic 17 beta-hydroxysteroid dehydrogenase complexed with 17 beta-estradiol

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The structure of a complex of human 17beta-hydroxysteroid dehydrogenase with estradiol and NADP+ identifies two principal targets for the design of inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Structure-activity relationships of estrogens. Effects of 14-dehydrogenation and axial methyl groups at C-7, C-9 and C-11

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Comparative binding affinity of estrogens and its relation to estrogenic potency

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Photoaffinity labels for estrogen binding proteins of rat uterus.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Hydrogen bonding and specificity. Fluorodeoxy sugars as probes of hydrogen bonding in the glycogen phosphorylase-glucose complex

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Hydrogen bond stereochemistry in protein structure and function

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Distributions of water around amino acid residues in proteins

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Molecular details of receptor binding and hormonal action of steroids derived from X-ray crystallographic investigations

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The crystal and molecular structures of an unusual estra-steroid and of its dihydroproduct

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Segmental motion in catalysis: investigation of a hydrogen bond critical for loop closure in the reaction of triosephosphate isomerase

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Some hypotheses about interactions between estrogen and androgen and their possible receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Internal water molecules and H‐bonding in biological macromolecules: A review of structural features with functional implications

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Ligand atom partial charges assignment for complementary electrostatic potentials

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Internal cavities and buried waters in globular proteins.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Use of NMR to detect water within nonpolar protein cavities

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Further development of hydrogen bond functions for use in determining energetically favorable binding sites on molecules of known structure. 1. Ligand probe groups with the ability to form two hydrogen bonds

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Solvent effect on binding thermodynamics of biopolymers

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Receptor Binding as a Tool in the Development of New Bioactive Steroids

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

A ligand-induced conformational change in the estrogen receptor is localized in the steroid binding domain

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Interactions of hormonal steroids: progestogens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The androgen receptor binding site: a conformational study of steroids in relation with their affinity--I. Interaction with the D-ring

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Shielding effects at 17 alpha-substituted estrogens. A tentative explanation for the low biological activity of 17 alpha-ethyl-estradiol based on i.r. and NMR spectroscopic studies.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

New hydrogen-bond potentials for use in determining energetically favorable binding sites on molecules of known structure

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Docking flexible ligands to macromolecular receptors by molecular shape

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Synthesis of new amino acid and peptide derivatives of estradiol and their binding affinities for the estrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Steroid binding to the cytosolic estrogen receptor from rat uterus. Influence of the orientation of substituents in the 17-position of the 8 beta- and 8 alpha-series

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Synthesis, receptor binding, and target-tissue uptake of carbon-11 labeled carbamate derivatives of estradiol and hexestrol

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

17-Desoxy estrogen analogues

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

2-hydroxyestradiol-17 alpha and 4-hydroxyestradiol-17 alpha, catechol estrogen analogs with reduced estrogen receptor affinity

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Influence of estrogen structure on nuclear binding and progesterone receptor induction by the receptor complex

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Steroid and phyto-oestrogen binding to sheep uterine receptors in vitro

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The specificity of the estrogen receptor of human uterus

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Structure-activity relationships of 9 beta-estrogens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Post-coital contraceptive activity and estrogen receptor binding affinity of phenolic steroids

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Uterine estrogen receptor binding of catecholestrogens and of estetrol (1,3,5(10)-estratriene-3,15α,16α,17β-tetrol)

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Coumestrol, NBD-norhexestrol, and dansyl-norhexestrol, fluorescent probes of estrogen-binding protiens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Photoreactivity of some light-sensitive estrogen derivatives. Use of an exchange assay to determine their photointeraction with the rat uterine estrogen binding protein

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

17 alpha-allyl estradiol analogues as candidates for development of high-affinity fluorescein-estradiol conjugates

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

17 alpha-substituted analogs of estradiol for the development of fluorescent estrogen receptor ligands

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Steroidal affinity labels of the estrogen receptor. 1. 17 alpha-(Bromoacetoxy)alkyl/alkynylestradiols

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Structure-activity relationships of estrogenic ligands: synthesis and evaluation of (17 alpha, 20E)- and (17 alpha, 20Z)-21-halo-19-norpregna-1,3,5(10),20-tetraene-3,17 beta-diols.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Synthesis and estrogen receptor binding of (17 alpha, 20E)- and (17 alpha, 20Z)-21-phenylthio- and 21-phenylseleno-19-norpregna-1,3,5(10),20-tetraene-3,17 beta-diols

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Synthesis, receptor binding, and tissue distribution of (17 alpha,20E)- and (17 alpha,20Z)-21-[125I]iodo-19-norpregna-1,3,5(10), 20-tetraene-3,17-diol

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

11 beta-Substituted estradiol derivatives, potential high-affinity carbon-11-labeled probes for the estrogen receptor: a structure-affinity relationship study

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Synthesis, receptor binding and biodistribution of the gem-21-chloro-21-iodovinylestradiol derivatives

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Bioorganometallic chemistry: a future direction for transition metal organometallic chemistry?

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Organometallic derivatives of estradiol as bioligands: targetted binding of the estradiol receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Syntheses and affinities of novel organometallic-labeled estradiol derivatives: a structure-affinity relationship

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Selenium labeling in nuclear medicine. 2. D ring substituted estrogens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The biologic activity of selenoestrogens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Ellipticine derivatives with an affinity to the estrogen receptor, an approach to develop intercalating drugs with a specific effect on the hormone-dependent breast cancer

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

3,17 beta-Dihydroxy-20,21-epoxy-19-norpregna-1,3,5(10)-trienes: synthesis, rearrangement, cytotoxicity, and estrogen-receptor binding

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Steroidal affinity labels of the estrogen receptor. 2. 17 alpha-[(Haloacetamido)alkyl]estradiols.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The steroid specificity of the estrogen-receptor of human breast carcinoma

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Estrogen receptor based imaging agents. 1. Synthesis and receptor binding affinity of some aromatic and D-ring halogenated estrogens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Estrogen and androgen receptor binding affinity of 10 beta-chloro-estrenen derivatives

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Synthesis, antitubulin and antimitotic activity, and cytotoxicity of analogs of 2-methoxyestradiol, an endogenous mammalian metabolite of estradiol that inhibits tubulin polymerization by binding to the colchicine binding site

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Synthesis and biological activity of 4-methylestradiol

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Classical electrostatics in biology and chemistry

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Thyroid hormone analogues. Synthesis of 3'-substituted 3,5-diiodo-L-thyronines and quantitative structure-activity studies of in vitro and in vivo thyromimetic activities in rat liver and heart.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Binding, X-ray and NMR studies of the three A-ring isomers of natural estradiol

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Estrogen receptor binding characteristics of 1,11 beta-ethanoestradiol: effect of a 1,11 beta-bridge on steroidal estrogen

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

2- and 4-fluorinated 16 alpha(-)[125I]iodoestradiol derivatives: synthesis and effect on estrogen receptor binding and receptor-mediated target tissue uptake

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Organometallic estrogens: synthesis, interaction with lamb uterine estrogen receptor, and detection by infrared spectroscopy

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Estrogen platinum-diamine complexes: Preparation of a non-steroidal estrogen platinum—diamine complex labeled with platinum-191 and a study of its binding to the estrogen receptor in vitro and its tissue distribution in vivo

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Binding of 2-hydroxyestradiol and 4-hydroxyestradiol to estrogen receptors from human breast cancers

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Impact of Continuously Administered Catechol Estrogens on Uterine Growth and Luteinizing Hormone Secretion*

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Steroid structure and function. Molecular conformation of 4-hydroxyestradiol and its relation to other catechol estrogens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Substituted derivatives of A-nor-5 alpha-androstane and A-nor-5 alpha-estrane--structure and affinity for hormonal receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Cation-pi interactions in chemistry and biology: a new view of benzene, Phe, Tyr, and Trp

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The nature of thyroxine and related compounds as electron donors.

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Regio and stereospecific synthesis of 11 beta-substituted 19-norsteroids. Influence of 11 beta-substitution on progesterone receptor affinity - (1)

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

11 beta-substituted estradiol derivatives. 2. Potential carbon-11- and iodine-labeled probes for the estrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Skeletal conformations and receptor binding of some 9,11-modified estradiols

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Synthesis and biologic activities of 11 beta-substituted estradiol as potential antiestrogens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

11 beta-Amidoalkoxyphenyl estradiols, a new series of pure antiestrogens

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

Estrogen receptor binding tolerance of 16 alpha-substituted estradiol derivatives

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The molecular structure of 16 alpha-iodo-17 beta-estradiol, a high affinity ligand for the estrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

The synthesis of 7 alpha-methyl-substituted estrogens labeled with fluorine-18: potential breast tumor imaging agents

1 reference

https://api.crossref.org/works/10.1016%2FS0039-128X%2896%2900242-5

7 January 2021

A synthesis of 7 alpha-substituted estradiols: synthesis and biological evaluation of a 7 alpha-pentyl-substituted BODIPY fluorescent conjugate and a fluorine-18-labeled 7 alpha-pentylestradiol analog

1 reference

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7 January 2021

Synthesis and structure-affinity of a series of 7 alpha-undecylestradiol derivatives: a potential vector for therapy and imaging of estrogen-receptor-positive cancers

1 reference

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7 January 2021

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1 reference

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7 January 2021

ICI 182,780, a new antioestrogen with clinical potential

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7 January 2021

Studies with steroid-fluorescein conjugates on oestrogen target tissues

1 reference

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7 January 2021

Steroid structure and function--IX. Molecular conformation and receptor binding of isomeric analogs of D-homo-estradiol

1 reference

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7 January 2021

Quantitative structure-activity relationships of estrogenic steroids substituted at C14, C15

1 reference

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7 January 2021

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1 reference

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7 January 2021

Principles of protein-protein recognition

1 reference

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7 January 2021

Displacement of Estradiol from Estrogen Receptors by Simple Alkyl Phenols*

1 reference

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7 January 2021

Computer-aided drug design

1 reference

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7 January 2021

Seco-oestradiols and some non-steroidal oestrogens: Structural correlates of oestrogenic action

1 reference

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7 January 2021

Synthesis and biological activity of some 15-oxaestranes

1 reference

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7 January 2021

Identification of thiol group at the estrogen-binding site on the cytoplasmic receptor from rabbit uterus by affinity labeling

1 reference

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7 January 2021

Sulfhydryl Groups and Estradiol-Receptor Interaction

1 reference

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7 January 2021

Cysteinyl-tRNA synthetase from Escherichia coli does not need an editing mechanism to reject serine and alanine. High binding energy of small groups in specific molecular interactions

1 reference

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7 January 2021

Identification of amino acids in the hormone binding domain of the human estrogen receptor important in estrogen binding

1 reference

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7 January 2021

Carboxymethylation of the human estrogen receptor ligand-binding domain-estradiol complex: HPLC/ESMS peptide mapping shows that cysteine 447 does not react with iodoacetic acid

1 reference

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7 January 2021

Binding Activity of Oestrogen Receptors destroyed by Iodination

1 reference

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7 January 2021

Differential inhibition of estrogen and antiestrogen binding to the estrogen receptor by diethylpyrocarbonate

1 reference

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7 January 2021

Differential interactions of estrogens and antiestrogens at the 17 beta-hydroxy or counterpart function with the estrogen receptor

1 reference

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7 January 2021

Evidence for involvement of tyrosine in estradiol binding by rat uterus estrogen receptor

1 reference

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7 January 2021

Contribution of hydrogen bonding to the conformational stability of ribonuclease T1

1 reference

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7 January 2021

Properties of a purified estradiol-dependent calf uterus tyrosine kinase

1 reference

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7 January 2021

Quantitative structure-activity relationships/comparative molecular field analysis (QSAR/CoMFA) for receptor-binding properties of halogenated estradiol derivatives

1 reference

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7 January 2021

Molecular structures, conformational analysis, and preferential modes of binding of 3-aroyl-2-arylbenzo[b]thiophene estrogen receptor ligands: LY117018 and aryl azide photoaffinity labeling analogs

1 reference

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7 January 2021

A MATHEMATICAL CONTRIBUTION TO STRUCTURE-ACTIVITY STUDIES.

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7 January 2021

Flexible Drug Molecules and Dynamic Receptors

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7 January 2021

Thermodynamic properties of ligand binding by monoclonal anti-fluorescyl antibodies.

1 reference

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7 January 2021

Molecular modelling of the human estrogen receptor and ligand interactions based on site-directed mutagenesis and amino acid sequence homology

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7 January 2021

A model for the determination of the 3D-spatial distribution of the functions of the hormone-binding domain of receptors that bind 3-keto-4-ene steroids

1 reference

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7 January 2021

Analysis of the binding of 3,3',5-triiodo-L-thyronine and its analogues to mutant human beta 1 thyroid hormone receptors: a model of the hormone binding site

1 reference

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7 January 2021

10.1016/S0039-128X(96)00242-5

Identifiers

DOI

1 reference

2 August 2017

1 reference

PubMed ID

9071738