(Q35105899)

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Histone methyltransferase inhibitors are orally bioavailable, fast-acting molecules with activity against different species causing malaria in humans

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Europe PubMed Central

PubMed publication ID

6 August 2017

Histone methyltransferase inhibitors are orally bioavailable, fast-acting molecules with activity against different species causing malaria in humans (English)

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Europe PubMed Central

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6 August 2017

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6 August 2017

François Nosten

9

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6 August 2017

Nicholas A Malmquist

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Nicholas A Malmquist

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Andrea Ruecker

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Michael J Delves

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Matthew Fuchter

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Matthew J Fuchter

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Sandra Duffy

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Vicky M Avery

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Sergio Wittlin

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6 August 2017

Sandeep Sundriyal

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Sandeep Sundriyal

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Santiago Ferrer

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Santiago Ferrer

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Maria Belen Jimenez-Diaz

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María Belén Jiménez-Díaz

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6 August 2017

Francisco Javier Gamo

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Francisco-Javier Gamo

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6 August 2017

Iñigo Angulo-Barturen

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Iñigo Angulo-Barturen

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6 August 2017

Robert E Sinden

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Robert E Sinden

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6 August 2017

8

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Laurent Renia

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6 August 2017

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Joachim Caron

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6 August 2017

Patty Chen

4

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6 August 2017

Benoit Witkowski

5

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6 August 2017

Rossarin Suwanarusk

7

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6 August 2017

María Santos Martínez

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6 August 2017

Laura M Sanz

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6 August 2017

Artur Scherf

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6 August 2017

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publication date

24 November 2014

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6 August 2017

Antimicrobial Agents and Chemotherapy

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6 August 2017

59

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6 August 2017

2

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6 August 2017

950-959

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6 August 2017

Development of diaminoquinazoline histone lysine methyltransferase inhibitors as potent blood-stage antimalarial compounds

1 reference

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Persistence and activation of malaria hypnozoites in long-term primary hepatocyte cultures

1 reference

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2,4-Diaminothienopyrimidines as orally active antimalarial agents

1 reference

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A molecular marker of artemisinin-resistant Plasmodium falciparum malaria

1 reference

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Single dose primaquine for clearance of Plasmodium falciparum gametocytes in children with uncomplicated malaria in Uganda: a randomised, controlled, double-blind, dose-ranging trial

1 reference

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Identification of inhibitors of Plasmodium falciparum gametocyte development

1 reference

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Novel phenotypic assays for the detection of artemisinin-resistant Plasmodium falciparum malaria in Cambodia: in-vitro and ex-vivo drug-response studies

1 reference

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PfSETvs methylation of histone H3K36 represses virulence genes in Plasmodium falciparum

1 reference

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Male and female Plasmodium falciparum mature gametocytes show different responses to antimalarial drugs

1 reference

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Reduced susceptibility of Plasmodium falciparum to artesunate in southern Myanmar

1 reference

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Silence, activate, poise and switch! Mechanisms of antigenic variation in Plasmodium falciparum.

1 reference

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Efficacy of dihydroartemisinin-piperaquine for treatment of uncomplicated Plasmodium falciparum and Plasmodium vivax in Cambodia, 2008 to 2010.

1 reference

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Reduced artemisinin susceptibility of Plasmodium falciparum ring stages in western Cambodia

1 reference

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9 July 2018

In vivo susceptibility of Plasmodium falciparum to artesunate in Binh Phuoc Province, Vietnam

1 reference

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9 July 2018

Small-molecule histone methyltransferase inhibitors display rapid antimalarial activity against all blood stage forms in Plasmodium falciparum

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4335868

9 July 2018

Cancer epigenetics: from mechanism to therapy

1 reference

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9 July 2018

Emergence of artemisinin-resistant malaria on the western border of Thailand: a longitudinal study

1 reference

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9 July 2018

P. falciparum in vitro killing rates allow to discriminate between different antimalarial mode-of-action

1 reference

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9 July 2018

PfSET10, a Plasmodium falciparum methyltransferase, maintains the active var gene in a poised state during parasite division

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4335868

9 July 2018

The threat of artemisinin-resistant malaria

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4335868

9 July 2018

Synthetic ozonide drug candidate OZ439 offers new hope for a single-dose cure of uncomplicated malaria

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4335868

9 July 2018

Protein lysine methyltransferase G9a inhibitors: design, synthesis, and structure activity relationships of 2,4-diamino-7-aminoalkoxy-quinazolines

1 reference

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9 July 2018

Targeting the hypnozoite reservoir of Plasmodium vivax: the hidden obstacle to malaria elimination

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4335868

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Improved murine model of malaria using Plasmodium falciparum competent strains and non-myelodepleted NOD-scid IL2Rgammanull mice engrafted with human erythrocytes

1 reference

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Dynamic histone H3 epigenome marking during the intraerythrocytic cycle of Plasmodium falciparum

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4335868

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Effective and cheap removal of leukocytes and platelets from Plasmodium vivax infected blood

1 reference

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Identification of a metabolically stable triazolopyrimidine-based dihydroorotate dehydrogenase inhibitor with antimalarial activity in mice

1 reference

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Genome-wide analysis of heterochromatin associates clonally variant gene regulation with perinuclear repressive centers in malaria parasites

1 reference

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Determinants of in vitro drug susceptibility testing of Plasmodium vivax

1 reference

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5' flanking region of var genes nucleate histone modification patterns linked to phenotypic inheritance of virulence traits in malaria parasites

1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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Simple and inexpensive fluorescence-based technique for high-throughput antimalarial drug screening.

1 reference

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1 reference

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Online analysis of in vitro resistance to antimalarial drugs through nonlinear regression

1 reference

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27 September 2018

Quantitative measurement of Plasmodium-infected erythrocytes in murine models of malaria by flow cytometry using bidimensional assessment of SYTO-16 fluorescence

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4335868

27 September 2018

Identifiers

10.1128/AAC.04419-14

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Europe PubMed Central

PubMed publication ID

6 August 2017

release_mnqocjcfdzd5rhnimjuuqzlf24

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https://api.fatcat.wiki/v0/release/mnqocjcfdzd5rhnimjuuqzlf24

24 November 2022

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PMC publication ID

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Europe PubMed Central

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6 August 2017

PubMed publication ID

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Europe PubMed Central

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6 August 2017

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