(Q35287517)

7 August 2017

title

Hydrophobic anions potently and uncompetitively antagonize GABA(A) receptor function in the absence of a conventional binding site (English)

1 reference

7 August 2017

1 reference

3

C F Zorumski

1 reference

7 August 2017

M Chisari

1

1 reference

7 August 2017

K Wu

series ordinal

2

1 reference

7 August 2017

S Mennerick

series ordinal

4

1 reference

7 August 2017

language of work or name

English

0 references

publication date

1 September 2011

1 reference

British Journal of Pharmacology

7 August 2017

published in

1 reference

7 August 2017

volume

164

1 reference

7 August 2017

issue

2b

1 reference

7 August 2017

page(s)

667-680

1 reference

GABA A,slow: causes and consequences.

7 August 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Structurally diverse amphiphiles exhibit biphasic modulation of GABAA receptors: similarities and differences with neurosteroid actions.

12 July 2018

1 reference

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The sticky issue of neurosteroids and GABA(A) receptors

12 July 2018

1 reference

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Submillisecond optical reporting of membrane potential in situ using a neuronal tracer dye.

12 July 2018

1 reference

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The influence of neuroactive steroid lipophilicity on GABAA receptor modulation: evidence for a low-affinity interaction

12 July 2018

1 reference

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Lipid bilayer-mediated regulation of ion channel function by amphiphilic drugs

12 July 2018

1 reference

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Effects on membrane capacitance of steroids with antagonist properties at GABAA receptors

12 July 2018

1 reference

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Cyclodextrins sequester neuroactive steroids and differentiate mechanisms that rate limit steroid actions

12 July 2018

1 reference

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Seizures and enhanced cortical GABAergic inhibition in two mouse models of human autosomal dominant nocturnal frontal lobe epilepsy.

12 July 2018

1 reference

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GABA(A) receptor function is regulated by lipid bilayer elasticity

12 July 2018

1 reference

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Structural model for gamma-aminobutyric acid receptor noncompetitive antagonist binding: widely diverse structures fit the same site

12 July 2018

1 reference

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Development of gamma-aminobutyric acidergic synapses in cultured hippocampal neurons

12 July 2018

1 reference

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Mechanism of action of memantine

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Neurosteroid access to the GABAA receptor

12 July 2018

1 reference

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A hybrid approach to measuring electrical activity in genetically specified neurons

12 July 2018

1 reference

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Diversity of inhibitory neurotransmission through GABA(A) receptors

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

A membrane-access mechanism of ion channel inhibition by voltage sensor toxins from spider venom

12 July 2018

1 reference

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3beta -hydroxypregnane steroids are pregnenolone sulfate-like GABA(A) receptor antagonists.

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Pregnenolone sulfate block of GABA(A) receptors: mechanism and involvement of a residue in the M2 region of the alpha subunit

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Neurosteroid analogues. 6. The synthesis and GABAA receptor pharmacology of enantiomers of dehydroepiandrosterone sulfate, pregnenolone sulfate, and (3alpha,5beta)-3-hydroxypregnan-20-one sulfate

12 July 2018

1 reference

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GABAA-receptor heterogeneity in the adult rat brain: differential regional and cellular distribution of seven major subunits

12 July 2018

1 reference

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Multiple mechanisms of picrotoxin block of GABA-induced currents in rat hippocampal neurons

12 July 2018

1 reference

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Induced capacitance in the squid giant axon. Lipophilic ion displacement currents

12 July 2018

1 reference

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Excitatory and inhibitory autaptic currents in isolated hippocampal neurons maintained in cell culture

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

The interaction of hydrophobic ions with lipid bilayer membranes

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Potential energy barriers to ion transport within lipid bilayers. Studies with tetraphenylborate

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Transport kinetics of hydrophobic ions in lipid bilayer membranes. Charge-pulse relaxation studies.

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Local anesthetics: hydrophilic and hydrophobic pathways for the drug-receptor reaction

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Guide to Receptors and Channels (GRAC), 4th Edition

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

The neurosteroids dehydroepiandrosterone sulfate and pregnenolone sulfate inhibit the UNC-49 GABA receptor through a common set of residues

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Enantiomers of neuroactive steroids support a specific interaction with the GABA-C receptor as the mechanism of steroid action

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Membrane voltage modulates the GABA(A) receptor gating in cultured rat hippocampal neurons.

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Gating charge displacement in voltage-gated ion channels involves limited transmembrane movement

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Slow actions of neuroactive steroids at GABAA receptors.

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Activation-dependent properties of pregnenolone sulfate inhibition of GABAA receptor-mediated current

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

How quickly can GABAA receptors open?

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Molecular pharmacology of gamma-aminobutyric acid type A receptor agonists and partial agonists in oocytes injected with different alpha, beta, and gamma receptor subunit combinations.

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Modification of dose-response curves by effector blockade and uncompetitive antagonism

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Membrane potential modulates the activation of GABA-gated channels

26 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188920

Transport kinetics of dipicrylamine through lipid bilayer membranes. Effects of membrane structure

26 September 2018

1 reference

Crossref

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2011.01396.X

Nonuniform probability of glutamate release at a hippocampal synapse

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2011.01396.X

Transport mechanism of hydrophobic ions through lipid bilayer membranes

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21457224

12 December 2020

inferred from PubMed ID database lookup

Pregnenolone sulfate modulates inhibitory synaptic transmission by enhancing GABA(A) receptor desensitization

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21457224

12 December 2020

inferred from PubMed ID database lookup

Passive and synaptic properties of hippocampal neurons grown in microcultures and in mass cultures

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21457224

12 December 2020

inferred from PubMed ID database lookup

Identifiers

DOI

10.1111/J.1476-5381.2011.01396.X

1 reference

release_wqatrj5vovfwjlp5f3twj72psy

7 August 2017

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/wqatrj5vovfwjlp5f3twj72psy

24 November 2022

mapped directly with Wikidata item

PMC publication ID

3188920

1 reference

7 August 2017

1 reference