(Q35778797)

10 August 2017

title

Design of triazole-stapled BCL9 α-helical peptides to target the β-catenin/B-cell CLL/lymphoma 9 (BCL9) protein-protein interaction (English)

1 reference

protein-protein interaction

10 August 2017

0 references

1 reference

Steven A Kawamoto

1

1 reference

10 August 2017

Adriana Coleska

2

1 reference

10 August 2017

Xu Ran

3

1 reference

10 August 2017

Han Yi

4

1 reference

10 August 2017

Chao-Yie Yang

5

1 reference

10 August 2017

Shaomeng Wang

6

1 reference

10 August 2017

language of work or name

English

0 references

publication date

24 January 2012

1 reference

Journal of Medicinal Chemistry

10 August 2017

published in

1 reference

10 August 2017

volume

55

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10 August 2017

issue

3

1 reference

10 August 2017

page(s)

1137-1146

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Direct inhibition of the NOTCH transcription factor complex

10 August 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Contemporary strategies for the stabilization of peptides in the alpha-helical conformation

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Synthesis and conformational analysis of a cyclic peptide obtained via i to i+4 intramolecular side-chain to side-chain azide-alkyne 1,3-dipolar cycloaddition

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Evaluation of biologically relevant short alpha-helices stabilized by a main-chain hydrogen-bond surrogate

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Single turn peptide alpha helices with exceptional stability in water

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

The growing impact of click chemistry on drug discovery

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

27 July 2018

Wnt signaling and cancer

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Deciphering rules of helix stability in peptides

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Helix propagation and N-cap propensities of the amino acids measured in alanine-based peptides in 40 volume percent trifluoroethanol

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Aromatic side-chain contribution to far-ultraviolet circular dichroism of helical peptides and its effect on measurement of helix propensities

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Analysis of the interaction of BCL9 with beta-catenin and development of fluorescence polarization and surface plasmon resonance binding assays for this interaction.

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Stereochemical effects of all-hydrocarbon tethers in i,i+4 stapled peptides.

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

An oncogenic hub: beta-catenin as a molecular target for cancer therapeutics

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Crystal structure of a beta-catenin/BCL9/Tcf4 complex

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

A stapled BID BH3 helix directly binds and activates BAX

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

A highly stable short alpha-helix constrained by a main-chain hydrogen-bond surrogate

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Activation of apoptosis in vivo by a hydrocarbon-stapled BH3 helix

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Development and optimization of a binding assay for the XIAP BIR3 domain using fluorescence polarization.

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Synthesis of alpha-amino acids via asymmetric phase transfer-catalyzed alkylation of achiral nickel(II) complexes of glycine-derived Schiff bases.

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3286869

Reactivation of the p53 tumor suppressor pathway by a stapled p53 peptide

25 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22196480

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Introduction of all-hydrocarbon i,i+3 staples into alpha-helices via ring-closing olefin metathesis

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22196480

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Highly Efficient Synthesis of Covalently Cross-Linked Peptide Helices by Ring-Closing Metathesis

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22196480

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JM201125D

1 reference

10 August 2017

1 reference

10 August 2017

1 reference