(Q35858434)

10 August 2017

A Bead-Based Proximity Assay for BRD4 Ligand Discovery (English)

1 reference

10 August 2017

Justin M Roberts

1

1 reference

PMC publication ID

4725578

10 August 2017

James E Bradner

series ordinal

2

1 reference

10 August 2017

2 December 2015

1 reference

Current protocols in chemical biology

10 August 2017

1 reference

10 August 2017

7

1 reference

10 August 2017

4

1 reference

10 August 2017

263-278

1 reference

Structure-guided DOT1L probe optimization by label-free ligand displacement

10 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Biased multicomponent reactions to develop novel bromodomain inhibitors.

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Targeting bromodomains: epigenetic readers of lysine acetylation

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Affinity map of bromodomain protein 4 (BRD4) interactions with the histone H4 tail and the small molecule inhibitor JQ1.

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Discovery and characterization of super-enhancer-associated dependencies in diffuse large B cell lymphoma.

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Small-molecule inhibition of BRDT for male contraception

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Pathogenesis of NUT midline carcinoma

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

BET bromodomain inhibition as a therapeutic strategy to target c-Myc

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

RNAi screen identifies Brd4 as a therapeutic target in acute myeloid leukaemia

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Redox cycling compounds generate H2O2 in HTS buffers containing strong reducing reagents--real hits or promiscuous artifacts?

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Selective inhibition of BET bromodomains

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

The use of AlphaScreen technology in HTS: current status

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

New substructure filters for removal of pan assay interference compounds (PAINS) from screening libraries and for their exclusion in bioassays

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

A homogeneous method for investigation of methylation-dependent protein-protein interactions in epigenetics

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Brd4 coactivates transcriptional activation of NF-kappaB via specific binding to acetylated RelA

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Recruitment of P-TEFb for stimulation of transcriptional elongation by the bromodomain protein Brd4

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Effect of detergent on "promiscuous" inhibitors

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

The double bromodomain protein Brd4 binds to acetylated chromatin during interphase and mitosis

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Luminescent oxygen channeling immunoassay: measurement of particle binding kinetics by chemiluminescence.

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4725578

Genome-wide localization of small molecules

11 July 2018

1 reference

https://api.crossref.org/works/10.1002%2F9780470559277.CH150024

Dual kinase-bromodomain inhibitors for rationally designed polypharmacology

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2F9780470559277.CH150024

Bromodomain-peptide displacement assays for interactome mapping and inhibitor discovery

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2F9780470559277.CH150024

Bromodomain: an acetyl-lysine binding domain

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2F9780470559277.CH150024

Luminescent oxygen channeling assay (LOCI): sensitive, broadly applicable homogeneous immunoassay method

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/26629616

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1002/9780470559277.CH150024

1 reference

10 August 2017

1 reference

PMC publication ID

4725578

10 August 2017

PubMed publication ID

26629616

1 reference

PMC publication ID

4725578