(Q36320975)

13 August 2017

Identification of potential inhibitors based on compound proposal contest: Tyrosine-protein kinase Yes as a target (English)

1 reference

13 August 2017

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

Y-h. Taguchi

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

Keisuke Yanagisawa

18

1 reference

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7 June 2020

Philip Prathipati

24

1 reference

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7 June 2020

Kenji Mizuguchi

27

1 reference

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7 June 2020

Masakazu Sekijima

31

1 reference

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7 June 2020

author name string

Shuntaro Chiba

1

1 reference

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7 June 2020

Kazuyoshi Ikeda

2

1 reference

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7 June 2020

Mitsuo Iwadate

6

1 reference

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7 June 2020

Hideaki Umeyama

7

1 reference

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7 June 2020

Kun-Yi Hsin

8

1 reference

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7 June 2020

Hiroaki Kitano

9

1 reference

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7 June 2020

Kazuki Yamamoto

10

1 reference

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7 June 2020

Nobuyoshi Sugaya

11

1 reference

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7 June 2020

Koya Kato

12

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7 June 2020

Tatsuya Okuno

13

1 reference

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7 June 2020

George Chikenji

14

1 reference

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7 June 2020

Masahiro Mochizuki

15

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7 June 2020

Nobuaki Yasuo

16

1 reference

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7 June 2020

Ryunosuke Yoshino

17

1 reference

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7 June 2020

Tomohiro Ban

19

1 reference

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7 June 2020

Reiji Teramoto

20

1 reference

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7 June 2020

Chandrasekaran Ramakrishnan

21

1 reference

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7 June 2020

A Mary Thangakani

22

1 reference

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7 June 2020

D Velmurugan

23

1 reference

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7 June 2020

Junichi Ito

25

1 reference

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7 June 2020

Yuko Tsuchiya

26

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

Teruki Honma

28

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

Takatsugu Hirokawa

29

1 reference

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7 June 2020

Yutaka Akiyama

30

1 reference

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7 June 2020

M Michael Gromiha

4

1 reference

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7 June 2020

language of work or name

English

0 references

publication date

26 November 2015

1 reference

13 August 2017

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

volume

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

page(s)

17209

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json

Creative Commons Attribution 4.0 International

7 June 2020

copyright license

start time

26 November 2015

1 reference

April 2022 Public Data File from Crossref

copyright status

copyrighted

0 references

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Loss-of-function screen in rhabdomyosarcoma identifies CRKL-YES as a critical signal for tumor growth

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Highly specific, bisubstrate-competitive Src inhibitors from DNA-templated macrocycles

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Computational screening for active compounds targeting protein sequences: methodology and experimental validation

30 September 2017

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Collation and data-mining of literature bioactivity data for drug discovery

30 September 2017

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A method to enhance the hit ratio by a combination of structure-based drug screening and ligand-based screening.

30 September 2017

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KX-01, a novel Src kinase inhibitor directed toward the peptide substrate site, synergizes with tamoxifen in estrogen receptor α positive breast cancer

30 September 2017

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The cost of drug development: a systematic review

30 September 2017

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DrugBank 3.0: a comprehensive resource for 'omics' research on drugs

30 September 2017

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PubChem as a public resource for drug discovery

30 September 2017

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Analysis and comparison of 2D fingerprints: insights into database screening performance using eight fingerprint methods

30 September 2017

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How to improve R&D productivity: the pharmaceutical industry's grand challenge

30 September 2017

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Therapeutic strategies underpinning the development of novel techniques for the treatment of HIV infection.

30 September 2017

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Comparison of ligand- and structure-based virtual screening on the DUD data set.

30 September 2017

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30 September 2017

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30 September 2017

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30 September 2017

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30 September 2017

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30 September 2017

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The Src Family Kinase c-Yes Is Required for Maturation of West Nile Virus Particles

30 September 2017

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The crystal structure of a c-Src complex in an active conformation suggests possible steps in c-Src activation

30 September 2017

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Insights into saquinavir resistance in the G48V HIV-1 protease: quantum calculations and molecular dynamic simulations

30 September 2017

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The many roles of computation in drug discovery

30 September 2017

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30 September 2017

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Reoptimization of MDL keys for use in drug discovery

30 September 2017

1 reference

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Approaches to the description and prediction of the binding affinity of small-molecule ligands to macromolecular receptors

30 September 2017

1 reference

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Prediction of drug solubility from structure

30 September 2017

1 reference

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SU6656, a selective src family kinase inhibitor, used to probe growth factor signaling

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Comparative protein structure modeling of genes and genomes

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Dissecting cellular processes using small molecules: identification of colchicine-like, taxol-like and other small molecules that perturb mitosis

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

30 September 2017

The Protein Data Bank

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Crystal structures of c-Src reveal features of its autoinhibitory mechanism

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Comparative protein modeling by satisfaction of spatial restraints

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Three-dimensional structure of the tyrosine kinase c-Src

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Deep neural nets as a method for quantitative structure-activity relationships

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Computational approaches to molecular recognition.

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Ligand efficiency indices for an effective mapping of chemico-biological space: the concept of an atlas-like representation.

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Cheminformatic tools for medicinal chemists.

22 September 2018

1 reference

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LigMatch: a multiple structure-based ligand matching method for 3D virtual screening.

22 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Bioinformatics based Ligand-Docking and in-silico screening.

22 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

Random forest: a classification and regression tool for compound classification and QSAR modeling

22 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4660442

An automatic homology modeling method consisting of database searches and simulated annealing

22 September 2018

1 reference

Crossref

https://api.crossref.org/works/10.1038%2FSREP17209

Identification of a calcium channel modulator using a high throughput yeast two-hybrid screen

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/26607293

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Prediction of drug absorption using multivariate statistics

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/26607293

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Random Forests

1 reference

Astrophysics Data System

15 December 2022

https://ui.adsabs.harvard.edu/abs/2001MachL..45....5B/citations

Identifiers

DOI

10.1038/SREP17209

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

0 references

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

PubMed publication ID

26607293

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26607293%20AND%20SRC:MED&resulttype=core&format=json