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Keynote review: allosterism in membrane receptors
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scholarly article
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
review article
1 reference
stated in
Europe PubMed Central
title
Keynote review: allosterism in membrane receptors
(English)
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
author name string
Zhan-Guo Gao
series ordinal
1
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
Kenneth A Jacobson
series ordinal
2
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
publication date
1 March 2006
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
published in
Drug Discovery Today
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
volume
11
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
issue
5-6
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
page(s)
191-202
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
cites work
ON THE NATURE OF ALLOSTERIC TRANSITIONS: A PLAUSIBLE MODEL
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7 January 2021
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Allosteric binding sites on cell-surface receptors: novel targets for drug discovery
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Allosteric mechanisms of signal transduction
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Crossref
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7 January 2021
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On the cooperativity of biological membranes
1 reference
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Crossref
reference URL
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7 January 2021
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GABAA receptor channels
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7 January 2021
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Galantamine: use in Alzheimer's disease and related disorders
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Cinacalcet hydrochloride (Sensipar).
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Cinacalcet HCl, an oral calcimimetic agent for the treatment of secondary hyperparathyroidism in hemodialysis and peritoneal dialysis: a randomized, double-blind, multicenter study
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Crystal structure of rhodopsin: A G protein-coupled receptor
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7 January 2021
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Allosteric functioning of dimeric class C G-protein-coupled receptors.
1 reference
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7 January 2021
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G-protein-coupled receptor oligomerization and its potential for drug discovery
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7 January 2021
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Monomeric G-protein-coupled receptor as a functional unit
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7 January 2021
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Receptor activity-independent recruitment of betaarrestin2 reveals specific signalling modes
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7 January 2021
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Emerging role of homo- and heterodimerization in G-protein-coupled receptor biosynthesis and maturation
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7 January 2021
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Activation mechanism of the heterodimeric GABA(B) receptor
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7 January 2021
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An amino-acid taste receptor
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7 January 2021
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Allosterism at muscarinic receptors: ligands and mechanisms
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7 January 2021
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Allosteric modulation of the adenosine family of receptors
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7 January 2021
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Allosteric modulation of dopamine receptors
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7 January 2021
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Mechanisms of peptide and nonpeptide ligand binding to Class B G-protein-coupled receptors
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7 January 2021
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Allosteric modulation of G protein-coupled receptors: perspectives and recent developments
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7 January 2021
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Using a radioalloster to test predictions of the cooperativity model for gallamine binding to the allosteric site of muscarinic acetylcholine M(2) receptors
1 reference
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Crossref
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https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
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Modeling the functional effects of allosteric modulators at pharmacological receptors: an extension of the two-state model of receptor activation.
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Crossref
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7 January 2021
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Allosteric modulation of the cannabinoid CB1 receptor
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Crossref
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https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Analysis of allosterism in functional assays
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Crossref
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7 January 2021
based on heuristic
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Allosteric modulation of the adenosine A(1) receptor. Synthesis and biological evaluation of novel 2-amino-3-benzoylthiophenes as allosteric enhancers of agonist binding.
1 reference
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7 January 2021
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2-Amino-3-aroyl-4,5-alkylthiophenes: agonist allosteric enhancers at human A(1) adenosine receptors
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7 January 2021
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Spinal noradrenergic activation mediates allodynia reduction from an allosteric adenosine modulator in a rat model of neuropathic pain
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7 January 2021
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Allosteric adenosine receptor modulation reduces hypersensitivity following peripheral inflammation by a central mechanism
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7 January 2021
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Allosteric enhancers of A1 adenosine receptors increase receptor-G protein coupling and counteract Guanine nucleotide effects on agonist binding
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Crossref
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7 January 2021
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Investigation of the Interaction of a Putative Allosteric Modulator,N-(2,3-Diphenyl-1,2,4-thiadiazole-5-(2H)-ylidene) Methanamine Hydrobromide (SCH-202676), with M1Muscarinic Acetylcholine Receptors
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7 January 2021
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Synthesis and biological evaluation of a new series of 2,3,5-substituted [1,2,4]-thiadiazoles as modulators of adenosine A1 receptors and their molecular mechanism of action
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7 January 2021
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Allosteric modulation of A2A adenosine receptors by amiloride analogues and sodium ions
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7 January 2021
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Selective allosteric enhancement of agonist binding and function at human A3 adenosine receptors by a series of imidazoquinoline derivatives
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
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Identification of Essential Residues Involved in the Allosteric Modulation of the Human A3Adenosine Receptor
1 reference
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Crossref
reference URL
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7 January 2021
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Inhibition of the actions of carbachol and DFP on guinea pig isolated atria by alkane-bis-ammonium compounds
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
The inhibitory effect of gallamine on muscarinic receptors
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Interactions of orthosteric and allosteric ligands with [3H]dimethyl-W84 at the common allosteric site of muscarinic M2 receptors
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Muscarinic allosteric enhancers of ligand binding: pivotal pharmacophoric elements in hexamethonio-type agents
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Discovery of an ectopic activation site on the M(1) muscarinic receptor
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Probing the molecular mechanism of interaction between 4-n-butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the muscarinic M(1) receptor: direct pharmacological evidence that AC-42 is an allosteric agonist
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
N-desmethylclozapine, an allosteric agonist at muscarinic 1 receptor, potentiates N-methyl- d -aspartate receptor activity
1 reference
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Crossref
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https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Fluorescent pirenzepine derivatives as potential bitopic ligands of the human M1 muscarinic receptor
1 reference
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Crossref
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https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Analogs of WIN 62,577 define a second allosteric site on muscarinic receptors
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Thiochrome enhances acetylcholine affinity at muscarinic M4 receptors: receptor subtype selectivity via cooperativity rather than affinity
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Atypical muscarinic allosteric modulation: cooperativity between modulators and their atypical binding topology in muscarinic M2 and M2/M5 chimeric receptors
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Allosteric binding sites on muscarinic acetylcholine receptors
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Design and synthesis of photoaffinity-labeling ligands of the L-prolyl-L-leucylglycinamide binding site involved in the allosteric modulation of the dopamine receptor
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
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Nonpeptide and peptide growth hormone secretagogues act both as ghrelin receptor agonist and as positive or negative allosteric modulators of ghrelin signaling
1 reference
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Crossref
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https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
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Chemokines: integrators of pain and inflammation
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7 January 2021
based on heuristic
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Identification of allosteric peptide agonists of CXCR4.
1 reference
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7 January 2021
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Noncompetitive allosteric inhibitors of the inflammatory chemokine receptors CXCR1 and CXCR2: prevention of reperfusion injury.
1 reference
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Crossref
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7 January 2021
based on heuristic
inferred from DOI database lookup
The CCR5 receptor-based mechanism of action of 873140, a potent allosteric noncompetitive HIV entry inhibitor
1 reference
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7 January 2021
based on heuristic
inferred from DOI database lookup
Allosteric alpha 1-adrenoreceptor antagonism by the conopeptide rho-TIA.
1 reference
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Crossref
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7 January 2021
based on heuristic
inferred from DOI database lookup
Positive allosteric modulator of the human 5-HT2C receptor
1 reference
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7 January 2021
based on heuristic
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Antagonists and the purinergic nerve hypothesis: 2, 2'-pyridylisatogen tosylate (PIT), an allosteric modulator of P2Y receptors. A retrospective on a quarter century of progress
1 reference
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7 January 2021
based on heuristic
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2,2'-Pyridylisatogen tosylate antagonizes P2Y1 receptor signaling without affecting nucleotide binding
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
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inferred from DOI database lookup
The oxytocin receptor system: structure, function, and regulation
1 reference
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https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Oleamide is a selective endogenous agonist of rat and human CB1 cannabinoid receptors
1 reference
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Crossref
reference URL
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7 January 2021
based on heuristic
inferred from DOI database lookup
Mechanism of corticotropin-releasing factor type I receptor regulation by nonpeptide antagonists
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Localization of agonist- and antagonist-binding domains of human corticotropin-releasing factor receptors
1 reference
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Crossref
reference URL
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7 January 2021
based on heuristic
inferred from DOI database lookup
Characterization of a novel, non-peptidyl antagonist of the human glucagon receptor
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Discovery of a non-peptide small molecule that selectively mimics the biological actions of calcitonin
1 reference
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Crossref
reference URL
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7 January 2021
based on heuristic
inferred from DOI database lookup
Effects of the high-affinity corticotropin-releasing hormone receptor 1 antagonist R121919 in major depression: the first 20 patients treated
1 reference
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Crossref
reference URL
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7 January 2021
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Calcitonin gene-related peptide receptor antagonist BIBN 4096 BS for the acute treatment of migraine
1 reference
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Crossref
reference URL
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7 January 2021
based on heuristic
inferred from DOI database lookup
Effects of a novel glucagon receptor antagonist (Bay 27-9955) on glucagon-stimulated glucose production in humans
1 reference
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Crossref
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https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Molecular mechanisms of GABA(B) receptor activation: new insights from the mechanism of action of CGP7930, a positive allosteric modulator.
1 reference
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Crossref
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7 January 2021
based on heuristic
inferred from DOI database lookup
BAY36-7620: a potent non-competitive mGlu1 receptor antagonist with inverse agonist activity
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Heptahelical domain of metabotropic glutamate receptor 5 behaves like rhodopsin-like receptors.
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
The cysteine-rich region of T1R3 determines responses to intensely sweet proteins
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Human Ca2+ receptor cysteine-rich domain. Analysis of function of mutant and chimeric receptors
1 reference
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Crossref
reference URL
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7 January 2021
based on heuristic
inferred from DOI database lookup
Subtype-selective noncompetitive modulators of metabotropic glutamate receptor subtype 1 (mGluR1).
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Positive allosteric modulators of the metabotropic glutamate receptor subtype 2 (mGluR2).
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Targeting the metabotropic glutamate receptor mGluR4 for the treatment of diseases of the central nervous system
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Discovery of positive allosteric modulators of metabotropic glutamate receptor subtype 5 (mGluR5).
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
New therapeutic frontiers for metabotropic glutamate receptors
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
2-Methyl-6-(phenylethynyl)-pyridine (MPEP), a potent, selective and systemically active mGlu5 receptor antagonist
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
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7 January 2021
based on heuristic
inferred from DOI database lookup
Positive and negative allosteric modulation of metabotropic glutamate receptors: emerging therapeutic potential
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Discovery of allosteric potentiators for the metabotropic glutamate 2 receptor: synthesis and subtype selectivity of N-(4-(2-methoxyphenoxy)phenyl)-N-(2,2,2- trifluoroethylsulfonyl)pyrid-3-ylmethylamine
1 reference
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Crossref
reference URL
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7 January 2021
based on heuristic
inferred from DOI database lookup
Phenyl-tetrazolyl acetophenones: discovery of positive allosteric potentiatiors for the metabotropic glutamate 2 receptor
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Allosteric modulation of group III metabotropic glutamate receptor 4: A potential approach to Parkinson's disease treatment
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
A family of highly selective allosteric modulators of the metabotropic glutamate receptor subtype 5.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
A novel selective allosteric modulator potentiates the activity of native metabotropic glutamate receptor subtype 5 in rat forebrain
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
A novel selective positive allosteric modulator of metabotropic glutamate receptor subtype 5 has in vivo activity and antipsychotic-like effects in rat behavioral models
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Benzazoles as allosteric potentiators of metabotropic glutamate receptor 2 (mGluR2): efficacy in an animal model for schizophrenia
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Anxiolytic effects of a novel group II metabotropic glutamate receptor agonist (LY354740) in the fear-potentiated startle paradigm in humans
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Effects of a metabotropic glutamate(2/3) receptor agonist (LY544344/LY354740) on panic anxiety induced by cholecystokinin tetrapeptide in healthy humans: preliminary results
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Calcimimetics with potent and selective activity on the parathyroid calcium receptor
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Identification of acidic residues in the extracellular loops of the seven-transmembrane domain of the human Ca2+ receptor critical for response to Ca2+ and a positive allosteric modulator
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Positive and negative allosteric modulators of the Ca2+-sensing receptor interact within overlapping but not identical binding sites in the transmembrane domain
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
L-amino acid sensing by the extracellular Ca2+-sensing receptor
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Modeling and Mutagenesis of the Binding Site of Calhex 231, a Novel Negative Allosteric Modulator of the Extracellular Ca2+-sensing Receptor
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
A region in the seven-transmembrane domain of the human Ca2+ receptor critical for response to Ca2+.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
A novel calcium-sensing receptor antagonist transiently stimulates parathyroid hormone secretion in vivo
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Sodium and potassium salt stimulation of taste receptor cells: an allosteric model
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Canine taste nerve responses to monosodium glutamate and disodium guanylate: differentiation between umami and salt components with amiloride
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Introductory remarks on umami taste
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
A novel family of mammalian taste receptors
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Allosteric receptors after 30 years
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Allosteric modulation of ligand-gated ion channels
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Modulation of P2X3 receptors by Mg2+ on rat DRG neurons in culture
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Modulation of BzATP and formalin induced nociception: attenuation by the P2X receptor antagonist, TNP-ATP and enhancement by the P2X(3) allosteric modulator, cibacron blue
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Tetramethylpyrazine inhibits ATP-activated currents in rat dorsal root ganglion neurons
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Alcohol action on membrane ion channels gated by extracellular ATP (P2X receptors).
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
An intersubunit zinc binding site in rat P2X2 receptors
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
P2X receptors: targets for novel analgesics?
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Glutamate receptor ion channels
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
The micromolar zinc-binding domain on the NMDA receptor subunit NR2B.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Adenosine triphosphate acts as both a competitive antagonist and a positive allosteric modulator at recombinant N-methyl-D-aspartate receptors
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
The benzodiazepine site of the GABAA receptor: an old target with new potential?
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Benzodiazepine actions mediated by specific gamma-aminobutyric acid(A) receptor subtypes.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
GABA-A receptor subtypes in the brain: a paradigm for CNS drug discovery?
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Synthesis and biological evaluation of 3-heterocyclyl-7,8,9,10-tetrahydro-(7,10-ethano)-1,2,4-triazolo[3,4-a]phthalazines and analogues as subtype-selective inverse agonists for the GABA(A)alpha5 benzodiazepine binding site.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Nicotinic acetylcholine receptors as drug targets
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Galantamine is an allosterically potentiating ligand of the human alpha4/beta2 nAChR
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Effect of galantamine on the human alpha7 neuronal nicotinic acetylcholine receptor, the Torpedo nicotinic acetylcholine receptor and spontaneous cholinergic synaptic activity
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Tyrosine kinases as targets for cancer therapy
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Signalling through the insulin receptor and the insulin-like growth factor-I receptor
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Structure of nerve growth factor complexed with the shared neurotrophin receptor p75
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
The yin and yang of neurotrophin action
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
p75 Co-receptors regulate ligand-dependent and ligand-independent Trk receptor activation, in part by altering Trk docking subdomains.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
The non-peptidyl fungal metabolite L-783,281 activates TRK neurotrophin receptors
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Small molecule Trk receptor agonists and other neurotrophic factor mimetics
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Ganglioside GM1 enhances induction by nerve growth factor of a putative dimer of TrkA
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
The staurosporine-like compound L-753,000 (NB-506) potentiates the neurotrophic effects of neurotrophin-3 by acting selectively at the TrkA receptor.
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Structural insights into the regulation and the activation mechanism of mammalian guanylyl cyclases
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
YC-1 activation of human soluble guanylyl cyclase has both heme-dependent and heme-independent components
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
NO-independent regulatory site on soluble guanylate cyclase
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
NO- and haem-independent activation of soluble guanylyl cyclase: molecular basis and cardiovascular implications of a new pharmacological principle
1 reference
stated in
Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS1359-6446%2805%2903689-5
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Identifiers
DOI
10.1016/S1359-6446(05)03689-5
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
PubMed ID
16580596
1 reference
stated in
Europe PubMed Central
PubMed ID
16580596
retrieved
14 August 2017
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