(Q36590244)

English

Synthesis, enantioresolution, and activity profile of chiral 6-methyl-2,4-disubstituted pyridazin-3(2H)-ones as potent N-formyl peptide receptor agonists

scientific article published on 27 April 2012

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scholarly article

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Europe PubMed Central

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1 February 2020

Synthesis, enantioresolution, and activity profile of chiral 6-methyl-2,4-disubstituted pyridazin-3(2H)-ones as potent N-formyl peptide receptor agonists (English)

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1 February 2020

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Agostino Cilibrizzi

1

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1 February 2020

Gianluca Bartolucci

3

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1 February 2020

Claudia Vergelli

10

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1 February 2020

Igor A Schepetkin

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Igor A Schepetkin

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1 February 2020

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Letizia Crocetti

4

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1 February 2020

Vittorio Dal Piaz

5

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1 February 2020

Maria Paola Giovannoni

6

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1 February 2020

Alessia Graziano

7

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1 February 2020

Liliya N Kirpotina

8

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1 February 2020

Mark T Quinn

9

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27 April 2012

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1 February 2020

Bioorganic & Medicinal Chemistry

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1 February 2020

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1 February 2020

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1 February 2020

3781-3792

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Therapeutic anti-inflammatory potential of formyl-peptide receptor agonists

1 reference

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Identification of novel small-molecule agonists for human formyl peptide receptors and pharmacophore models of their recognition.

1 reference

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International Union of Basic and Clinical Pharmacology. LXXIII. Nomenclature for the formyl peptide receptor (FPR) family

1 reference

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Formyl-peptide receptors revisited

1 reference

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Reversal of elution order during the chiral separation in high performance liquid chromatography

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1 reference

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30 September 2017

6-methyl-2,4-disubstituted pyridazin-3(2H)-ones: a novel class of small-molecule agonists for formyl peptide receptors

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Urokinase induces basophil chemotaxis through a urokinase receptor epitope that is an endogenous ligand for formyl peptide receptor-like 1 and -like 2.

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12 December 2020

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10.1016/J.BMC.2012.04.043

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1 February 2020

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1 February 2020

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1 February 2020

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