(Q37176219)

English

The importance of micelle-bound states for the bioactivities of bifunctional peptide derivatives for delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists

scientific article published on 27 September 2008

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

The importance of micelle-bound states for the bioactivities of bifunctional peptide derivatives for delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists (English)

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

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author name string

Takashi Yamamoto

1

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Padma Nair

2

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Neil E Jacobsen

3

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Peg Davis

4

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Shou-wu Ma

5

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Edita Navratilova

6

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Sharif Moye

7

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Josephine Lai

8

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Henry I Yamamura

9

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Todd W Vanderah

10

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Frank Porreca

11

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Europe PubMed Central

PMC publication ID

18 August 2017

Victor J Hruby

12

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Europe PubMed Central

PMC publication ID

18 August 2017

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publication date

27 September 2008

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Europe PubMed Central

PMC publication ID

18 August 2017

Journal of Medicinal Chemistry

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Europe PubMed Central

PMC publication ID

18 August 2017

51

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Europe PubMed Central

PMC publication ID

18 August 2017

20

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

6334-6347

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

A structure-activity relationship study and combinatorial synthetic approach of C-terminal modified bifunctional peptides that are delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Design, synthesis, and biological evaluation of novel bifunctional C-terminal-modified peptides for delta/mu opioid receptor agonists and neurokinin-1 receptor antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Secondary structure provides a template for the folding of nearby polypeptides

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Structure-activity relationships of bifunctional peptides based on overlapping pharmacophores at opioid and cholecystokinin receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Design and synthesis of novel hydrazide-linked bifunctional peptides as delta/mu opioid receptor agonists and CCK-1/CCK-2 receptor antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Virtual Computational Chemistry Laboratory – Design and Description

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Is paradoxical pain induced by sustained opioid exposure an underlying mechanism of opioid antinociceptive tolerance?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Role of NK-1 neurotransmission in opioid-induced hyperalgesia

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Glycopeptides related to beta-endorphin adopt helical amphipathic conformations in the presence of lipid bilayers.

1 reference

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6 September 2017

Neurodegenerative aspects of protein aggregation.

1 reference

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6 September 2017

Recent advances in the investigation of the bioactive conformation of peptides active at the micro-opioid receptor. conformational analysis of endomorphins

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Substance P: structure, function, and therapeutics

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Opioid receptors and their ligands

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Recent advances in selective opioid receptor agonists and antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Folding proteins in fatal ways

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Protein folding and misfolding

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Protein aggregation and aggregate toxicity: new insights into protein folding, misfolding diseases and biological evolution

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Glycopeptide-Membrane Interactions: Glycosyl Enkephalin Analogues Adopt Turn Conformations by NMR and CD in Amphipathic Media

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

NMR solution structure of the glucagon antagonist [desHis1, desPhe6, Glu9]glucagon amide in the presence of perdeuterated dodecylphosphocholine micelles

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Natural peptide analgesics: the role of solution conformation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Exendin-4 and glucagon-like-peptide-1: NMR structural comparisons in the solution and micelle-associated states

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Mechanisms of tryptophan fluorescence shifts in proteins

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Structure of outer membrane protein A transmembrane domain by NMR spectroscopy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Conformational toxicity and sporadic conformational diseases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Biological activity of fragments and analogues of the potent dimeric opioid peptide, biphalin

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

High-resolution solution structure of the EGF-like domain of heregulin-alpha

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

The peptide binding site of the substance P (NK-1) receptor localized by a photoreactive analogue of substance P: presence of a disulfide bond

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

A two-dimensional nuclear Overhauser enhancement (2D NOE) experiment for the elucidation of complete proton-proton cross-relaxation networks in biological macromolecules

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Conformation of glucagon in a lipid-water interphase by 1H nuclear magnetic resonance

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Role of membrane lipids in peptide hormone function: binding of enkephalins to micelles

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Application of phase sensitive two-dimensional correlated spectroscopy (COSY) for measurements of 1H-1H spin-spin coupling constants in proteins

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Analysis and prediction of the different types of beta-turn in proteins

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Membrane lipid phase as catalyst for peptide-receptor interactions

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

An evaluation of computational strategies for use in the determination of protein structure from distance constraints obtained by nuclear magnetic resonance.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

pH-dependent structural transitions of Alzheimer amyloid peptides

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

The chemical shift index: a fast and simple method for the assignment of protein secondary structure through NMR spectroscopy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Gradient-tailored excitation for single-quantum NMR spectroscopy of aqueous solutions

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

The solution structure of eglin c based on measurements of many NOEs and coupling constants and its comparison with X‐ray structures

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Identification of two related pentapeptides from the brain with potent opiate agonist activity

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Brownian motion in biological membranes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

6 September 2017

Protein folding and misfolding: a paradigm of self-assembly and regulation in complex biological systems

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

14 September 2017

Time-resolved fluorescence of proteins

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

14 September 2017

Conformation of [Leu 5 ]Enkephalin from X-Ray Diffraction: Features Important for Recognition at Opiate Receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

14 September 2017

Modes of peptide binding in G protein-coupled receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

27 June 2018

Structure-activity relationships of enkephalin analogs at opiate and enkephalin receptors: Correlation with analgesia

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

27 June 2018

Roles of mu, delta and kappa opioid receptors in spinal and supraspinal mediation of gastrointestinal transit effects and hot-plate analgesia in the mouse

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

27 June 2018

Role of mu and delta receptors in the supraspinal and spinal analgesic effects of [D-Pen2, D-Pen5]enkephalin in the mouse.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

27 June 2018

Opioid agonist affinity in the guinea-pig ileum and mouse vas deferens

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

27 June 2018

Solution Structures of β Peptide and Its Constituent Fragments: Relation to Amyloid Deposition

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

27 June 2018

Resolved fluorescence emission spectra of PRODAN in ethanol/buffer solvents.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

3 September 2018

Resting and evoked spinal substance P release during chronic intrathecal morphine infusion: parallels with tolerance and dependence

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

3 September 2018

Inhibition of neurokinin-1-substance P receptor and prostanoid activity prevents and reverses the development of morphine tolerance in vivo and the morphine-induced increase in CGRP expression in cultured dorsal root ganglion neurons

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

3 September 2018

Lack of self-administration and behavioural sensitisation to morphine, but not cocaine, in mice lacking NK1 receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

3 September 2018

Analysis of main chain torsion angles in proteins: prediction of NMR coupling constants for native and random coil conformations

1 reference

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3 September 2018

Measurement of guanine nucleotide-binding protein activation by A1 adenosine receptor agonists in bovine brain membranes: stimulation of guanosine-5'-O-(3-[35S]thio)triphosphate binding.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

3 September 2018

Spinal co-administration of peptide substance P antagonist increases antinociceptive effect of the opioid peptide biphalin

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2675940

3 September 2018

Sequence Dependence of Amyloid Fibril Formation: Insights from Molecular Dynamics Simulations

1 reference

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4 December 2018

Folding of apocytochrome c in lipid micelles: formation of alpha-helix precedes membrane insertion

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Structure, Dynamics, and Insertion of a Chloroplast Targeting Peptide in Mixed Micelles†

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Morphine treatment induced calcitonin gene-related peptide and substance P increases in cultured dorsal root ganglion neurons

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Conformational analysis of Met-enkephalin in both aqueous solution and in the presence of sodium dodecyl sulfate micelles using multidimensional NMR and molecular modeling

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Implicit solvent simulations of DPC micelle formation

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

2D NMR and structural model for a mitochondrial signal peptide bound to a micelle

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

An all atom force field for simulations of proteins and nucleic acids

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Nuclear magnetic resonance identification of "half-turn" and 3(10)-helix secondary structure in rabbit liver metallothionein-2

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Affinity of normorphine for its pharmacologic receptor in the naive and morphine-tolerant guinea-pig isolated ileum

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Characterization of the interaction of N-acyl-L-tryptophan benzyl ester neurokinin antagonists with the human neurokinin-1 receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Tryptophan-derived NK1 antagonists: conformationally constrained heterocyclic bioisosteres of the ester linkage

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Structure of glucagon-like peptide (7-36) amide in a dodecylphosphocholine micelle as determined by 2D NMR

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The use of dodecylphosphocholine micelles in solution NMR

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Conformational study of [Met5]enkephalin-Arg-Phe in the presence of phosphatidylserine vesicles

1 reference

https://pubmed.ncbi.nlm.nih.gov/18821747

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1021/JM800389V

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

ResearchGate publication ID

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